S. Buchwald

发表

Dialkylbiaryl Phosphines in Pd-Catalyzed Amination: A User's Guide.

S. Buchwald, Stephen L Buchwald, David S Surry, 2010, Chemical science.

Palladium-Mediated Incorporation of Carboranes into Small Molecules, Peptides, and Proteins.

S. Buchwald, A. Loas, B. Pentelute, 2022, Journal of the American Chemical Society.

Yeast Reveal a “Druggable” Rsp5/Nedd4 Network that Ameliorates α-Synuclein Toxicity in Neurons

Daniel F Tardiff, S. Buchwald, S. Lindquist, 2013, Science.

Palladium-Catalyzed Amination of Unprotected Five-Membered Heterocyclic Bromides

S. Buchwald, Naoyuki Hoshiya, Mingjuan Su, 2014, Organic letters.

Identification and Rescue of α-Synuclein Toxicity in Parkinson Patient–Derived Neurons

Michael D. Pluth, D. Krainc, P. Auluck, 2013, Science.

Identification and Rescue of -Synuclein Toxicity in Parkinson Patient-Derived Neurons

Michael D. Pluth, R. Jaenisch, L. Tsai, 2013 .

Mild and highly selective palladium-catalyzed monoarylation of ammonia enabled by the use of bulky biarylphosphine ligands and palladacycle precatalysts.

D. Surry, C. Cheung, S. Buchwald, 2013, Organic letters.

Scope and limitations of the Pd/BINAP-catalyzed amination of aryl bromides.

S. Buchwald, J. Wolfe, John P. Wolfe† and, 2000, The Journal of organic chemistry.

The Palladium-Catalyzed Trifluoromethylation of Aryl Chlorides

S. Buchwald, Yong Zhang, E. Cho, 2010, Science.

Diamine Ligands in Copper-Catalyzed Reactions.

D. Surry, S. Buchwald, 2010, Chemical science.

Palladium-Catalyzed Negishi Coupling of α-CF3 Oxiranyl Zincate: Access to Chiral CF3-Substituted Benzylic Tertiary Alcohols.

S. Buchwald, Hu Zhang, S. Buchwald, 2017, Journal of the American Chemical Society.

Palladium-Catalyzed Fluorination of Cyclic Vinyl Triflates: Effect of TESCF3 as an Additive.

S. Buchwald, Yuxuan Ye, T. Takada, 2016, Angewandte Chemie.

A Fluorinated Ligand Enables Room-Temperature and Regioselective Pd-Catalyzed Fluorination of Aryl Triflates and Bromides

S. Buchwald, P. Müller, Yang Yang, 2015, Journal of the American Chemical Society.

In-Depth Assessment of the Palladium-Catalyzed Fluorination of Five-Membered Heteroaryl Bromides

S. Buchwald, Phillip J. Milner, Yang Yang, 2015, Organometallics.

Dosage Delivery of Sensitive Reagents Enables Glove Box-Free Synthesis

S. Buchwald, Hong Geun Lee, Aaron C. Sather, 2015, Nature.

Design of New Ligands for the Palladium-Catalyzed Arylation of α-Branched Secondary Amines.

Nathaniel H. Park, S. Buchwald, E. Vinogradova, 2015, Angewandte Chemie.

Palladium-catalyzed intramolecular C-H difluoroalkylation: synthesis of substituted 3,3-difluoro-2-oxindoles.

S. Buchwald, Shi‐Liang Shi, S. Buchwald, 2014, Angewandte Chemie.

Studying Regioisomer Formation in the Pd-Catalyzed Fluorination of Aryl Triflates by Deuterium Labeling

S. Buchwald, Phillip J. Milner, Yong Zhang, 2014, Journal of the American Chemical Society.

Pd-Catalyzed Nucleophilic Fluorination of Aryl Bromides

S. Buchwald, Phillip J. Milner, Hong Geun Lee, 2014, Journal of the American Chemical Society.

An improved catalyst system for the Pd-catalyzed fluorination of (hetero)aryl triflates.

S. Buchwald, Phillip J. Milner, Hong Geun Lee, 2013, Organic letters.

Rapid and efficient trifluoromethylation of aromatic and heteroaromatic compounds using potassium trifluoroacetate enabled by a flow system.

S. Buchwald, Mao Chen, S. Buchwald, 2013, Angewandte Chemie.

Synthesis of optically pure 2-trifluoromethyl lactic acid by asymmetric hydroformylation.

S. Buchwald, Xiao Wang, S. Buchwald, 2013, The Journal of organic chemistry.

Room temperature copper(II)-catalyzed oxidative cyclization of enamides to 2,5-disubstituted oxazoles via vinylic C-H functionalization.

S. Buchwald, C. Cheung, S. Buchwald, 2012, The Journal of organic chemistry.

Copper-catalyzed oxytrifluoromethylation of unactivated alkenes.

R. Zhu, S. Buchwald, 2012, Journal of the American Chemical Society.

Iron(II)-catalyzed trifluoromethylation of potassium vinyltrifluoroborates.

A. T. Parsons, T. Senecal, S. Buchwald, 2012, Angewandte Chemie.

Organic chemistry: A radical approach to diversity

S. Buchwald, A. T. Parsons, S. Buchwald, 2011, Nature.

The palladium-catalyzed trifluoromethylation of vinyl sulfonates.

S. Buchwald, E. Cho, S. Buchwald, 2011, Organic letters.

Evidence for in situ catalyst modification during the Pd-catalyzed conversion of aryl triflates to aryl fluorides.

Yong Zhang, T. Maimone, M. Takase, 2011, Journal of the American Chemical Society.

Accelerating palladium-catalyzed C-F bond formation: use of a microflow packed-bed reactor.

Timothy Noël, S. Buchwald, T. Noël, 2011, Angewandte Chemie.

Copper-catalyzed trifluoromethylation of unactivated olefins.

S. Buchwald, A. T. Parsons, S. Buchwald, 2011, Angewandte Chemie.

Formation of ArF from LPdAr(F): Catalytic Conversion of Aryl Triflates to Aryl Fluorides

Yong Zhang, D. Watson, Georgiy Teverovskiy, 2009, Science.

Copper-diamine-catalyzed N-arylation of pyrroles, pyrazoles, indazoles, imidazoles, and triazoles.

S. Buchwald, Jeremy M. Baskin, J. Antilla, 2004, The Journal of organic chemistry.

C-H functionalization/C-N bond formation: copper-catalyzed synthesis of benzimidazoles from amidines.

S. Buchwald, Gordon Brasche, S. Buchwald, 2008, Angewandte Chemie.

An improved system for the palladium-catalyzed borylation of aryl halides with pinacol borane.

S. Buchwald, K. Billingsley, S. Buchwald, 2008, The Journal of organic chemistry.

Suzuki-Miyaura cross-coupling of unprotected, nitrogen-rich heterocycles: substrate scope and mechanistic investigation.

S. Buchwald, M. A. Düfert, K. Billingsley, 2013, Journal of the American Chemical Society.

A new palladium precatalyst allows for the fast Suzuki-Miyaura coupling reactions of unstable polyfluorophenyl and 2-heteroaryl boronic acids.

S. Buchwald, Yong Zhang, T. Kinzel, 2010, Journal of the American Chemical Society.

A general and efficient method for the Suzuki-Miyaura coupling of 2-pyridyl nucleophiles.

S. Buchwald, K. Billingsley, S. Buchwald, 2008, Angewandte Chemie.

Highly efficient monophosphine-based catalyst for the palladium-catalyzed suzuki-miyaura reaction of heteroaryl halides and heteroaryl boronic acids and esters.

S. Buchwald, K. Billingsley, S. Buchwald, 2007, Journal of the American Chemical Society.

Design and Preparation of New Palladium Precatalysts for C-C and C-N Cross-Coupling Reactions.

S. Buchwald, Stephen L Buchwald, M. Tudge, 2012, Chemical science.

A new class of easily activated palladium precatalysts for facile C-N cross-coupling reactions and the low temperature oxidative addition of aryl chlorides.

