D. Bonnet‐Delpon

发表

Bioorganic and Medicinal Chemistry of Fluorine

D. Bonnet-Delpon, J. Bégué, Jean-Pierre Bégué, 2008 .

Improved Ritter reaction with CF3-containing oxirane for an access to central units of protease inhibitors

B. Crousse, D. Bonnet-Delpon, M. Santos, 2009 .

Novel fluorinated pseudopeptides as proteasome inhibitors.

N. Basse, M. Reboud-Ravaux, X. Maréchal, 2009, Bioorganic & medicinal chemistry letters.

Recent advances (1995–2005) in fluorinated pharmaceuticals based on natural products ☆

D. Bonnet-Delpon, J. Bégué, D. Bonnet‐Delpon, 2006 .

Mild and Selective Oxidation of Sulfur Compounds in Trifluoroethanol: Diphenyl Disulfide and Methyl Phenyl Sulfoxide

V. Kesavan, B. Crousse, D. Bonnet-Delpon, 2003 .

Role of Hexafluoro‐2‐propanol in Selective Oxidation of Sulfide to Sulfoxide: Efficient Preparation of Glycosyl Sulfoxides

Yongming Zhang, D. Bonnet-Delpon, J. Bégué, 1998 .

Stereoselective Synthesis of Peptidyl Trifluoromethyl Alcohols and Ketones: Inhibitory Potency Against Human Leucocyte Elastase, Cathepsin G, Porcine Pancreatic Elastase and HIV‐1 Protease

D. Bonnet-Delpon, J. Bégué, A. Amour, 1998, The Journal of pharmacy and pharmacology.

Stereoselective synthesis and inhibitor properties towards human leucocyte elastase of chiral β-peptidyl trifluoromethyl alcohols.

D. Bonnet-Delpon, J. Bégué, A. Amour, 1994 .

Preparation of trifluoromethyl ketones and related fluorinated ketones

D. Bonnet-Delpon, J. Bégué, D. Bonnet‐Delpon, 1991 .

[Fluorine, an essential element for medicinal chemistry].

D. Bonnet-Delpon, D. Bonnet‐Delpon, 2008, Annales pharmaceutiques francaises.

A convenient synthesis of fluoroalkyl and fluoroaryl glycosides using Mitsunobu conditions

D. Bonnet-Delpon, J. Bégué, D. Gueyrard, 1999 .

The effect of 10 alpha-trifluoromethylhydroartemisinin on Plasmodium berghei infection and its toxicity in experimental animals.

L. Cong, D. Bonnet-Delpon, J. Bégué, 2002, Transactions of the Royal Society of Tropical Medicine and Hygiene.

Short and efficient preparation of trifluoromethyl vinyl sulphides

D. Bonnet-Delpon, J. Bégué, Abderrahim M'bida, 1993 .

The Wittig reaction of perfluoro acid derivatives: access to fluorinated enol ethers, enamines, and ketones

D. Bonnet-Delpon, J. Bégué, Sheng-Wen Wu, 1992 .

A SELECTIVE CONVERSION OF SULFIDE TO SULFOXIDE IN HEXAFLUORO-2-PROPANOL

D. Bonnet-Delpon, J. Bégué, K. S. Ravikumar, 1998 .

1-Trifluoromethyl epoxy ethers. Effect of hexafluoro-2-propanol on reactions with secondary aromatic amines: synthesis of 3-trifluoromethyl indole derivatives.

D. Bonnet-Delpon, J. Bégué, I. Rodrigues, 2001, The Journal of organic chemistry.

Fluoro alcohol as reaction medium: one-pot synthesis of β-hydroxy sulfoxides from epoxides

V. Kesavan, D. Bonnet-Delpon, J. Bégué, 2000 .

Biological Impacts of Fluorination

D. Bonnet-Delpon, J. Bégué, D. Bonnet‐Delpon, 2008 .

A concise synthesis of functionalised gem-difluoroalkenes, via the addition of organolithium reagents to α-trifluoromethylstyrene

D. Bonnet-Delpon, J. Bégué, M. Rock, 1995 .

The addition of N-lithiated amines to 1,1,1-trifluoromethylstyrene, a concise synthesis of 3-gem-difluoro-2-phenyl allylic amines

D. Bonnet-Delpon, J. Bégué, M. Rock, 1995 .

Addition of organolithium reagents to α-(trifluoromethyl)styrene: concise synthesis of functionalised gem-difluoroalkenes

D. Bonnet-Delpon, J. Bégué, M. Rock, 1996 .

Facile syntheses of gem-difluoroalkenes from chlorodifluoromethylketones

R. Wilkes, J. Percy, D. Bonnet-Delpon, 1995 .

TRIFLUOROMETHYLALKENES IN CYCLOADDITION REACTIONS

D. Bonnet-Delpon, J. Bégué, T. Lequeux, 1996 .

Synthesis of allylic trifluoromethyl alcohols from 1-trifluoromethyl-epoxy ethers

