Phaedra Geer

Discovery of Nanomolar Melanocortin-3 Receptor (MC3R)-Selective Small Molecule Pyrrolidine Bis-Cyclic Guanidine Agonist Compounds Via a High-Throughput "Unbiased" Screening Campaign.

Radleigh G. Santos, M. Giulianotti, R. Houghten, 2021, Journal of medicinal chemistry.

Synthesis and biological evaluations of novel endomorphin analogues containing α-hydroxy-β-phenylalanine (AHPBA) displaying mixed μ/δ opioid receptor agonist and δ opioid receptor antagonist activities.

Austin B. Yongye, Radleigh G. Santos, M. Giulianotti, 2015, European journal of medicinal chemistry.

Identification of Tetrapeptides from a Mixture Based Positional Scanning Library That Can Restore nM Full Agonist Function of the L106P, I69T, I102S, A219V, C271Y, and C271R Human Melanocortin-4 Polymorphic Receptors (hMC4Rs)

Clemencia Pinilla, Michael A. Walters, Richard A. Houghten, 2014, Journal of medicinal chemistry.

Discovery of Mixed Pharmacology Melanocortin-3 Agonists and Melanocortin-4 Receptor Tetrapeptide Antagonist Compounds (TACOs) Based on the Sequence Ac-Xaa1-Arg-(pI)DPhe-Xaa4-NH2.

Radleigh G. Santos, M. Giulianotti, R. Houghten, 2017, Journal of medicinal chemistry.

Dissociation of Antimicrobial and Hemolytic Activities of Gramicidin S through N‐Methylation Modification

Austin B. Yongye, R. Houghten, Nina Bionda, 2013, ChemMedChem.