S. Buchwald, B. Fors, M. R. Biscoe, 2008, Journal of the American Chemical Society.

Mild and general conditions for negishi cross-coupling enabled by the use of palladacycle precatalysts.

S. Buchwald, Yang Yang, Nathan J. Oldenhuis, 2012, Angewandte Chemie.

A general method for Suzuki-Miyaura coupling reactions using lithium triisopropyl borates.

S. Buchwald, M. Oberli, S. Buchwald, 2012, Organic letters.

Palladium-catalyzed Suzuki-Miyaura cross-coupling reactions employing dialkylbiaryl phosphine ligands.

S. Buchwald, Rúben Martín, R. Martín, 2008, Accounts of chemical research.

Palladium-catalyzed borylation of aryl chlorides: scope, applications, and computational studies.

S. Buchwald, Timothy E. Barder, K. Billingsley, 2007, Angewandte Chemie.

N-Substituted 2-Aminobiphenylpalladium Methanesulfonate Precatalysts and Their Use in C–C and C–N Cross-Couplings

S. Buchwald, Nicholas C. Bruno, N. Niljianskul, 2014, The Journal of organic chemistry.

Synthesis and application of palladium precatalysts that accommodate extremely bulky di-tert-butylphosphino biaryl ligands.

S. Buchwald, Nicholas C. Bruno, S. Buchwald, 2013, Organic letters.

Structural Insights into Active Catalyst Structures and Oxidative Addition to (Biaryl)phosphine−Palladium Complexes via Density Functional Theory and Experimental Studies

S. Buchwald, Timothy E. Barder, and Mark R. Biscoe, 2007 .

Mild and efficient copper-catalyzed amination of aryl bromides with primary alkylamines.

S. Buchwald, F. Kwong, S. Buchwald, 2003, Organic letters.

Copper-catalyzed coupling of alkylamines and aryl iodides: an efficient system even in an air atmosphere.

S. Buchwald, A. Klapars, F. Kwong, 2002, Organic letters.

Palladium-catalyzed intramolecular C-O bond formation.

S. Buchwald, K. E. Torraca, S. Kuwabe, 2001, Journal of the American Chemical Society.

Copper-catalyzed domino halide exchange-cyanation of aryl bromides.

S. Buchwald, J. Zanon, A. Klapars, 2003, Journal of the American Chemical Society.

Pd-catalyzed Suzuki–Miyaura reactions of aryl halides using bulky biarylmonophosphine ligands

S. Buchwald, Ryan A. Altman, S. Buchwald, 2007, Nature Protocols.

Catalyst-controlled chemoselective arylation of 2-aminobenzimidazoles.

S. Buchwald, S. Ueda, S. Buchwald, 2012, Angewandte Chemie.

Catalysts for Suzuki-Miyaura coupling processes: scope and studies of the effect of ligand structure.

S. Buchwald, J. R. Martinelli, Timothy E. Barder, 2005, Journal of the American Chemical Society.

Catalytic Asymmetric Synthesis of α-Arylpyrrolidines and Benzo-fused Nitrogen Heterocycles.

S. Buchwald, Xi-Jie Dai, Thierry León, 2019, Angewandte Chemie.

An Ammonia Equivalent for the Palladium-Catalyzed Amination of Aryl Halides and Triflates

S. Buchwald, J. Wolfe, J. Ahman, 1997 .

Aryl amination using ligand-free Ni(II) salts and photoredox catalysis

I. Davies, D. MacMillan, S. Dreher, 2016, Science.

Copper-catalyzed coupling of aryl iodides with aliphatic alcohols.

S. Buchwald, M. Wolter, G. Nordmann, 2002, Organic letters.

Copper Hydride Catalyzed Enantioselective Synthesis of Axially Chiral 1,3-Disubstituted Allenes

S. Buchwald, Liela Bayeh-Romero, S. Buchwald, 2019, Journal of the American Chemical Society.

Mechanistically Guided Design of Ligands That Significantly Improve the Efficiency of CuH-Catalyzed Hydroamination Reactions.

Peng Liu, Andy A Thomas, Klaus Speck, 2018, Journal of the American Chemical Society.

Ligand-Substrate Dispersion Facilitates the Copper-Catalyzed Hydroamination of Unactivated Olefins.

D. Lambrecht, Peng Liu, Yang Yang, 2017, Journal of the American Chemical Society.

Microfluidic electrochemistry for single-electron transfer redox-neutral reactions

S. Buchwald, K. Jensen, N. Gershenfeld, 2020, Science.

An improved Cu-based catalyst system for the reactions of alcohols with aryl halides.

Phillip A Lichtor, S. Buchwald, Ryan A. Altman, 2008, The Journal of organic chemistry.

Practical Palladium Catalysts for C-N and C-O Bond Formation

S. Buchwald, Alexander R. Muci, S. Buchwald, 2002 .

Biaryl phosphane ligands in palladium-catalyzed amination.

D. Surry, S. Buchwald, 2008, Angewandte Chemie.

Catalytic enantioselective conjugate reduction of lactones and lactams.

S. Buchwald, G. Hughes, M. Kimura, 2003, Journal of the American Chemical Society.

Asymmetric Conjugate Reduction of α,β-Unsaturated Esters Using a Chiral Phosphine−Copper Catalyst

S. Buchwald, Y. Moritani, R. Shintani, 1999 .

Pd-catalyzed synthesis of Ar-SCF3 compounds under mild conditions.

Georgiy Teverovskiy, D. Surry, S. Buchwald, 2011, Angewandte Chemie.

Combined oxypalladation/C-H functionalization: palladium(II)-catalyzed intramolecular oxidative oxyarylation of hydroxyalkenes.

S. Buchwald, R. Zhu, S. Buchwald, 2012, Angewandte Chemie.

Room temperature aryl trifluoromethylation via copper-mediated oxidative cross-coupling.

S. Buchwald, A. T. Parsons, T. Senecal, 2011, The Journal of organic chemistry.

Copper-Catalyzed Oxytrifluoromethylation of Unactivated Alkenes

S. Buchwald, R. Zhu, S. Buchwald, 2012 .

Continuous-Flow Synthesis of Biaryls by Negishi Cross-Coupling of Fluoro- and Trifluoromethyl-Substituted (Hetero)arenes.

S. Buchwald, Stefan Roesner, S. Buchwald, 2016, Angewandte Chemie.

The Evolution of Pd0/PdII-Catalyzed Aromatic Fluorination

Aaron C. Sather, S. Buchwald, 2016, Accounts of chemical research.

Pd-catalyzed conversion of aryl chlorides, triflates, and nonaflates to nitroaromatics.

S. Buchwald, B. Fors, S. Buchwald, 2009, Journal of the American Chemical Society.

Structural reevaluation of the electrophilic hypervalent iodine reagent for trifluoromethylthiolation supported by the crystalline sponge method for X-ray analysis.

S. Buchwald, P. Müller, E. Vinogradova, 2014, Angewandte Chemie.

A chemoselective strategy for late-stage functionalization of complex small molecules with polypeptides and proteins

Zachary Shriver, Kenneth D. Johnson, Scott J. Miller, 2018, Synthesis.

Rapid Synthesis of Aryl Fluorides in Continuous Flow through the Balz-Schiemann Reaction.

Nathaniel H. Park, S. Buchwald, Timothy J Senter, 2016, Angewandte Chemie.

A versatile catalyst system for Suzuki-Miyaura cross-coupling reactions of C(sp(2))-tosylates and mesylates.

S. Buchwald, Brijesh Bhayana, B. Fors, 2009, Organic letters.

A highly active catalyst for Suzuki-Miyaura cross-coupling reactions of heteroaryl compounds.

S. Buchwald, K. Anderson, K. Billingsley, 2006, Angewandte Chemie.

Monophosphine Ligands Promote Pd-Catalyzed C-S Cross-Coupling Reactions at Room Temperature with Soluble Bases.

