Paul S. Watson

发表

Nonconventional Stereochemical Issues in the Design of the Synthesis of the Vancomycin Antibiotics: Challenges Imposed by Axial and Nonplanar Chiral Elements in the Heptapeptide Aglycons.

T. I. Richardson, Davidr . Evans, C. Dinsmore, 1998, Angewandte Chemie.

Approaches to the Synthesis of the Vancomycin Antibiotics. Synthesis of Orienticin C (Bis-dechlorovancomycin) Aglycon

J. Barrow, Davidr . Evans, J. Ellman, 1997 .

A diastereoselective synthesis of 2,4-disubstituted piperidines: scaffolds for drug discovery.

B. Jiang, B. Jiang, P. S. Watson, 2000, Organic letters.

Indazoles: regioselective protection and subsequent amine coupling reactions.

J. Lampe, W. Bodnar, David J. Slade, 2009, The Journal of organic chemistry.

From rigid cyclic templates to conformationally stabilized acyclic scaffolds. Part I: the discovery of CCR3 antagonist development candidate BMS-639623 with picomolar inhibition potency against eosinophil chemotaxis.

I. Kariv, S. Mandlekar, A. Tebben, 2008, Bioorganic & medicinal chemistry letters.

2,4-Disubstituted piperidines as selective CC chemokine receptor 3 (CCR3) antagonists: synthesis and selectivity.

G. Trainor, M. Covington, C. Decicco, 2006, Bioorganic & medicinal chemistry letters.

Discovery of N-propylurea 3-benzylpiperidines as selective CC chemokine receptor-3 (CCR3) antagonists.

G. Trainor, M. Covington, C. Decicco, 2004, Bioorganic & medicinal chemistry letters.

CCR3 antagonists: a potential new therapy for the treatment of asthma. Discovery and structure-activity relationships.

G. Trainor, M. Covington, C. Decicco, 2002, Bioorganic & medicinal chemistry letters.

Adenosine analogues as inhibitors of P2Y12 receptor mediated platelet aggregation.

J. Boyer, S. Mahanty, J. Douglass, 2008, Bioorganic & medicinal chemistry letters.

Lipophilic modifications to dinucleoside polyphosphates and nucleotides that confer antagonist properties at the platelet P2Y12 receptor.

J. Boyer, J. Douglass, C. Redick, 2008, Journal of medicinal chemistry.