Rabah A T Serya

发表

An overview on the prospective CDKs inhibitors as anti-cancer drugs : Review article

K. Abouzid, R. Serya, Khulood H. Oudah, 2017 .

Thieno[2,3-d]pyrimidine based derivatives as kinase inhibitors and anticancer agents

D. A. E. Ella, K. Abouzid, N. S. Ismail, 2015 .

Fragment‐Based Drug Discovery in the Bromodomain and Extra‐Terminal Domain Family

R. Serya, M. Radwan, Rabah A T Serya, 2017, Archiv der Pharmazie.

Pyrazolo[3,4-d]pyrimidine based scaffold derivatives targeting kinases as anticancer agents

D. A. Ibrahim, D. A. E. Ella, N. S. Ismail, 2016 .

Design, synthesis and biological evaluation of indazole–pyrimidine based derivatives as anticancer agents with anti-angiogenic and antiproliferative activities

D. A. E. Ella, K. Abouzid, M. Tolba, 2016 .

Structure-based design and synthesis of novel pseudosaccharine derivatives as antiproliferative agents and kinase inhibitors.

M. Linscheid, K. Abouzid, R. Serya, 2013, European journal of medicinal chemistry.

How to train your inhibitor: Design strategies to overcome resistance to Epidermal Growth Factor Receptor inhibitors.

K. Abouzid, Deena S. Lasheen, R. Serya, 2017, European journal of medicinal chemistry.

Virtual Screening and Synthesis of New Chemical Scaffolds as VEGFR-2 Kinase Inhibitors

K. Abouzid, R. Serya, Mohamed S. A. Elsayed, 2012, Arzneimittelforschung/Drug Research.

Novel quinoline-3-carboxamides (Part 2): Design, optimization and synthesis of quinoline based scaffold as EGFR inhibitors with potent anticancer activity.

S. Abbas, D. A. Abou El Ella, A. Esmat, 2017, Bioorganic chemistry.

Development of Potent Adenosine Monophosphate Activated Protein Kinase (AMPK) Activators

S. Kulp, K. Abouzid, N. S. Ismail, 2015, ChemMedChem.

Discovery of potent thieno[2,3-d]pyrimidine VEGFR-2 inhibitors: Design, synthesis and enzyme inhibitory evaluation supported by molecular dynamics simulations.

K. Abouzid, D. A. Abou El Ella, R. Serya, 2021, Bioorganic chemistry.

Penicillin binding protein 2a: An overview and a medicinal chemistry perspective.

K. Abouzid, R. Serya, M. Shalaby, 2020, European journal of medicinal chemistry.

Surmounting the resistance against EGFR inhibitors through the development of thieno[2,3-d]pyrimidine-based dual EGFR/HER2 inhibitors.

S. Minucci, K. Abouzid, Deena S. Lasheen, 2018, European journal of medicinal chemistry.

Rational design, synthesis and 2D-QSAR studies of antiproliferative tropane-based compounds

Adel S. Girgis, Riham F. George, Fady N. Baselious, 2016 .

Molecular design, synthesis and biological evaluation of novel 1,2,5-trisubstituted benzimidazole derivatives as cytotoxic agents endowed with ABCB1 inhibitory action to overcome multidrug resistance in cancer cells

M. Wink, K. Abouzid, M. Sobeh, 2022, Journal of enzyme inhibition and medicinal chemistry.

Anti-acetylcholinesterase activity of essential oils and their major constituents from four Ocimum species

M. Farag, S. Ezzat, M. Salama, 2016, Zeitschrift fur Naturforschung. C, Journal of biosciences.

Alkoxyphenylthiazoles with broad-spectrum activity against multidrug-resistant gram-positive bacterial pathogens.

M. Seleem, K. Abouzid, A. Taher, 2018, European journal of medicinal chemistry.

Ligand design and synthesis of new imidazo[5,1-b]quinazoline derivatives as alpha1-adrenoceptor agonists and antagonists.

K. Abouzid, M. Ismail, R. Serya, 2006, Bioorganic & medicinal chemistry.

Synthesis and molecular docking studies of some novel Schiff bases incorporating 6-butylquinolinedione moiety as potential topoisomerase IIβ inhibitors

R. Serya, Hany M Hassanin, M. Mostafa, 2018, Royal Society Open Science.

Design, synthesis, biological evaluation and dynamics simulation of indazole derivatives with antiangiogenic and antiproliferative anticancer activity.

Marawan Ahmed, K. Barakat, K. Abouzid, 2019, Bioorganic chemistry.

Molecular design and synthesis of 1,4-disubstituted piperazines as α(1)-adrenergic receptor blockers.