S. Buchwald, C. Yeung, Richard Y. Liu, 2019, ACS catalysis.

Oxidative Addition Complexes as Precatalysts for Cross-Coupling Reactions Requiring Extremely Bulky Biarylphosphine Ligands.

S. Buchwald, Bryan T. Ingoglia, S. Buchwald, 2017, Organic letters.

Investigating the dearomative rearrangement of biaryl phosphine-ligated Pd(II) complexes.

Jiahao Chen, P. Müller, T. Maimone, 2012, Journal of the American Chemical Society.

An Improved Synthesis of BrettPhos and RockPhos-Type Biarylphosphine Ligands.

S. Buchwald, Naoyuki Hoshiya, N. Hoshiya, 2012, Advanced synthesis & catalysis.

A single phosphine ligand allows palladium-catalyzed intermolecular C-O bond formation with secondary and primary alcohols.

B. Fors, Xiaoxing Wu, S. Buchwald, 2011, Angewandte Chemie.

An improved palladium-catalyzed conversion of aryl and vinyl triflates to bromides and chlorides.

S. Buchwald, Yong Zhang, Jun Pan, 2011, Organic letters.

Palladium-catalyzed conversion of aryl and vinyl triflates to bromides and chlorides.

Xiaoqiang Shen, Alan M. Hyde, S. Buchwald, 2010, Journal of the American Chemical Society.

Pd-catalyzed O-arylation of ethyl acetohydroximate: synthesis of O-arylhydroxylamines and substituted benzofurans.

S. Buchwald, T. Maimone, S. Buchwald, 2010, Journal of the American Chemical Society.

A highly active catalyst for Pd-catalyzed amination reactions: cross-coupling reactions using aryl mesylates and the highly selective monoarylation of primary amines using aryl chlorides.

S. Buchwald, B. Fors, D. Watson, 2008, Journal of the American Chemical Society.

CuH-Catalyzed Asymmetric Hydroamidation of Vinylarenes.

S. Buchwald, J. Bandar, Yujing Zhou, 2018, Angewandte Chemie.

Enantioselective functionalization of radical intermediates in redox catalysis: copper-catalyzed asymmetric oxytrifluoromethylation of alkenes.

S. Buchwald, R. Zhu, S. Buchwald, 2013, Angewandte Chemie.

Palladium(0)-catalyzed arylative dearomatization of phenols.

Sophie A. L. Rousseaux, J. García-Fortanet, Miguel Angel Del Aguila Sanchez, 2011, Journal of the American Chemical Society.

A Dual CuH- and Pd-Catalyzed Stereoselective Synthesis of Highly Substituted 1,3-Dienes.

S. Buchwald, Anton Z Ni, James Levi Knippel, 2021, Organic letters.

Copper-catalyzed coupling of arylboronic acids and amines.

S. Buchwald, J. Antilla, S. Buchwald, 2001, Organic letters.

Palladium-Catalyzed α-Arylation of Esters

S. Buchwald, W. Moradi, S. Buchwald, 2001 .

Catalytic asymmetric vinylation of ketone enolates.

S. Buchwald, A. Chieffi, J. Ahman, 2001, Organic letters.

A Highly Active Catalyst for Palladium-Catalyzed Cross-Coupling Reactions: Room-Temperature Suzuki Couplings and Amination of Unactivated Aryl Chlorides

John P. Wolfe, Stephen L. Buchwald, S. Buchwald, 1998 .

Pd(PhCN)(2)Cl(2)/P(t-Bu)(3): a versatile catalyst for Sonogashira reactions of aryl bromides at room temperature.

S. Buchwald, G. C. Fu, A. Littke, 2000, Organic letters.

Copper-catalyzed C-P bond construction via direct coupling of secondary phosphines and phosphites with aryl and vinyl halides.

D. Gelman, Lei Jiang, S. Buchwald, 2003, Organic letters.

Enantioselective CuH-Catalyzed Hydroacylation Employing Unsaturated Carboxylic Acids as Aldehyde Surrogates.

S. Buchwald, J. Bandar, Yujing Zhou, 2017, Journal of the American Chemical Society.

Enantioselective CuH-Catalyzed Reductive Coupling of Aryl Alkenes and Activated Carboxylic Acids

S. Buchwald, J. Bandar, E. Ascic, 2016, Journal of the American Chemical Society.

Use of tunable ligands allows for intermolecular Pd-catalyzed C--O bond formation.

S. Buchwald, Xiaohua Huang, A. Vorogushin, 2005, Journal of the American Chemical Society.

Palladium-catalyzed formation of aryl tert-butyl ethers from unactivated aryl halides.

S. Buchwald, C. Parrish, S. Buchwald, 2001, The Journal of organic chemistry.

A High-Yield, General Method for the Catalytic Formation of Oxygen Heterocycles

S. Buchwald, K. E. Torraca, and Shin-Itsu Kuwabe, 2000 .

Novel Electron-Rich Bulky Phosphine Ligands Facilitate the Palladium-Catalyzed Preparation of Diaryl Ethers

S. Buchwald, J. Wolfe, A. Aranyos, 1999 .

ELECTRONIC DEPENDENCE OF C-O REDUCTIVE ELIMINATION FROM PALLADIUM (ARYL)NEOPENTOXIDE COMPLEXES

S. Buchwald, R. Widenhoefer, S. Buchwald, 1998 .

DIRECT OBSERVATION OF C-O REDUCTIVE ELIMINATION FROM PALLADIUM ARYL ALKOXIDE COMPLEXES TO FORM ARYL ETHERS

S. Buchwald, R. Widenhoefer, A. Zhong, 1997 .

Synthesis of Oxygen Heterocycles via a Palladium-Catalyzed C−O Bond-Forming Reaction

S. Buchwald, J. Wolfe, M. Palucki, 1996 .

Mild Pd-Catalyzed Aminocarbonylation of (Hetero)Aryl Bromides with a Palladacycle Precatalyst

S. Buchwald, T. Skrydstrup, Stig D. Friis, 2014, Organic letters.

Unexpected Formation of Hexasubstituted Arenes through a Twofold Palladium-Mediated Ligand Arylation.

S. Buchwald, Corin C. Wagen, Bryan T. Ingoglia, 2019, The Journal of organic chemistry.

Palladium-Mediated Arylation of Lysine in Unprotected Peptides.

S. Buchwald, B. Pentelute, Hong Geun Lee, 2017, Angewandte Chemie.

Structure and Reactivity of [(L•Pd)n•(1,5-cyclooctadiene)] (n=1-2) Complexes Bearing Biaryl Phosphine Ligands.

Michael T. Colvin, S. Buchwald, L. Andreas, 2014, Inorganica chimica acta.

Palladium-catalyzed cross-coupling of aryl chlorides and triflates with sodium cyanate: a practical synthesis of unsymmetrical ureas.

S. Buchwald, B. Fors, E. Vinogradova, 2012, Journal of the American Chemical Society.

Palladium-catalyzed N-arylation of 2-aminothiazoles.

S. Buchwald, Jaclyn L Henderson, Meredeth A. McGowan, 2012, Organic letters.

A bulky biaryl phosphine ligand allows for palladium-catalyzed amidation of five-membered heterocycles as electrophiles.

S. Buchwald, Mingjuan Su, S. Buchwald, 2012, Angewandte Chemie.

Synthesis of unsymmetrical diarylureas via Pd-catalyzed C-N cross-coupling reactions.

S. Buchwald, B. Fors, S. Breitler, 2011, Organic letters.

Pd-catalyzed cross-coupling reactions of amides and aryl mesylates.

S. Buchwald, B. Fors, K. Dooleweerdt, 2010, Organic letters.

An Efficient System For the Pd-Catalyzed Cross-Coupling of Amides and Aryl Chlorides.

S. Buchwald, B. Fors, Qingle Zeng, 2009, Tetrahedron.

Completely N1-selective palladium-catalyzed arylation of unsymmetric imidazoles: application to the synthesis of nilotinib.