J. Bégué, N. Fischer‐Durand, A. Kornilov, 1996 .

Transition metal-catalyzed cyclopropanation of alkenes in fluorinated alcohols

B. Crousse, D. Bonnet-Delpon, Kaouther Azzouzi-Zriba, 2011 .

Urea‐Hydrogen Peroxide/Hexafluoro‐2‐propanol: An Efficient System for a Catalytic Epoxidation Reaction without a Metal

J. Legros, B. Crousse, D. Bonnet-Delpon, 2002 .

Methyltrioxorhenium-catalysed epoxidation of alkenes: enhancement of reactivity in hexafluoro-2-propanol

D. Bonnet-Delpon, J. Bégué, J. Iskra, 2002 .

Transport of fluoroalkyl dihydroartemisinin derivatives across rat intestinal tissue

F. Bigucci, G. Ponchel, M. Besnard, 2008, The Journal of pharmacy and pharmacology.

Solvent‐Promoted and ‐Controlled Aza‐Michael Reaction with Aromatic Amines.

B. Crousse, Kavita De, Julien Legros, 2010 .

Solvent-promoted and -controlled aza-Michael reaction with aromatic amines.

J. Legros, B. Crousse, D. Bonnet-Delpon, 2009, The Journal of organic chemistry.

Comparative study of the ring opening of 1-CF3-epoxy ethers mediated by Brönsted acids and hexafluoro-2-propanol

D. Bonnet-Delpon, J. Bégué, J. Iskra, 2005 .

Direct access to CF3-propargyl amines and conversion to difluoromethyl imines

B. Crousse, D. Bonnet-Delpon, Guillaume Magueur, 2005 .

Diastereoselective Synthesis of the Nonracemic Methyl syn-(3-Fluoroalkyl)isoserinates

D. Bonnet-Delpon, J. Bégué, A. Abouabdellah, 1997 .

Cobalt-Induced C-N and C-C Bond Formation via Metal-Stabilized alpha-CF(3) Carbenium Ion.

B. Malézieux, J. Bégué, H. Amouri, 2000, Organic letters.

Design, Synthesis and Antimalarial Activity of Trifluoromethylartemisinin–Mefloquine Dual Molecules

P. Grellier, D. Bonnet-Delpon, J. Bégué, 2005, Chembiochem : a European journal of chemical biology.

The chemistry of trifluoromethyl imines and related acetals derived from fluoral.

J. Legros, B. Crousse, D. Bonnet-Delpon, 2005, Chemical Society reviews.

Effects of Fluorine Substitution on Biological Properties

J. Bégué, D. Bonnet‐Delpon, 2007 .

Fluoro-artemisinins: When a gem-difluoroethylene replaces a carbonyl group

B. Crousse, D. Bonnet-Delpon, J. Bégué, 2006 .

Orally active antimalarials: hydrolytically stable derivatives of 10-trifluoromethyl anhydrodihydroartemisinin.

B. Pradines, Sébastien Charneau, W. Charman, 2004, Journal of medicinal chemistry.

Fluoroartemisinin: trifluoromethyl analogues of artemether and artesunate.

Sébastien Charneau, P. Grellier, B. Crousse, 2004, Journal of medicinal chemistry.

Preparation of 10-trifluoromethyl artemether and artesunate. Influence of hexafluoropropan-2-ol on substitution reaction.

B. Crousse, D. Bonnet-Delpon, J. Bégué, 2003, The Journal of organic chemistry.

Anhydrodihydroartemisinin and its 10-trifluoromethyl analogue: access to novel d-ring-contracted artemisinin trifluoromethyl ketones.

B. Crousse, D. Bonnet-Delpon, J. Bégué, 2002, The Journal of organic chemistry.

New catalytic oxidation of trifluoromethyl carbinols by a ruthenium(II) complex

V. Kesavan, S. Chandrasekaran, D. Bonnet-Delpon, 2000 .

Barbier Conditions for Reformatsky and Alkylation Reactions on Trifluoromethyl Aldimines

B. Crousse, M. Santos, D. Bonnet‐Delpon, 2008 .

Trifluoromethylcyclohexane as a new solvent? Limits of use

J. Legros, B. Crousse, D. Bonnet-Delpon, 2002 .

Fluoroartemisinins: Metabolically More Stable Antimalarial Artemisinin Derivatives

D. Bonnet-Delpon, J. Bégué, D. Bonnet‐Delpon, 2007, ChemMedChem.

S(N)/S(N)' competition: selective access to new 10-fluoro artemisinins.

B. Crousse, D. Bonnet-Delpon, C. Chollet, 2006, The Journal of organic chemistry.

Synthesis and antimalarial activities of fluoroalkyl derivatives of dihydroartemisinin.

B. Pradines, D. Bonnet-Delpon, J. Bégué, 1998, Journal of medicinal chemistry.

Determination of Z and E configurations in trifluoromethylated vinyl compounds: 3J(CF) coupling constants as a criterion for configurational assignments

D. Bonnet-Delpon, J. Bégué, M. Ourévitch, 1991 .

A one-pot synthesis of 3-trifluoromethyl-2-isoxazolines from trifluoromethyl aldoxime

B. Crousse, D. Bonnet-Delpon, R. S. Gonçalves, 2013, Beilstein journal of organic chemistry.

Trifluoromethyl nitrones: from fluoral to optically active hydroxylamines.

