Eduard Sergienko

发表

Table 3, Probe and Analog Submissions to MLSMR (Evotec) for P. falciparum G-6PDH antagonists

Stefan Vasile, Eigo Suyama, Michael Vicchiarelli, 2013 .

Figure 4, Screening and Hit advancement flowchart

Tudor I. Oprea, Bruce S. Edwards, Larry A. Sklar, 2013 .

Scheme 1, Proposed Synthesis of MLS-0092727

Thomas D.Y. Chung, Eduard Sergienko, Derek Stonich, 2010 .

Figure 1, Key SAR for our first library

Darren Finlay, Kristiina Vuori, Robert Ardecky, 2011 .

Table 2, Submission information on Probe and analogs

Thomas D.Y. Chung, Eduard Sergienko, Derek Stonich, 2010 .

Table 4, Probe and Analog Submissions to MLSMR (BioFocus DPI) for Gli-Sufu Antagonist ML340

Santhi Ganji, Ian Pass, Robert Ardecky, 2014 .

Table 4, Summary of the existing probes and the corresponding commercial vendors

Thomas D.Y. Chung, Eduard Sergienko, Derek Stonich, 2010 .

[Table, Primary Screen Protocol].

Susanne Heynen-Genel, Michelle Sauer, Shenghua Shi, 2010 .

Table 1, Listing of all Assays and AIDs for this project

Susanne Heynen-Genel, Shenghua Shi, Thomas D.Y. Chung, 2010 .

Scheme 1, Synthesis of ML307, conditions

Santhi Ganji, Ian Pass, Robert Ardecky, 2014 .

Table 2, Structures and data for the lead triazoles

Thomas D.Y. Chung, Eduard Sergienko, Derek Stonich, 2010 .

Table 5A, Submission information on Probe 1: CID2286812 and analogs

Susanne Heynen-Genel, Michelle Sauer, Shenghua Shi, 2010 .

Table 8, Comparative data for probe specificity

Mahesh Peddibhotla, Thomas D.Y. Chung, Eduard Sergienko, 2010 .

Table 4, Probe and Analog Submissions to MLSMR (BioFocus DPI) for UBC13 Inhibitors

Santhi Ganji, Ian Pass, Robert Ardecky, 2013 .

Table 3, Pharmacologic Properties of MLS-01014097, MLS-0107074

Layton H. Smith, Thomas D.Y. Chung, Eduard Sergienko, 2010 .

Table 5, Probe and Analog Submissions to the MLMR (BioFocus DPI)

Susanne Heynen-Genel, Thomas D.Y. Chung, Palak Gosalia, 2010 .

Table 5, Submission of Probe and analogs

Darren Finlay, Kristiina Vuori, Robert Ardecky, 2011 .

Table 1, SAR results generated using analogue-by-catalogue (ABC)

Layton H. Smith, Thomas D.Y. Chung, Eduard Sergienko, 2010 .

Table 3, CID 56639556 [ML307] MLS-0471611

Santhi Ganji, Ian Pass, Robert Ardecky, 2014 .

[Figure], Critical Path Flowchart for KOR Antagonist Project

Susanne Heynen-Genel, Thomas D.Y. Chung, Palak Gosalia, 2010 .

Scheme 1, Synthesis of ML304

Stefan Vasile, Eigo Suyama, Michael Vicchiarelli, 2013 .

Scheme 1, Synthesis of ML260

Jiwen Zou, Santhi Ganji, Ian Pass, 2013 .

Table 4, Submission of Probe and 5 analogs to the MLSMR

Stefan Vasile, Thomas D.Y. Chung, Eduard Sergienko, 2010 .

Table 5, Submission of Probe and 6 analogs to the MLSMR (MLSMR)

Mahesh Peddibhotla, Thomas D.Y. Chung, Eduard Sergienko, 2010 .

Table 5B, Submission information on Probe#2: CID1542103 and analogs

Susanne Heynen-Genel, Michelle Sauer, Shenghua Shi, 2010 .

[Table, A tabular presentation summarizing known probe properties (computed properties, must match from PubChem)].

Susanne Heynen-Genel, Michael Vicchiarelli, Shenghua Shi, 2011 .

[Table, Image Acquisition and Analysis].

Susanne Heynen-Genel, Michelle Sauer, Shenghua Shi, 2011 .

Figure 2, Key SAR for our second library

Darren Finlay, Kristiina Vuori, Robert Ardecky, 2011 .

Table 8, Comparative Downstream assays by Assay Provider for CID9581011

Susanne Heynen-Genel, Michelle Sauer, Shenghua Shi, 2011 .

Figure 5, Screening results and Hit validation

John C. Reed, Santhi Ganji, Ian Pass, 2011 .

Table 8, Comparison of prior art and current probe

Susanne Heynen-Genel, Thomas D.Y. Chung, Palak Gosalia, 2010 .

Scheme 1, Synthetic scheme

Thomas D.Y. Chung, Eduard Sergienko, Derek Stonich, 2010 .

Table 9, Comparative summary of two current probes CID5236771 & CID44601470 to literature examples

Susanne Heynen-Genel, Thomas D.Y. Chung, Palak Gosalia, 2010 .

Table 4, Submission information on Probe 1 and analogs

Thomas D.Y. Chung, Michael Hedrick, Eduard Sergienko, 2010 .

Table 3, Probe and Analog Submissions to MLSMR (BioFocus DPI) for APJ Antagonists

Stefan Vasile, Eigo Suyama, Michael Vicchiarelli, 2013 .

Scheme 1, Synthesis of ML276

Stefan Vasile, Eigo Suyama, Michael Vicchiarelli, 2013 .

Table 1, PubChem Assay Summaries for Probe project

Darren Finlay, Robert Ardecky, Thomas D.Y. Chung, 2010 .

Selective HePTP Inhibitors: Probe 1

Thomas D.Y. Chung, Eduard Sergienko, Russell Dahl, 2010 .

Figure 2, The GPR35 Antagonist Probe Flowchart summarizes the compound triage and decision tree for advancement of the compounds

Susanne Heynen-Genel, Michelle Sauer, Shenghua Shi, 2010 .

Table 5, Exploration of the left hand side of the lead structure

Thomas D.Y. Chung, Eduard Sergienko, Derek Stonich, 2010 .