S. Buchwald, S. Ueda, Mingjuan Su, 2012, Journal of the American Chemical Society.

Palladium-catalyzed silylation of aryl chlorides with hexamethyldisilane.

S. Buchwald, Timothy E. Barder, Eric McNeill, 2007, Organic letters.

Pd-catalyzed N-arylation of secondary acyclic amides: catalyst development, scope, and computational study.

S. Buchwald, J. Hicks, Alan M. Hyde, 2009, Journal of the American Chemical Society.

Mechanistic studies on the copper-catalyzed N-arylation of amides.

S. Buchwald, E. Strieter, Brijesh Bhayana, 2008, Journal of the American Chemical Society.

Palladium-catalyzed method for the synthesis of carbazoles via tandem C-H functionalization and C-N bond formation.

Rachel Munday, Gordon Brasche, N. Zheng, 2008, The Journal of organic chemistry.

Pd-catalyzed amidation of aryl chlorides using monodentate biaryl phosphine ligands: a kinetic, computational, and synthetic investigation.

S. Buchwald, M. R. Biscoe, Takashi Ikawa, 2007, Journal of the American Chemical Society.

Combined C-H functionalization/C-N bond formation route to carbazoles.

S. Buchwald, N. Zheng, W. Tsang, 2005, Journal of the American Chemical Society.

A general and efficient copper catalyst for the amidation of aryl halides.

S. Buchwald, A. Klapars, Xiaohua Huang, 2002, Journal of the American Chemical Society.

Applications of Palladium-Catalyzed C–N Cross-Coupling Reactions

Stephen L. Buchwald, S. Buchwald, Paula Ruiz-Castillo, 2016, Chemical reviews.

A Simple Catalytic Method for the Conversion of Aryl Bromides to Arylamines

S. Buchwald, R. Rennels, A. Guram, 1995 .

A general, efficient, and inexpensive catalyst system for the coupling of aryl iodides and thiols.

S. Buchwald, F. Kwong, S. Buchwald, 2002, Organic letters.

General catalysts for the Suzuki-Miyaura and Sonogashira coupling reactions of aryl chlorides and for the coupling of challenging substrate combinations in water.

S. Buchwald, K. Anderson, S. Buchwald, 2005, Angewandte Chemie.

Palladium Mediated Synthesis of Protein-Polyarene Conjugates.

S. Buchwald, B. Pentelute, Heemal H. Dhanjee, 2022, Journal of the American Chemical Society.

Highly Enantioselective Imine Hydrosilylation Using (S,S)-Ethylenebis(η5-tetrahydroindenyl)titanium Difluoride

S. Buchwald, X. Verdaguer, Udo E W Lange, 1996 .

A catalytic method for the reduction of esters to alcohols

S. Buchwald, Scott C. Berk, S. Berk, 1991 .

On the role of metal contaminants in catalyses with FeCl3.

S. Buchwald, C. Bolm, S. Buchwald, 2009, Angewandte Chemie.

Pd-Catalyzed C-N Coupling Reactions Facilitated by Organic Bases: Mechanistic Investigation Leads to Enhanced Reactivity in the Arylation of Weakly Binding Amines.

S. Buchwald, J. Dennis, Richard Y. Liu, 2019, ACS catalysis.

Palladium-Catalyzed Synthesis of Monodisperse, Controlled-Length, and Functionalized Oligoanilines

S. Buchwald, J. Sadighi, A. Singer, 1998 .

A GENERAL SYNTHESIS OF END-FUNCTIONALIZED OLIGOANILINES VIA PALLADIUM-CATALYZED AMINATION

S. Buchwald, J. Sadighi, R. Singer, 1998 .

An integrated microreactor system for self-optimization of a Heck reaction: from micro- to mesoscale flow systems.

Klavs F Jensen, Matthew T. Stone, S. Buchwald, 2010, Angewandte Chemie.

Stereochemistry of nucleophilic displacement on two phosphoric monoesters and a phosphoguanidine: the role of metaphosphate

S. Buchwald, J. Knowles, J. Friedman, 1984 .

Suzuki–Miyaura cross-coupling optimization enabled by automated feedback

Klavs F. Jensen, Brandon J. Reizman, Stephen L. Buchwald, 2016, Reaction chemistry & engineering.

Copper-catalyzed vinylation of hydrazides. A regioselective entry to highly substituted pyrroles.

S. Buchwald, M. Rivero, S. Buchwald, 2007, Organic letters.

Domino cu-catalyzed C--N coupling/hydroamidation: a highly efficient synthesis of nitrogen heterocycles.

S. Buchwald, Ruben Martin, M. Rodríguez Rivero, 2006, Angewandte Chemie.

A general method for the preparation of zirconocene complexes of substituted benzynes: in situ generation, coupling reactions, and use in the synthesis of polyfunctionalized aromatic compounds

W. A. Nugent, S. Buchwald, R. Lum, 1987 .

Synthesis of Pyrroles Through the CuH-Catalyzed Coupling of Enynes and Nitriles.

S. Buchwald, P. Liu, Peng Liu, 2020, Journal of the American Chemical Society.

Cu-catalyzed tandem C-N bond formation for the synthesis of pyrroles and heteroarylpyrroles.

S. Buchwald, A. Cuenca, Rúben Martín, 2007, Organic letters.

Copper-catalyzed enantioselective stereodivergent synthesis of amino alcohols

S. Buchwald, Shi‐Liang Shi, Zackary L. Wong, 2016, Nature.

Copper Hydride Catalyzed Hydroamination of Alkenes and Alkynes.

Michael T Pirnot, Yi‐Ming Wang, S. Buchwald, 2015, Angewandte Chemie.

Enantioselective synthesis of α-aminosilanes by copper-catalyzed hydroamination of vinylsilanes.

S. Buchwald, Shaolin Zhu, N. Niljianskul, 2014, Angewandte Chemie.

Enantioselective CuH-Catalyzed Anti-Markovnikov Hydroamination of 1,1-Disubstituted Alkenes

S. Buchwald, Shaolin Zhu, S. Buchwald, 2014, Journal of the American Chemical Society.

The zirconocene induced coupling of benzyne with nitriles: Synthesis, structure and reactions of novel azametallacyclopentenes

S. Buchwald, J. Dewan, J. C. Dewan, 1987 .

Cu-catalyzed arylation of phenols: synthesis of sterically hindered and heteroaryl diaryl ethers.

S. Buchwald, D. Maiti, S. Buchwald, 2010, The Journal of organic chemistry.

New insights into Xantphos/Pd-Catalyzed C-N bond forming reactions : A structural and kinetic study

Stephen L. Buchwald, S. Buchwald, E. Strieter, 2006 .

Studying Regioisomer Formation in the Pd-Catalyzed Fluorination of Cyclic Vinyl Triflates: Evidence for in situ Ligand Modification.

M. Baik, Yuxuan Ye, Seoung-Tae Kim, 2023, Angewandte Chemie.

Overcoming the Challenges of Solid Bridging and Constriction during Pd-Catalyzed C−N Bond Formation in Microreactors

Klavs F. Jensen, Nikolay Zaborenko, Ryan L. Hartman, 2010 .

PALLADIUM-CATALYZED AMINATION OF ARYL IODIDES

S. Buchwald, J. Wolfe, S. Buchwald, 1996 .

Rapid and efficient copper-catalyzed Finkelstein reaction of (hetero)aromatics under continuous-flow conditions.

S. Buchwald, Mao Chen, Stephen L Buchwald, 2015, Angewandte Chemie.

N- versus O-arylation of aminoalcohols: orthogonal selectivity in copper-based catalysts.

Phillip A Lichtor, S. Buchwald, A. Shafir, 2007, Journal of the American Chemical Society.

Palladium‐Catalyzed Aromatic Carbon‐Nitrogen Bond Formation

S. Buchwald, Lei Jiang, S. Buchwald, 2008 .

4,7-Dimethoxy-1,10-phenanthroline: an excellent ligand for the Cu-catalyzed N-arylation of imidazoles.

