Petro O. Borysko

发表

(Chlorosulfonyl)benzenesulfonyl Fluorides-Versatile Building Blocks for Combinatorial Chemistry: Design, Synthesis and Evaluation of a Covalent Inhibitor Library.

Yurii S. Moroz, M. Platonov, S. Zozulya, 2018, ACS combinatorial science.

Photochemical In-Flow Synthesis of 2,4-Methanopyrrolidines: Pyrrolidine Analogues with Improved Water Solubility and Reduced Lipophilicity.

A. Tolmachev, S. Zozulya, Oleg M. Michurin, 2018, The Journal of organic chemistry.

Photochemical Synthesis of 2-Azabicyclo[3.2.0]heptanes: Advanced Building Blocks for Drug Discovery. Synthesis of 2,3-Ethanoproline.

S. Zozulya, Pavel K. Mykhailiuk, P. Borysko, 2018, The Journal of organic chemistry.

2-Oxabicyclo[2.1.1]hexanes as saturated bioisosteres of the ortho-substituted phenyl ring

Pavel K. Mykhailiuk, G. Al-Maali, N. Voloshchuk, 2023, Nature Chemistry.

An iterative compound screening contest method for identifying target protein inhibitors using the tyrosine-protein kinase Yes

Daisuke Kihara, Takashi Ishida, Masakazu Sekijima, 2017, Scientific Reports.

Effect of gem-difluorination on the key physicochemical properties relevant to medicinal chemistry: the case of functionalized cycloalkanes.

O. Grygorenko, D. Volochnyuk, S. Ryabukhin, 2022, Chemistry.

Design of potentially active ligands for SH2 domains by molecular modeling methods

Vasyl V. Hurmach, O. M. Balinskyi, M. O. Platonov, 2014 .

Continued SAR exploration of 1,2,4-thiadiazole-containing scaffolds in the design of free fatty acid receptor 1 (GPR40) agonists.

I. Tikhonova, S. Zozulya, O. Onopchenko, 2017, European journal of medicinal chemistry.

Difluoromethyl Nitrile Oxide (CF2HCNO): A Neglected Chemical Reagent

Pavel K. Mykhailiuk, P. Borysko, Bohdan A. Chalyk, 2017 .

Anionic amphiphilic calixarenes for peptide assembly and delivery.

Y. Mély, R. Rodik, V. Kalchenko, 2022, Journal of colloid and interface science.

Straightforward hit identification approach in fragment-based discovery of bromodomain-containing protein 4 (BRD4) inhibitors.

Yurii S. Moroz, V. Hurmach, S. Zozulya, 2018, Bioorganic & Medicinal Chemistry.

The iterative application of a large chemical space in the drug discovery process

Yurii S. Moroz, Dmytro V. Dudenko, Igor Dziuba, 2021, Journal of Organic and Pharmaceutical Chemistry.

SAR by Space: Enriching Hit Sets from the Chemical Space

Christian Lemmen, Franca-Maria Klingler, Marcus Gastreich, 2019, Molecules.

Pros and cons of virtual screening based on public "Big Data": In silico mining for new bromodomain inhibitors.

Jürgen Bajorath, Dragos Horvath, Alexandre Varnek, 2019, European journal of medicinal chemistry.

Phosphine Oxides (-POMe2) for Medicinal Chemistry: Synthesis, Properties, and Applications.

H. Kuznietsova, Pavel K. Mykhailiuk, P. Borysko, 2021, The Journal of organic chemistry.

Anticancer activity features of imidazole-based ionic liquids and lysosomotropic detergents: in silico and in vitro studies.

V. Kovalishyn, D. Hodyna, Anastasiia Gryniukova, 2024, Molecular diversity.

Magnet for the Needle in Haystack: "Crystal Structure First" Fragment Hits Unlock Active Chemical Matter Using Targeted Exploration of Vast Chemical Spaces.

Yurii S. Moroz, G. Klebe, M. Gastreich, 2022, Journal of medicinal chemistry.

Oxa-spirocycles: synthesis, properties and applications

H. Kuznietsova, Pavel K. Mykhailiuk, P. Borysko, 2021, Chemical science.