Melissa M. Cadelis

发表

Discovery and preliminary structure-activity relationship studies on tecomaquinone I and tectol as novel farnesyltransferase and plasmodial inhibitors.

M. Bourguet-Kondracki, B. Copp, D. Barker, 2016, Bioorganic & medicinal chemistry.

A Review of Fungal Protoilludane Sesquiterpenoid Natural Products

S. Wiles, B. Copp, M. Cadelis, 2020, Antibiotics.

Investigation of α,ω-Disubstituted Polyamine-Cholic Acid Conjugates Identifies Hyodeoxycholic and Chenodeoxycholic Scaffolds as Non-Toxic, Potent Antimicrobials

M. Bourguet-Kondracki, J. Brunel, B. Copp, 2023, Antibiotics.

Efficacy of a series of alpha-pyrone derivatives against Leishmania (L.) infantum and Trypanosoma cruzi.

G. Wynne, B. Copp, A. Tempone, 2017, European journal of medicinal chemistry.

Terrien, a metabolite made by Aspergillus terreus, has activity against Cryptococcus neoformans

S. Wiles, B. Copp, M. Cadelis, 2022, PeerJ.

Preclinical Evaluation of Discorhabdins in Antiangiogenic and Antitumor Models

Kristina M. Cook, K. Gustafson, W. Figg, 2018, Marine drugs.

Exploration of the Electrophilic Reactivity of the Cytotoxic Marine Alkaloid Discorhabdin C and Subsequent Discovery of a New Dimeric C-1/N-13-Linked Discorhabdin Natural Product

B. Copp, M. Cadelis, Cary F. C. Lam, 2020, Marine drugs.

Screening and Biological Effects of Marine Pyrroloiminoquinone Alkaloids: Potential Inhibitors of the HIF-1α/p300 Interaction.

Kristina M. Cook, K. Gustafson, D. Venzon, 2016, Journal of natural products.

Investigation of the electrophilic reactivity of the biologically active marine sesquiterpenoid onchidal and model compounds

B. Copp, Melissa M. Cadelis, 2018, Beilstein journal of organic chemistry.

Synthesis and Antibacterial Analysis of Analogues of the Marine Alkaloid Pseudoceratidine

B. Copp, D. Barker, V. Sarojini, 2020, Molecules.

Exploration of the influence of spiro-dienone moiety on biological activity of the cytotoxic marine alkaloid discorhabdin P

B. Copp, M. Cadelis, Cary F. C. Lam, 2017 .

Antimicrobial Natural Products from Plant Pathogenic Fungi

S. Wiles, B. Copp, M. Cadelis, 2023, Molecules.

Antimicrobial Metabolites against Methicillin-Resistant Staphylococcus aureus from the Endophytic Fungus Neofusicoccum australe

S. Wiles, B. Copp, Bevan Simon Weir, 2021, Molecules.

Total synthesis of panicein A2

B. Copp, D. Barker, L. Pilkington, 2015, Beilstein journal of organic chemistry.

Valorisation of the diterpene podocarpic acid - Antibiotic and antibiotic enhancing activities of polyamine conjugates.

M. Bourguet-Kondracki, B. Copp, Hana Douafer, 2022, Bioorganic & medicinal chemistry.

Total Synthesis of the Four Stereoisomers of Cyclo(l-Trp-l-Arg) Raises Uncertainty of the Structures of the Natural Products and Invalidates Their Promising Antimicrobial Activities

M. Bourguet-Kondracki, J. Brunel, B. Copp, 2022, Molecules.

Repurposing primaquine as a polyamine conjugate to become an antibiotic adjuvant.

M. Bourguet-Kondracki, J. Brunel, B. Copp, 2021, Bioorganic & medicinal chemistry.

6-Bromoindolglyoxylamido derivatives as antimicrobial agents and antibiotic enhancers.

M. Bourguet-Kondracki, J. Brunel, B. Copp, 2019, Bioorganic & medicinal chemistry.

α,ω-Diacyl-Substituted Analogues of Natural and Unnatural Polyamines: Identification of Potent Bactericides That Selectively Target Bacterial Membranes

M. Bourguet-Kondracki, J. Brunel, B. Copp, 2023, International journal of molecular sciences.

Discovery and Preliminary Structure-Activity Investigation of 3-Substituted-1H-imidazol-5-yl-1H-indoles with In Vitro Activity towards Methicillin-Resistant Staphylococcus aureus

M. Bourguet-Kondracki, J. Brunel, B. Copp, 2022, Antibiotics.

Spermine Derivatives of Indole‐3‐carboxylic Acid, Indole‐3‐acetic Acid and Indole‐3‐acrylic Acid as Gram‐Negative Antibiotic Adjuvants

M. Bourguet-Kondracki, J. Brunel, B. Copp, 2020, ChemMedChem.

Exploration of the antibiotic potentiating activity of indolglyoxylpolyamines.

M. Bourguet-Kondracki, J. Brunel, B. Copp, 2019, European journal of medicinal chemistry.

Screening of Fungi for Antimycobacterial Activity Using a Medium-Throughput Bioluminescence-Based Assay

T. Lumley, S. Wiles, B. Copp, 2021, Frontiers in Microbiology.

Antimicrobial Polyketide Metabolites from Penicillium bissettii and P. glabrum

S. Wiles, B. Copp, Bevan Simon Weir, 2021, Molecules.

Isolation of a Novel Polyketide from Neodidymelliopsis sp.

S. Wiles, B. Copp, A. Grey, 2021, Molecules.

Epipyrone A, a Broad-Spectrum Antifungal Compound Produced by Epicoccum nigrum ICMP 19927

Alex J. Lee, S. Villas-Bôas, S. Swift, 2020, Molecules.

Exploration of Bis-Cinnamido-Polyamines as Intrinsic Antimicrobial Agents and Antibiotic Enhancers

M. Bourguet-Kondracki, J. Brunel, B. Copp, 2023, Biomolecules.

Indole-3-Acetamido-Polyamines as Antimicrobial Agents and Antibiotic Adjuvants

M. Bourguet-Kondracki, J. Brunel, B. Copp, 2023, Biomolecules.

Investigation of Naphthyl–Polyamine Conjugates as Antimicrobials and Antibiotic Enhancers

M. Bourguet-Kondracki, J. Brunel, B. Copp, 2023, Antibiotics.

Structure–Activity Relationship Studies of Indolglyoxyl-Polyamine Conjugates as Antimicrobials and Antibiotic Potentiators

M. Bourguet-Kondracki, J. Brunel, B. Copp, 2023, Pharmaceuticals.

Structure-activity relationship studies on thiaplidiaquinones A and B as novel inhibitors of Plasmodium falciparum and farnesyltransferase.

M. Bourguet-Kondracki, J. Brunel, B. Copp, 2017, Bioorganic & Medicinal Chemistry.

A Revised Structure and Assigned Absolute Configuration of Theissenolactone A

S. Wiles, B. Copp, Bevan Simon Weir, 2020, Molecules.