S. Buchwald, Ryan A. Altman, S. Buchwald, 2006, Organic letters.

A general and efficient copper catalyst for the amidation of aryl halides and the N-arylation of nitrogen heterocycles.

S. Buchwald, J. Antilla, A. Klapars, 2001, Journal of the American Chemical Society.

An efficient copper-catalyzed coupling of aryl halides with imidazoles

S. Buchwald, J. Marcoux, Ayumu Kiyomori, 1999 .

Computational explorations of mechanisms and ligand-directed selectivities of copper-catalyzed Ullmann-type reactions.

K. Houk, Peng Liu, Gavin O. Jones, 2010, Journal of the American Chemical Society.

The copper-catalyzed N-arylation of indoles.

S. Buchwald, J. Antilla, A. Klapars, 2002, Journal of the American Chemical Society.

Orthogonal Cu- and Pd-based catalyst systems for the O- and N-arylation of aminophenols.

S. Buchwald, D. Maiti, S. Buchwald, 2009, Journal of the American Chemical Society.

A new biarylphosphine ligand for the Pd-catalyzed synthesis of diaryl ethers under mild conditions.

S. Buchwald, N. Davis, Luca Salvi, 2011, Organic letters.

Significantly improved method for the pd-catalyzed coupling of phenols with aryl halides: understanding ligand effects.

S. Buchwald, Xiaohua Huang, Timothy E. Barder, 2006, Angewandte Chemie.

Room-Temperature Cu-Catalyzed Amination of Aryl Bromides Enabled by DFT-Guided Ligand Design.

S. Buchwald, Albert Cabré, M. Strauss, 2023, Journal of the American Chemical Society.

Orthogonal Cu‐ and Pd‐Based Catalyst Systems for the O‐ and N‐Arylation of Aminophenols.

D. Maiti, S. Buchwald, 2009 .

A domino copper-catalyzed C-O coupling-Claisen rearrangement process.

S. Buchwald, G. Nordmann, S. Buchwald, 2003, Journal of the American Chemical Society.

Design of Modified Amine Transfer Reagents Allows the Synthesis of α-Chiral Secondary Amines via CuH-Catalyzed Hydroamination

S. Buchwald, D. Niu, S. Buchwald, 2015, Journal of the American Chemical Society.

Organometallic Palladium Reagents for Cysteine Bioconjugation

Alexander M. Spokoyny, Bradley L. Pentelute, Stephen L. Buchwald, 2015, Nature.

Engineering Bioactive Dimeric Transcription Factor Analogs via Palladium Rebound Reagents.

Carly K. Schissel, S. Buchwald, Isaac A. Klein, 2021, Journal of the American Chemical Society.

Accelerating reactions with microreactors at elevated temperatures and pressures: profiling aminocarbonylation reactions.

Klavs F Jensen, Nikolay Zaborenko, S. Buchwald, 2007, Angewandte Chemie.

Rational Ligand Design for the Arylation of Hindered Primary Amines Guided by Reaction Progress Kinetic Analysis

S. Buchwald, D. Blackmond, Paula Ruiz-Castillo, 2015, Journal of the American Chemical Society.

Packed-bed reactors for continuous-flow C-N cross-coupling.

S. Buchwald, J. R. Naber, John R Naber, 2010, Angewandte Chemie.

Industrial-Scale Palladium-Catalyzed Coupling of Aryl Halides and Amines –A Personal Account

S. Buchwald, G. Mignani, C. Mauger, 2006 .

Use of precatalysts greatly facilitate palladium-catalyzed alkynylations in batch and continuous-flow conditions

S. Buchwald, W. Shu, S. Buchwald, 2011 .

Continuous-flow synthesis of biaryls enabled by multistep solid-handling in a lithiation/borylation/Suzuki-Miyaura cross-coupling sequence.

S. Buchwald, M. Oberli, Stephen L Buchwald, 2011, Angewandte Chemie.

Cross-coupling in flow.

Timothy Noël, Stephen L. Buchwald, S. Buchwald, 2011, Chemical Society reviews.

Concise palladium-catalyzed synthesis of dibenzodiazepines and structural analogues.

S. Buchwald, D. Tsvelikhovsky, S. Buchwald, 2011, Journal of the American Chemical Society.

Multistep microchemical synthesis enabled by microfluidic distillation.

Ryan L Hartman, Klavs F Jensen, Ryan L. Hartman, 2010, Angewandte Chemie.

Palladium‐Catalyzed Stille Cross‐Coupling Reaction of Aryl Chlorides using a Pre‐Milled Palladium Acetate and XPhos Catalyst System

S. Buchwald, J. R. Naber, S. Buchwald, 2008 .

Protein-Protein Cross-Coupling via Palladium-Protein Oxidative Addition Complexes from Cysteine Residues.

Ivan V. Buslov, S. Buchwald, B. Pentelute, 2020, Journal of the American Chemical Society.

Arylation Chemistry for Bioconjugation.

B. Pentelute, Chi Zhang, Stephen L Buchwald, 2019, Angewandte Chemie.

Divergent unprotected peptide macrocyclisation by palladium-mediated cysteine arylation† †Electronic supplementary information (ESI) available. See DOI: 10.1039/c6sc05454d Click here for additional data file.

S. Buchwald, B. Pentelute, Chi Zhang, 2016, Chemical science.

Oligonucleotide Bioconjugation with Bifunctional Palladium Reagents.

S. Buchwald, A. Loas, B. Pentelute, 2021, Angewandte Chemie.

Palladium Oxidative Addition Complexes for Peptide and Protein Cross-linking.

P. Dai, B. Pentelute, K. Kubota, 2018, Journal of the American Chemical Society.

Palladium-Protein Oxidative Addition Complexes by Amine-Selective Acylation.

Ivan V. Buslov, S. Buchwald, R. Raines, 2020, Journal of the American Chemical Society.

A palladium-catalyzed regiospecific synthesis of N-aryl benzimidazoles.

S. Buchwald, H. Nguyen, Xiaohua Huang, 2007, Angewandte Chemie.

Large Increase in External Quantum Efficiency by Dihedral Angle Tuning in a Sky‐Blue Thermally Activated Delayed Fluorescence Emitter

T. Van Voorhis, H. Chae, Markus Einzinger, 2019, Advanced Optical Materials.

Palladium-Catalyzed N-Arylation of Iminodibenzyls and Iminostilbenes with Aryl- and Heteroaryl Halides.

S. Buchwald, Wenliang Huang, S. Buchwald, 2016, Chemistry.

An Improved Catalyst System for Aromatic Carbon−Nitrogen Bond Formation: The Possible Involvement of Bis(Phosphine) Palladium Complexes as Key Intermediates

John P. Wolfe, Stephen L. Buchwald, S. Buchwald, 1996 .

The Regioselective Synthesis of Halophenols.

S. Buchwald, F. D. Rege, S. Buchwald, 1995 .

Rh-catalyzed asymmetric hydroformylation of functionalized 1,1-disubstituted olefins.

S. Buchwald, Xiao Wang, S. Buchwald, 2011, Journal of the American Chemical Society.

Highly N2-selective palladium-catalyzed arylation of 1,2,3-triazoles.

S. Buchwald, S. Ueda, Mingjuan Su, 2011, Angewandte Chemie.

Monodentate phosphines provide highly active catalysts for Pd-catalyzed C-N bond-forming reactions of heteroaromatic halides/amines and (H)N-heterocycles.

S. Buchwald, Ryan A. Altman, Takashi Ikawa, 2006, Angewandte Chemie.

Palladium-catalyzed amination reactions in flow: overcoming the challenges of clogging via acoustic irradiation

Jonathan P. McMullen, Klavs F. Jensen, Timothy Noël, 2011 .

A multiligand based Pd catalyst for C-N cross-coupling reactions.

