I. Domračeva

发表

Peptide/β-Peptoid Hybrids with Ultrashort PEG-Like Moieties: Effects on Hydrophobicity, Antibacterial Activity and Hemolytic Properties

H. Franzyk, F. Björkling, O. Pugovics, 2021, International journal of molecular sciences.

Development of oxathiino[6,5-b]pyridine 2,2-dioxide derivatives as selective inhibitors of tumor-related carbonic anhydrases IX and XII.

C. Supuran, A. Nocentini, A. Grandane, 2020, European journal of medicinal chemistry.

Plasmepsin inhibitory activity and structure-guided optimization of a potent hydroxyethylamine-based antimalarial hit.

A. Jirgensons, M. Blackman, K. Tārs, 2014, ACS medicinal chemistry letters.

Design, synthesis, and biological evaluation of novel derivatives of dithiodiglycolic acid prepared via oxidative coupling of thiols

M. Pešić, R. Žalubovskis, M. Krasavin, 2019, Journal of enzyme inhibition and medicinal chemistry.

Fragment-Based Discovery of 2-Aminoquinazolin-4(3H)-ones As Novel Class Nonpeptidomimetic Inhibitors of the Plasmepsins I, II, and IV.

A. Jirgensons, M. Blackman, K. Tārs, 2016, Journal of medicinal chemistry.

Alternating Cationic‐Hydrophobic Peptide/Peptoid Hybrids: Influence of Hydrophobicity on Antibacterial Activity and Cell Selectivity

P. Hansen, H. Franzyk, F. Björkling, 2020, ChemMedChem.

Atropo/Tropo Flexibility: A Tool for Design and Synthesis of Self-Adaptable Inhibitors of Carbonic Anhydrases and Their Antiproliferative Effect.

C. Supuran, A. Kazaks, A. Nocentini, 2023, Journal of medicinal chemistry.

Novel electrophilic amides amenable by the Ugi reaction perturb thioredoxin system via thioredoxin reductase 1 (TrxR1) inhibition: Identification of DVD-445 as a new lead compound for anticancer therapy.

M. Pešić, S. Glišić, V. Sharoyko, 2019, European journal of medicinal chemistry.

Base-Free Catalytic Wittig-/Cross-Coupling Reaction Sequence as Short Synthetic Strategy for the Preparation of Highly Functionalized Arylbenzoxepinones

T. Werner, A. Grandane, R. Žalubovskis, 2021, Synthesis.

Peptide/β-Peptoid Hybrids with Activity against Vancomycin-Resistant Enterococci: Influence of Hydrophobicity and Structural Features on Antibacterial and Hemolytic Properties

M. Vestergaard, H. Ingmer, H. Franzyk, 2021, International journal of molecular sciences.

Structure-activity study of oncocin: On-resin guanidinylation and incorporation of homoarginine, 4-hydroxyproline or 4,4-difluoroproline residues.

Ashif Y. Shaikh, D. Żabicka, A. Kreicberga, 2023, Bioorganic chemistry.

Synthesis and study of new 5-substituted 1-acetyl-4-phenyl-3-pyrrolin-2-ones as potential antitumor agents

A. Leonchiks, S. Belyakov, M. Petrova, 2018, Chemistry of Heterocyclic Compounds.