Kazuaki Takami

发表

Discovery of Novel 5-(Piperazine-1-carbonyl)pyridin-2(1H)-one Derivatives as Orally eIF4A3-Selective Inhibitors.

K. Fukuda, Y. Imaeda, Y. Kosugi, 2017, ACS medicinal chemistry letters.

Synthesis, structure-activity relationship, and pharmacological studies of novel melanin-concentrating hormone receptor 1 antagonists 3-aminomethylquinolines: reducing human ether-a-go-go-related gene (hERG) associated liabilities.

J. Kunitomo, Masaharu Nakayama, Koki Kato, 2012, Journal of medicinal chemistry.

Discovery of Pyrazolo[1,5-a]pyrazin-4-ones as Potent and Brain Penetrant GluN2A-Selective Positive Allosteric Modulators Reducing AMPA Receptor Binding Activity.

Tomoaki Hasui, M. Corsi, M. Kamata, 2021, Bioorganic & medicinal chemistry.

Discovery of Brain-Penetrant Glucosylceramide Synthase Inhibitors with a Novel Pharmacophore.

H. Oki, T. Ohashi, Yuta Tanaka, 2022, Journal of medicinal chemistry.

Discovery of a novel series of GPR119 agonists: Design, synthesis, and biological evaluation of N-(Piperidin-4-yl)-N-(trifluoromethyl)pyrimidin-4-amine derivatives.

Kenjiro Sato, S. Iwasaki, Koji Watanabe, 2021, Bioorganic & medicinal chemistry.

Design and Identification of a GPR40 Full Agonist (SCO-267) Possessing a 2-Carbamoylphenyl Piperidine Moiety.

Mitsugi Ookawara, Masanori Watanabe, Y. Moritoh, 2020, Journal of medicinal chemistry.

Trans-hydrometalation of alkynes by a combination of InCl3 and DIBAL-H: one-pot access to functionalized (Z)-alkenes.

H. Yorimitsu, K. Oshima, K. Takami, 2002, Organic letters.

Palladium-catalyzed cross-coupling reaction of organoindiums with aryl halides in aqueous media.

H. Shinokubo, H. Yorimitsu, K. Oshima, 2001, Organic letters.

Triethylborane-induced radical reactions with gallium- and indium hydrides

S. Mikami, H. Shinokubo, H. Yorimitsu, 2003 .

Discovery of a novel series of medium-sized cyclic enteropeptidase inhibitors.

Sachiko Itono, K. Fukuda, Naohiro Taya, 2023, Bioorganic & medicinal chemistry.