S. Buchwald, B. Fors, S. Buchwald, 2010, Journal of the American Chemical Society.

Palladium-Catalyzed Coupling of Functionalized Primary and Secondary Amines with Aryl and Heteroaryl Halides: Two Ligands Suffice in Most Cases.

S. Buchwald, D. Maiti, Jaclyn L Henderson, 2010, Chemical science.

Expanding Pd-catalyzed C-N bond-forming processes: the first amidation of aryl sulfonates, aqueous amination, and complementarity with Cu-catalyzed reactions.

S. Buchwald, A. Klapars, Xiaohua Huang, 2003, Journal of the American Chemical Society.

CuH-Catalyzed Asymmetric Reduction of α,β-Unsaturated Carboxylic Acids to β-Chiral Aldehydes.

S. Buchwald, J. Bandar, Yujing Zhou, 2018, Journal of the American Chemical Society.

Synthesis of aryl sulfonamides via palladium-catalyzed chlorosulfonylation of arylboronic acids.

J. R. Debergh, N. Niljianskul, S. Buchwald, 2013, Journal of the American Chemical Society.

Development of an air-stable nickel precatalyst for the amination of aryl chlorides, sulfamates, mesylates, and triflates.

Nathaniel H. Park, Georgiy Teverovskiy, S. Buchwald, 2013, Organic letters.

Insights into amine binding to biaryl phosphine palladium oxidative addition complexes and reductive elimination from biaryl phosphine arylpalladium amido complexes via density functional theory.

S. Buchwald, Timothy E. Barder, S. Buchwald, 2007, Journal of the American Chemical Society.

Rational Development of Practical Catalysts for Aromatic Carbon−Nitrogen Bond Formation

John P. Wolfe, Stephen L. Buchwald, S. Buchwald, 1998 .

Palladium-catalyzed intermolecular coupling of aryl halides and amides.

S. Buchwald, Jingjun Yin, J. Yin, 2000, Organic letters.

Palladium-Catalyzed Aromatic Aminations with in situ Generated Aminostannanes

S. Buchwald, A. Guram, S. Buchwald, 1994 .

Twofold C-H functionalization: palladium-catalyzed ortho arylation of anilides.

S. Buchwald, Gordon Brasche, J. García-Fortanet, 2008, Organic letters.

Cp2TiCH2 complexes in synthetic applications

S. Buchwald, R. Grubbs, L. Clawson, 1983 .

A Nickel(0)-Catalyzed Process for the Transformation of Enynes to Bicyclic Cyclopentenones.

S. Buchwald, Minghui Zhang, Ming-hui Zhang, 1996, The Journal of organic chemistry.

CuH-Catalyzed Enantioselective Ketone Allylation with 1,3-Dienes: Scope, Mechanism, and Applications.

S. Buchwald, Peng Liu, Yang Yang, 2018, Journal of the American Chemical Society.

Palladium-catalyzed enantioselective alpha-arylation and alpha-vinylation of oxindoles facilitated by an axially chiral P-stereogenic ligand.

Ryan A. Altman, S. Buchwald, Alexander M Taylor, 2009, Journal of the American Chemical Society.

Use of a Droplet Platform To Optimize Pd-Catalyzed C–N Coupling Reactions Promoted by Organic Bases

S. Buchwald, K. Jensen, J. Dennis, 2019, Organic Process Research & Development.

Intramolecular palladium-catalyzed aryl amination and aryl amidation

S. Buchwald, J. Wolfe, R. Rennels, 1996 .

Reevaluation of the mechanism of the amination of aryl halides catalyzed by BINAP-ligated palladium complexes.

S. Buchwald, E. Strieter, S. Shekhar, 2006, Journal of the American Chemical Society.

Biaryl Monophosphine Ligands in Palladium-Catalyzed C-N Coupling: An Updated User's Guide.

S. Buchwald, Corin C. Wagen, Bryan T. Ingoglia, 2019, Tetrahedron.

Simple, efficient catalyst system for the palladium-catalyzed amination of aryl chlorides, bromides, and triflates.

S. Buchwald, J. Wolfe, Jingjun Yin, 2000, The Journal of organic chemistry.

Copper-catalyzed regiospecific synthesis of N-alkylbenzimidazoles.

S. Buchwald, N. Zheng, S. Buchwald, 2007, Organic letters.

Highly selective room-temperature copper-catalyzed C-N coupling reactions.

S. Buchwald, A. Shafir, S. Buchwald, 2006, Journal of the American Chemical Society.

Synthesis of N-aryl hydrazides by copper-catalyzed coupling of hydrazides with aryl iodides.

S. Buchwald, M. Wolter, A. Klapars, 2001, Organic letters.

Palladium-catalyzed asymmetric dearomatization of naphthalene derivatives.

S. Buchwald, F. Kessler, J. García-Fortanet, 2009, Journal of the American Chemical Society.

An Improved System for the Aqueous Lipshutz-Negishi Cross-Coupling of Alkyl Halides with Aryl Electrophiles.

S. Buchwald, B. O’Neill, Vasudev R. Bhonde, 2016, Angewandte Chemie.

Enantioselective Allylation Using Allene, a Petroleum Cracking Byproduct.

S. Buchwald, Yang Yang, Yujing Zhou, 2019, Journal of the American Chemical Society.

Rhodium-catalyzed asymmetric intramolecular hydroamination of unactivated alkenes.

S. Buchwald, Xiaoqiang Shen, S. Buchwald, 2009, Angewandte Chemie.

Copper-catalyzed selective hydroamination reactions of alkynes

S. Buchwald, Shi‐Liang Shi, S. Buchwald, 2014, Nature Chemistry.

Catalytic Method for the Reduction of Lactones to Lactols

Scott C. Berk, X. Verdaguer, S. Buchwald, 1995 .

Palladium-Catalyzed α-Arylation of Ketones

S. Buchwald, M. Palucki, S. Buchwald, 1997 .

The selective reaction of aryl halides with KOH: synthesis of phenols, aromatic ethers, and benzofurans.

S. Buchwald, Takashi Ikawa, K. Anderson, 2006, Journal of the American Chemical Society.

A rationally designed universal catalyst for Suzuki-Miyaura coupling processes.

S. Buchwald, J. R. Martinelli, Timothy E. Barder, 2004, Angewandte Chemie.

Highly Active Palladium Catalysts for Suzuki Coupling Reactions

S. Buchwald, J. Wolfe, Bryant H. Yang, 1999 .

Synthesis of 5,5-disubstituted butenolides based on a Pd-catalyzed gamma-arylation strategy.

S. Buchwald, Alan M. Hyde, S. Buchwald, 2009, Organic letters.

A Mild General Procedure for the One‐Pot Conversion of Amides to Aldehydes

S. Buchwald, S. Bower, K. A. Kreutzer, 1996 .

A Highly Active Catalyst for the Room-Temperature Amination and Suzuki Coupling of Aryl Chlorides.

Buchwald, Wolfe, S. Buchwald, 1999, Angewandte Chemie.

Palladium-catalyzed completely linear-selective Negishi cross-coupling of allylzinc halides with aryl and vinyl electrophiles.

S. Buchwald, Yang Yang, P. Cheong, 2013, Angewandte Chemie.

Ligand-controlled palladium-catalyzed regiodivergent Suzuki-Miyaura cross-coupling of allylboronates and aryl halides.

S. Buchwald, Yang Yang, S. Buchwald, 2013, Journal of the American Chemical Society.

Evidence for the formation and structure of palladacycles during Pd-catalyzed C-N bond formation with catalysts derived from bulky monophosphinobiaryl ligands.

S. Buchwald, E. Strieter, S. Buchwald, 2006, Angewandte Chemie.

Synthesis of Substituted Oxindoles from α-Chloroacetanilides via Palladium-Catalyzed C−H Functionalization

E. Hennessy, S. Buchwald, S. Buchwald, 2003 .

Palladium-catalyzed regioselective hydrodebromination of dibromoindoles: application to the enantioselective synthesis of indolodioxane U86192A.