A. M. Al-Abd, K. Abouzid, D. Saleh, 2014, Bioorganic chemistry.

Pyrrolopyrimidine: A Versatile Scaffold for Construction of Targeted Anti-cancer Agents

K. Abouzid, Deena S. Lasheen, R. Serya, 2017 .

Pyrrolopyrimidine, A Multifaceted Scaffold in Cancer Targeted Therapy

K. Abouzid, Deena S. Lasheen, R. Serya, 2018, Drug Research.

Discovery of Potent VEGFR-2 Inhibitors based on Furopyrimidine and Thienopyrimidne Scaffolds as Cancer Targeting Agents

A. Mansour, K. Abouzid, Deena S. Lasheen, 2016, Scientific Reports.

Design, synthesis and molecular docking of novel pyrazolo[1,5-a][1,3,5]triazine derivatives as CDK2 inhibitors.

K. Abouzid, R. Serya, Khulood H. Oudah, 2019, Bioorganic chemistry.

Molecular design, synthesis and in vitro biological evaluation of thienopyrimidine–hydroxamic acids as chimeric kinase HDAC inhibitors: a challenging approach to combat cancer

N. Farag, K. Abouzid, Samar Mowafy, 2021, Journal of enzyme inhibition and medicinal chemistry.

Selective Small Molecule Myeloid Cell Leukemia-1 (MCL-1) Inhibitors: Novel Agents in Cancer Therapy

Deena S. Lasheen, R. Serya, H. Ibrahim, 2019, Archives of Pharmaceutical Sciences Ain Shams University.

A Fluorescence-Based Assay to Probe Inhibitory Effect of Fructose Mimics on GLUT5 Transport in Breast Cancer Cells

F. Wuest, K. Abouzid, Deena S. Lasheen, 2022, ACS bio & med chem Au.

Pyrazolo[1,5-a][1,3,5]triazine based scaffold as purine analogues with diverse biological activity

K. Abouzid, R. Serya, Mazin A. A. Najm, 2017 .

Targeting apoptotic machinery as approach for anticancer therapy: Smac mimetics as anticancer agents

D. A. E. Ella, K. Abouzid, R. Serya, 2015 .

Identification of Novel 4-Oxo-4H-chromen-Hydroxamic Acid Derivative Targeting Selected HDAC Isoforms

Rabah A T Serya, Rosaline Ashraf, Mai Adel, 2023, Archives of Pharmaceutical Sciences Ain Shams University.

Design, synthesis, 3D pharmacophore, QSAR, and docking studies of carboxylic acid derivatives as Histone Deacetylase inhibitors and cytotoxic agents.

N. Farag, K. Abouzid, R. Serya, 2014, Bioorganic chemistry.

Identification of novel pyrazole and benzimidazole based derivatives as PBP2a inhibitors: Design, synthesis, and biological evaluation

K. Abouzid, R. Serya, M. A. Shalaby, 2019, Archives of Pharmaceutical Sciences Ain Shams University.

Identification of new pyrrolo[2,3-d]pyrimidines as potent VEGFR-2 tyrosine kinase inhibitors: Design, synthesis, biological evaluation and molecular modeling.

K. Abouzid, Deena S. Lasheen, R. Serya, 2018, Bioorganic chemistry.

Synthesis, ADMET Properties, and Biological Evaluation of Benzothiazole Compounds Targeting Chemokine Receptor 2 (CXCR2)

N. Neamati, Tiangong Lu, K. Abouzid, 2017, ChemMedChem.

Synthesis and in vitro antiproliferative activity of certain novel pyrazolo[3,4‐b]pyridines with potential p38α MAPK‐inhibitory activity

H. Abdel‐Aziz, E. Samir, M. Y. Zaki, 2021, Archiv der Pharmazie.

Advances in non-Hydroxamate based Histone Deacetylase Inhibitors as Anticancer Agents

Rabah A T Serya, Khaled Abouzid, Nadine Wafik, 2024, Archives of Pharmaceutical Sciences Ain Shams University.

Synthesis and in vitro antiproliferative activity of novel pyrazolo[3,4-d]pyrimidine derivatives

K. Abouzid, N. S. Ismail, A. Esmat, 2015 .

Novel sulfonamide-indolinone hybrids targeting mitochondrial respiration of breast cancer cells.

M. Henary, D. A. Abou El Ella, Eman Z Elrazaz, 2024, European journal of medicinal chemistry.

Advances in the discovery of activin receptor-like kinase 5 (ALK5) inhibitors.

K. Abouzid, G. S. Hassan, Maiy Y. Jaballah, 2024, Bioorganic chemistry.

Molecular Dynamic Study and Synthesis of 1H-benzo[d]imidazole-5-carboxamide Derivatives as Inhibitors for Yellow Fever and Zika Virus Replication

J. Neyts, S. Kaptein, R. Serya, 2020, Archives of Pharmaceutical Sciences Ain Shams University.

Click and Release: SO2 Prodrugs with Tunable Release Rates.

B. Wang, K. Abouzid, Deena S. Lasheen, 2017, Organic letters.

Pyridazine Based Scaffolds as Privileged Structures in anti-Cancer Therapy

K. Abouzid, R. Serya, Maiy Jaballah, 2017, Drug Research.