Rob Leurs

Predicting the target landscape of kinase inhibitors using 3D convolutional neural networks

Georgi K. Kanev, I. D. de Esch, C. de Graaf, 2023, PLoS Comput. Biol..

G protein‐coupled receptors: walking hand‐in‐hand, talking hand‐in‐hand?

H. Vischer, S. Nijmeijer, Rob Leurs, 2011, British journal of pharmacology.

Structural basis of ligand recognition and design of antihistamines targeting histamine H4 receptor

A. Windhorst, H. Vischer, Yu Qian, 2024, Nature communications.

Pharmacological characterization of seven human histamine H3 receptor isoforms

H. Vischer, Meichun Gao, Rob Leurs, 2023, bioRxiv.

Histamine H3 Receptor Isoforms: Insights from Alternative Splicing to Functional Complexity

H. Vischer, Meichun Gao, Rob Leurs, 2024, Biomolecules.

Ligand-directed biased agonism at human histamine H3 receptor isoforms across Gαi/o- and β-arrestin2-mediated pathways.

C. Langmead, A. Christopoulos, C. Valant, 2023, Biochemical pharmacology.

Synthesis and Pharmacological Characterization of New Photocaged Agonists for Histamine H3 and H4 Receptors

H. Vischer, M. Wijtmans, Yang Zheng, 2024, Pharmaceuticals.