S. Buchwald, Junghyun Chae, S. Buchwald, 2004, The Journal of organic chemistry.

An improved protocol for the Pd-catalyzed alpha-arylation of aldehydes with aryl halides.

S. Buchwald, Rúben Martín, R. Martín, 2008, Organic letters.

A General Method for the Direct α‐Arylation of Aldehydes with Aryl Bromides and Chlorides

S. Buchwald, Rúben Martín, R. Martín, 2007 .

A Titanocene-Catalyzed Intramolecular Ene Reaction: Cycloisomerization of Enynes and Dienynes

S. Buchwald, S. Sturla, Natasha M. Kablaoui, 1999 .

Negishi coupling of secondary alkylzinc halides with aryl bromides and chlorides.

Chong Han, S. Buchwald, 2009, Journal of the American Chemical Society.

CuH-Catalyzed Regio- and Enantioselective Hydrocarboxylation of Allenes: Toward Carboxylic Acids with Acyclic Quaternary Centers.

S. Buchwald, Shengyu Feng, S. Buchwald, 2021, Journal of the American Chemical Society.

Diastereoselective Synthesis of γ-Butyrolactones from Enones Mediated or Catalyzed by a Titanocene Complex

S. Buchwald, Natasha M. Kablaoui, Frederick A. Hicks, 1996 .

Scope of the Intramolecular Titanocene-Catalyzed Pauson−Khand Type Reaction1

S. Buchwald, Natasha M. Kablaoui, Frederick A. Hicks, 1999 .

Titanocene-Catalyzed Cyclocarbonylation of Enynes to Cyclopentenones

S. Buchwald, Natasha M. Kablaoui, Frederick A. Hicks, 1996 .

CuH-Catalyzed Olefin Functionalization: From Hydroamination to Carbonyl Addition.

S. Buchwald, Richard Y. Liu, S. Buchwald, 2020, Accounts of chemical research.

Copper-catalyzed asymmetric conjugate reduction as a route to novel beta-azaheterocyclic acid derivatives.

S. Buchwald, Y. Aye, Matthew P. Rainka, 2004, Proceedings of the National Academy of Sciences of the United States of America.

Conjugate Reduction of α,β-Unsaturated Carbonyl Compounds Catalyzed by a Copper Carbene Complex

S. Buchwald, J. Sadighi, Valdas Jurkauskas, 2003 .

Palladium-Catalyzed Intramolecular C-H Difluoroalkylation: Synthesis of Substituted 3,3-Difluoro-2- oxindoles

S. Buchwald, 2015 .

Copper-Catalyzed Enantioselective Addition of Styrene-Derived Nucleophiles to Imines Enabled by Ligand-Controlled Chemoselective Hydrocupration

S. Buchwald, Yang Yang, Ian B. Perry, 2016, Journal of the American Chemical Society.

Palladium-Catalyzed Hydroxylation of Aryl and Heteroaryl Halides Enabled by the Use of a Palladacycle Precatalyst

S. Buchwald, C. Cheung, S. Buchwald, 2014, The Journal of organic chemistry.

A Practical Electrophilic Nitrogen Source for the Synthesis of Chiral Primary Amines by Copper-Catalyzed Hydroamination.

S. Buchwald, Sheng-Mei Guo, Jeffrey C Yang, 2018, Journal of the American Chemical Society.

Enantioselective Hydroalkenylation of Olefins with Enol Sulfonates Enabled by Dual Copper Hydride and Palladium Catalysis.

S. Buchwald, James Levi Knippel, Gustavo M. Borrajo-Calleja, 2021, Journal of the American Chemical Society.

Direct 11CN-Labeling of Unprotected Peptides via Palladium-Mediated Sequential Cross-Coupling Reactions.

S. Buchwald, J. Hooker, Hong Geun Lee, 2017, Journal of the American Chemical Society.

Selective palladium-catalyzed arylation of ammonia: synthesis of anilines as well as symmetrical and unsymmetrical di- and triarylamines.

S. Buchwald, D. Surry, S. Buchwald, 2007, Journal of the American Chemical Society.

A direct approach to amines with remote stereocenters by enantioselective CuH-catalysed reductive relay hydroamination

S. Buchwald, Shaolin Zhu, N. Niljianskul, 2015, Nature chemistry.

Selective, zirconium-mediated cross-coupling of alkynes: the synthesis of isomerically pure 1,3-dienes and 1,4-diiodo-1,3-dienes

S. Buchwald, R. Nielsen, S. Buchwald, 1989 .

Asymmetric Hydroarylation of Vinylarenes Using a Synergistic Combination of CuH and Pd Catalysis

S. Buchwald, Michael T Pirnot, Stig D. Friis, 2016, Journal of the American Chemical Society.

An improved catalyst for the asymmetric arylation of ketone enolates.

S. Buchwald, A. Chieffi, J. Ahman, 2002, Journal of the American Chemical Society.

Asymmetric Cu-Catalyzed 1,4-Dearomatization of Pyridines and Pyridazines without Preactivation of the Heterocycle or Nucleophile.

S. Buchwald, Sheng-Mei Guo, Michael W. Gribble, 2018, Journal of the American Chemical Society.

A Combined Zirconocene Benzyne−Palladium Cross-Coupling Route to Substituted Biphenyls and Terphenyls

S. Buchwald, A. Peat, D. Pérez, 1999 .

Copper-catalyzed N-arylation of imidazoles and benzimidazoles.

S. Buchwald, E. Koval, Ryan A. Altman, 2007, The Journal of organic chemistry.

Expedited palladium-catalyzed amination of aryl nonaflates through the use of microwave-irradiation and soluble organic amine bases.

S. Buchwald, K. Anderson, Rachel E. Tundel, 2006, The Journal of organic chemistry.

Efficient pd-catalyzed amination of heteroaryl halides.

S. Buchwald, M. D. Charles, P. Schultz, 2005, Organic letters.

Mechanistic insights into the Pd(BINAP)-catalyzed amination of aryl bromides: kinetic studies under synthetically relevant conditions.

S. Buchwald, E. Strieter, D. Blackmond, 2002, Journal of the American Chemical Society.

New ammonia equivalents for the Pd-catalyzed amination of aryl halides.

S. Buchwald, X. Huang, S. Buchwald, 2001, Organic letters.

Use of polymer-supported dialkylphosphinobiphenyl ligands for palladium-catalyzed amination and Suzuki reactions.

S. Buchwald, C. Parrish, S. Buchwald, 2001, The Journal of organic chemistry.

An improved method for the palladium-catalyzed amination of aryl iodides.

S. Buchwald, Mayssam H. Ali, M. H. Ali, 2001, The Journal of organic chemistry.

Sequential N-Arylation of Primary Amines as a Route To Alkyldiarylamines

S. Buchwald, M. C. Harris, Oliver Geis, 1999 .

Palladium-catalyzed amination of aryl halides and sulfonates

S. Buchwald, Bryant H. Yang, S. Buchwald, 1999 .

Room Temperature Catalytic Amination of Aryl Iodides

S. Buchwald, J. Wolfe, S. Buchwald, 1997 .

Mild Palladium-Catalyzed Cyanation of (Hetero)aryl Halides and Triflates in Aqueous Media

S. Buchwald, Daniel T. Cohen, S. Buchwald, 2015, Organic letters.

A Fungal-Selective Cytochrome bc1 Inhibitor Impairs Virulence and Prevents the Evolution of Drug Resistance.

Raja R Srinivas, S. Buchwald, B. Tidor, 2016, Cell chemical biology.

Copper-Catalyzed Enantioselective Hydroamination of Alkenes.

Richard Y. Liu, S. Buchwald, 2019, Organic syntheses; an annual publication of satisfactory methods for the preparation of organic chemicals.

The Synthesis of Aminopyridines: A Method Employing Palladium-Catalyzed Carbon-Nitrogen Bond Formation.