B. Crousse, D. Bonnet-Delpon, T. Milcent, 2010, Organic & biomolecular chemistry.

Cyclic oxonium salts:13C magnetic resonance spectroscopy. The correlation of chemical shifts with the calculated charge density

D. Bonnet-Delpon, J. Bégué, D. Bonnet‐Delpon, 1980 .

Fluorinated Alcohols: A New Medium for Selective and Clean Reaction

B. Crousse, D. Bonnet-Delpon, J. Bégué, 2004 .

Synthesis and in vivo antimatarial activity of 12α-trifluoromethyl-hydroartemisinin

D. Bonnet-Delpon, J. Bégué, J. Gantier, 1996 .

Alkylation of manganese(II) tetraphenylporphyrin by antimalarial fluorinated artemisinin derivatives.

B. Meunier, D. Bonnet-Delpon, J. Bégué, 2003, Bioorganic & medicinal chemistry letters.

First synthesis of 10 alpha-(trifluoromethyl)deoxoartemisinin.

B. Crousse, D. Bonnet-Delpon, J. Bégué, 2002, Organic letters.

Self-Promoted Nucleophilic Addition of Hexafluoro-2-propanol to Vinyl Ethers

B. Crousse, D. Bonnet-Delpon, A. Salvo, 2006 .

Manganese (III) acetate dihydrate catalyzed aerobic epoxidation of unfunctionalized olefins in fluorous solvents

D. Bonnet-Delpon, J. Bégué, K. S. Ravikumar, 1998 .

Claisen rearrangement of α-(F-alkyl)enol ethers prepared via Wittig olefination of allyl perfluoroalkanoates

T. Nakai, D. Bonnet-Delpon, J. Bégué, 1994 .

Fluorous tagging of DABCO through halogen bonding: recyclable catalyst for the Morita-Baylis-Hillman reaction.

J. Legros, B. Crousse, D. Bonnet-Delpon, 2011, Chemical communications.

Syntheses, Biological Activity, and Conformational Analysis of Fluorine-Containing Taxoids

S. Kuduk, S. Chakravarty, J. Veith, 1996 .

Vinylogous Mannich reactions. Additions of trimethylsilyloxyfuran to fluorinated aldimines

B. Crousse, D. Bonnet-Delpon, J. Bégué, 2004 .

Solubility switch of gold nanoparticles through hydrogen bond association.

J. Legros, B. Crousse, D. Bonnet-Delpon, 2008, Chemical communications.

Self-assembly between 1,4-diazabicyclo[2.2.2]octane and bis(hexafluoroalcohols): solid/liquid phase switching for catalyst recycling

A. Slawin, J. Legros, B. Crousse, 2012 .

Influence of the structure of polyfluorinated alcohols on Brønsted acidity/hydrogen-bond donor ability and consequences on the promoter effect.

A. Slawin, J. Legros, B. Crousse, 2011, The Journal of organic chemistry.

A crystalline H-bond cluster of hexafluoroisopropanol (HFIP) and piperidine: Structure determination by X ray diffraction

G. Morgant, N. Ghermani, B. Crousse, 2007 .

Facile ring opening of oxiranes with aromatic amines in fluoro alcohols

V. Kesavan, Kesavan, B. Crousse, 2000, The Journal of organic chemistry.

Synthesis and evaluation of fluorinated analogues of monoamine reuptake inhibitors

D. Bonnet-Delpon, J. Kaffy, T. Milcent, 2012 .

Synthesis of 2-CF(3)-tetrahydroquinoline and quinoline derivatives from CF(3)-N-aryl-aldimine.

B. Crousse, D. Bonnet-Delpon, J. Bégué, 2000, The Journal of organic chemistry.

Synthesis of tetrahydroquinoline derivatives from α-CF3-N-arylaldimine and vinyl ethers

B. Crousse, D. Bonnet-Delpon, J. Bégué, 1998 .

Recent Advances (1995‐2005) in Fluorinated Pharmaceuticals Based on Natural Products

D. Bonnet-Delpon, J. Bégué, D. Bonnet‐Delpon, 2006 .

In vitro antileishmanial activity of fluoro-artemisinin derivatives against Leishmania donovani.

C. Bories, P. Loiseau, B. Crousse, 2008, Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie.

An efficient and robust fluoroketone catalyst epoxidation

J. Legros, B. Crousse, D. Bonnet-Delpon, 2001 .

Facile Access to Fluorinated Aryl and Vinyl Ethers through Copper‐Catalysed Reaction of Fluoro Alcohols

J. Legros, B. Crousse, D. Bonnet-Delpon, 2009 .

Solvent-promoted and -controlled aza-Michael reaction with aromatic amines.

B. Crousse, Kavita De, Julien Legros, 2009, The Journal of organic chemistry.

Aza-Diels–Alder reaction in fluorinated alcohols. A one-pot synthesis of tetrahydroquinolines

B. Crousse, D. Bonnet-Delpon, J. Bégué, 2003 .