Céline Bruyère

发表

N-(2-{3-[3,5-bis(trifluoromethyl)phenyl]ureido}ethyl)-glycyrrhetinamide (6b): a novel anticancer glycyrrhetinic acid derivative that targets the proteasome and displays anti-kinase activity.

R. Kiss, M. Prévost, V. Mathieu, 2011, Journal of medicinal chemistry.

Synthesis and anticancer activity evaluation of 2(4-alkoxyphenyl)cyclopropyl hydrazides and triazolo phthalazines.

R. Kiss, P. De, C. Bruyère, 2010, Bioorganic & medicinal chemistry.

Actomyosin contractility scales with myoblast elongation and enhances differentiation through YAP nuclear export

C. Bruyère, S. Gabriele, Marie Versaevel, 2019, Scientific Reports.

Ferrocifen derivatives that induce senescence in cancer cells: selected examples.

R. Kiss, A. Vessières, G. Jaouen, 2014, Journal of inorganic biochemistry.

Probing cytoskeletal pre-stress and nuclear mechanics in endothelial cells with spatiotemporally controlled (de-)adhesion kinetics on micropatterned substrates

W. D. De Vos, Thomas Grevesse, S. Gabriele, 2017, Cell adhesion & migration.

Targeting cyclin-dependent kinases in anti-neoplastic therapy.

L. Meijer, C. Bruyère, Céline Bruyère, 2013, Current opinion in cell biology.

Innovative Tools for Mechanobiology: Unraveling Outside-In and Inside-Out Mechanotransduction

C. Bruyère, S. Gabriele, Marie Versaevel, 2019, Front. Bioeng. Biotechnol..

Lycorine, the main phenanthridine Amaryllidaceae alkaloid, exhibits significant antitumor activity in cancer cells that display resistance to proapoptotic stimuli: an investigation of structure-activity relationship and mechanistic insight.

R. Kiss, A. Kornienko, V. Mathieu, 2009, Journal of medicinal chemistry.

Long-term in vitro treatment of human glioblastoma cells with temozolomide increases resistance in vivo through up-regulation of GLUT transporter and aldo-keto reductase enzyme AKR1C expression.

Gianluca Bontempi, Benjamin Haibe-Kains, R. Kiss, 2010, Neoplasia.

CDK/CK1 inhibitors roscovitine and CR8 downregulate amplified MYCN in neuroblastoma cells

Eugenia G. Giannopoulou, L. Meijer, N. Loaëc, 2014, Oncogene.

Matrix stiffness modulates formation and activity of neuronal networks of controlled architectures.

Stéphanie P Lacour, Danahe Mohammed, Sylvain Gabriele, 2016, Biomaterials.

Secondary Metabolites from a Culture of the Fungus Neosartorya pseudofischeri and Their In Vitro Cytostatic Activity in Human Cancer Cells

R. Kiss, L. Manoch, V. Mathieu, 2012, Planta Medica.

Growth inhibitory activities of oxyprenylated and non-prenylated naturally occurring phenylpropanoids in cancer cell lines.

R. Kiss, S. Genovese, M. Curini, 2011, Bioorganic & medicinal chemistry letters.

JLK1486, a Bis 8-Hydroxyquinoline-Substituted Benzylamine, Displays Cytostatic Effects in Experimental Gliomas through MyT1 and STAT1 Activation and, to a Lesser Extent, PPARγ Activation.

R. Kiss, J. Kraus, V. Mathieu, 2011, Translational oncology.

Temozolomide modifies caveolin-1 expression in experimental malignant gliomas in vitro and in vivo.

R. Kiss, R. Senetta, P. Cassoni, 2011, Translational oncology.

Synthesis and biological evaluation of analogs of the marine alkaloids granulatimide and isogranulatimide.

L. Meijer, R. Kiss, B. Ducommun, 2012, European journal of medicinal chemistry.

Long-term temozolomide treatment induces marked amino metabolism modifications and an increase in TMZ sensitivity in Hs683 oligodendroglioma cells.

Gianluca Bontempi, Benjamin Haibe-Kains, R. Kiss, 2010, Neoplasia.

Structure-Activity Relationship in the Leucettine Family of Kinase Inhibitors.

Y. Hérault, L. Meijer, Thu Lan Nguyen, 2021, Journal of medicinal chemistry.

Temozolomide-induced modification of the CXC chemokine network in experimental gliomas.

S. Spiegl-Kreinecker, W. Berger, R. Kiss, 2011, International journal of oncology.

Engineering slit-like channels for studying the growth of epithelial tissues in 3D-confined spaces.

C. Bruyère, S. Gabriele, Marie Versaevel, 2020, Biotechnology and bioengineering.

Collective migration during a gap closure in a two-dimensional haptotactic model

O. Theodoly, C. Bruyère, S. Gabriele, 2021, Scientific Reports.

Structure and in vitro antitumor activity evaluation of brominated diterpenes from the red alga Sphaerococcus coronopifolius.

R. Kiss, V. Roussis, C. Vagias, 2010, Bioorganic & medicinal chemistry.

New 5-Aryl-1H-imidazoles display in vitro antitumor activity against apoptosis-resistant cancer models, including melanomas, through mitochondrial targeting.

C. Pirker, W. Berger, R. Kiss, 2013, Journal of medicinal chemistry.

Investigations of fungal secondary metabolites with potential anticancer activity.

R. Kiss, V. Mathieu, A. Cimmino, 2010, Journal of natural products.

Natural product extracts of the Canadian prairie plant, Thermopsis rhombifolia, have anti-cancer activity in phenotypic cell-based assays

P. Colas, R. Golsteyn, S. Ruchaud, 2015, Natural product research.

Novel trisubstituted harmine derivatives with original in vitro anticancer activity.

R. Kiss, J. Wouters, A. Backlund, 2012, Journal of medicinal chemistry.

Growth inhibitory activity for cancer cell lines of lapachol and its natural and semi-synthetic derivatives.

R. Kiss, V. Mathieu, S. Genovese, 2014, Bioorganic & medicinal chemistry letters.

3D-QSAR, design, synthesis and characterization of trisubstituted harmine derivatives with in vitro antiproliferative properties.

R. Kiss, J. Wouters, C. Meinguet, 2015, European journal of medicinal chemistry.

Determination of the absolute configuration and evaluation of the in vitro antitumor activity of dilospirane B

R. Kiss, V. Mathieu, E. Ioannou, 2012 .

UNBS5162, a novel naphthalimide that decreases CXCL chemokine expression in experimental prostate cancers.

Gianluca Bontempi, Benjamin Haibe-Kains, R. Kiss, 2008, Neoplasia.