S. Buchwald, S. Wagaw, S. Buchwald, 1996, The Journal of organic chemistry.

Cu-catalyzed Goldberg and Ullmann reactions of aryl halides using chelating N- and O-based ligands

S. Buchwald, Ryan A. Altman, S. Buchwald, 2007, Nature Protocols.

Use of a "Catalytic" Cosolvent, N,N-Dimethyl Octanamide, Allows the Flow Synthesis of Imatinib with no Solvent Switch.

S. Buchwald, D. Niu, Jeffrey C Yang, 2016, Angewandte Chemie.

Group 4 Metal Complexes of Benzynes, Cycloalkynes, Acyclic Alkynes, and Alkenes

S. Buchwald, R. Nielsen, S. Buchwald, 1988 .

One-pot sequential Cu-catalyzed reduction and Pd-catalyzed arylation of silyl enol ethers.

S. Buchwald, Junghyun Chae, J. Yun, 2004, Organic letters.

A general and mild copper-catalyzed arylation of diethyl malonate.

E. Hennessy, S. Buchwald, S. Buchwald, 2002, Organic letters.

A GENERAL COPPER-CATALYZED SYNTHESIS OF DIARYL ETHERS

S. Buchwald, J. Marcoux, A. S. Doye, 1997 .

Titanocene-Catalyzed Asymmetric Ketone Hydrosilylation: The Effect of Catalyst Activation Protocol and Additives on the Reaction Rate and Enantioselectivity

S. Buchwald, J. Yun, S. Buchwald, 1999 .

Enantioselective hydrosilylation of ketones with a chiral titanocene catalyst

S. Buchwald, B. Schiøtt, A. Gutiérrez, 1994 .

Enantioselective β-arylation of ketones enabled by lithiation/borylation/1,4-addition sequence under flow conditions.

S. Buchwald, W. Shu, S. Buchwald, 2012, Angewandte Chemie.

Continuous-flow synthesis of 3,3-disubstituted oxindoles by a palladium-catalyzed α-arylation/alkylation sequence.

S. Buchwald, Pengfei Li, S. Buchwald, 2011, Angewandte Chemie.

Suzuki-Miyaura cross-coupling reactions in flow: multistep synthesis enabled by a microfluidic extraction.

S. Kuhn, K. Jensen, T. Noël, 2011, Angewandte Chemie.

Synthesis of medium ring nitrogen heterocycles via a tandem copper-catalyzed C-N bond formation-ring-expansion process.

Artis Klapars, S. Buchwald, Stephen L Buchwald, 2004, Journal of the American Chemical Society.

Direct and selective elimination of specific prions and amyloids by 4,5-dianilinophthalimide and analogs

Andrew D. Steele, Martin L. Duennwald, J. King, 2008, Proceedings of the National Academy of Sciences.

Visible Light-Mediated (Hetero)aryl Amination Using Ni(II) Salts and Photoredox Catalysis in Flow: A Synthesis of Tetracaine.

S. Buchwald, Michael T Pirnot, Boyoung Y. Park, 2020, The Journal of organic chemistry.

Synthesis of solid 2-pyridylzinc reagents and their application in Negishi reactions.

S. Buchwald, P. Knochel, Sebastian Bernhardt, 2013, Organic letters.

Pd-catalyzed intermolecular amidation of aryl halides: the discovery that xantphos can be trans-chelating in a palladium complex.

S. Buchwald, Jingjun Yin, S. Buchwald, 2002, Journal of the American Chemical Society.

Efficient Synthesis of Well-Defined, High Molecular Weight, and Processible Polyanilines under Mild Conditions via Palladium-Catalyzed Amination

S. Buchwald, Xiao-xiang Zhang, J. Sadighi, 2000 .

A highly active palladium catalyst system for the arylation of anilines

S. Buchwald, J. Sadighi, M. C. Harris, 1998 .

An extremely active catalyst for the Negishi cross-coupling reaction.

S. Buchwald, Jacqueline E. Milne, S. Buchwald, 2004, Journal of the American Chemical Society.

Mechanistic Insight Facilitates Discovery of a Mild and Efficient Copper-Catalyzed Dehydration of Primary Amides to Nitriles Using Hydrosilanes.

S. Buchwald, Richard Y. Liu, Minwoo Bae, 2018, Journal of the American Chemical Society.

Water-Soluble Palladium Reagents for Cysteine S-Arylation under Ambient Aqueous Conditions.

Bradley L. Pentelute, Stephen L. Buchwald, S. Buchwald, 2017, Organic letters.

Cis difunctionalization of cyclic olefins with use of organozirconium intermediates

S. Buchwald, G. Cuny, A. Gutiérrez, 1991 .

Stibathiolanes: synthesis, solid-state structure, and solution behavior

W. M. Davis, S. Buchwald, R. Nielsen, 1991 .

An efficient one-pot method for the preparation of polysubstituted benzothiophenes

S. Buchwald, Qun Fang, S. Buchwald, 1989 .

Sequential Cu-catalyzed amidation-base-mediated camps cyclization: a two-step synthesis of 2-Aryl-4-quinolones from o-halophenones.

S. Buchwald, K. Anderson, Carrie P. Jones, 2007, The Journal of organic chemistry.

Enantioselective Hydrocarbamoylation of Alkenes

Yuyang Dong, Shengyu Feng, S. Buchwald, 2022, Angewandte Chemie.

Palladium-catalyzed amination of unprotected halo-7-azaindoles.

S. Buchwald, Jaclyn L Henderson, Sarah M. McDermott, 2010, Organic letters.

Synthesis of indolines via a domino Cu-catalyzed amidation/cyclization reaction.

S. Buchwald, A. Minatti, S. Buchwald, 2008, Organic letters.

Cascade palladium catalysis: a predictable and selectable regiocontrolled synthesis of N-arylbenzimidazoles.

S. Buchwald, N. Jui, S. Buchwald, 2013, Angewandte Chemie.

CuH-Catalyzed Regioselective Intramolecular Hydroamination for the Synthesis of Alkyl-Substituted Chiral Aziridines.

S. Buchwald, Jeffrey C Yang, Haoxuan Wang, 2017, Journal of the American Chemical Society.

Amine Additives Greatly Expand the Scope of Asymmetric Hydrosilylation of Imines.

S. Buchwald, X. Verdaguer, Udo E W Lange, 1998, Angewandte Chemie.

A method for the asymmetric hydrosilylation of N-aryl imines.

S. Buchwald, M. C. Hansen, S. Buchwald, 2000, Organic letters.

Efficient kinetic resolution in the asymmetric hydrosilylation of imines of 3-substituted indanones and 4-substituted tetralones.

S. Buchwald, J. Yun, S. Buchwald, 2000, The Journal of organic chemistry.

Synthesis of NPS R-568 utilizing titanium-catalyzed asymmetric hydrosilylation

S. Buchwald, M. Hansen, Marcus C. Hansen, 1999 .

Short Enantioselective Total Syntheses of the Piperidine Alkaloids (S)-Coniine and (2R,6R)-trans-Solenopsin A via Catalytic Asymmetric Imine Hydrosilylation.

S. Buchwald, Matthew T. Reding, S. Buchwald, 1998, The Journal of organic chemistry.

Preparation of Novel Titanium Complexes Bearing o-Phosphinophenol Ligands

W. M. Davis, S. Buchwald, C. A. Willoughby, 1996 .

An Inexpensive Air-Stable Titanium-Based System for the Conversion of Esters to Primary Alcohols

S. Buchwald, Matthew T. Reding, S. Buchwald, 1995 .

Titanocene-Catalyzed Reduction of Esters Using Polymethylhydrosiloxane as the Stoichiometric Reductant

S. Buchwald, Scott C. Berk, K. Barr, 1994 .

Asymmetric hydrogenation of unfunctionalized trisubstituted olefins with a chiral titanocene catalyst

S. Buchwald, R. Broene, S. Buchwald, 1993 .

Rationale behind the resistance of dialkylbiaryl phosphines toward oxidation by molecular oxygen.

S. Buchwald, Timothy E. Barder, S. Buchwald, 2007, Journal of the American Chemical Society.