Pascal Villa

发表

Use of a fluorescent polarization based high throughput assay to identify new calmodulin ligands.

C. Wermuth, J. Haiech, C. Pigault, 2006, Biochimica et biophysica acta.

Design, synthesis, and pharmacological evaluation of N-acylhydrazones and novel conformationally constrained compounds as selective and potent orally active phosphodiesterase-4 inhibitors.

J. Bourguignon, N. Romeiro, M. Martins, 2012, Journal of medicinal chemistry.

Identification by high-throughput screening of inhibitors of Schistosoma mansoni NAD(+) catabolizing enzyme.

E. Kellenberger, D. Rognan, J. Haiech, 2010, Bioorganic & medicinal chemistry.

Chemical Library Screening and Structure-Function Relationship Studies Identify Bisacodyl as a Potent and Selective Cytotoxic Agent Towards Quiescent Human Glioblastoma Tumor Stem-Like Cells

Jacques Haiech, Samir Mameri, Maria Zeniou, 2015, PloS one.

Screening and Structure-Function Relationship Studies Identify Bisacodyl as a Potent and Selective Cytotoxic Agent Towards Quiescent Human Glioblastoma Tumor Stem-Like Cells

M. Junier, S. Kahn, E. El-Habr, 2019 .

Overexpression of the MSK1 Kinase in Patients With Chronic Lung Allograft Dysfunction and Its Confirmed Role in a Murine Model

L. Reber, N. Frossard, M. Stern, 2020, Transplantation.

Antiallodynic action of phosphodiesterase inhibitors in a mouse model of peripheral nerve injury

M. Barrot, J. Bourguignon, S. Hugel, 2021, Neuropharmacology.

Design, Synthesis and Biological Evaluation of Arylpyridin-2-yl Guanidine Derivatives and Cyclic Mimetics as Novel MSK1 Inhibitors. An Application in an Asthma Model

D. Rognan, F. Bihel, J. Bourguignon, 2021, Molecules.

Clearance of persistent hepatitis C virus infection using a claudin-1-targeting monoclonal antibody

Lars Kaderali, Ralf Bartenschlager, Patrick Pessaux, 2015, Nature Biotechnology.

Nile Red-Based GPCR Ligands as Ultrasensitive Probes of the Local Lipid Microenvironment of the Receptor.

A. Klymchenko, D. Bonnet, P. Villa, 2020, ACS chemical biology.

Treating leishmaniasis in Amazonia, part 2: Multi-target evaluation of widely used plants to understand medicinal practices.

M. Ginouves, G. Prévot, E. Bourreau, 2022, Journal of ethnopharmacology.

Liposomal encapsulation of trans-crocetin enhances oxygenation in patients with COVID-19-related ARDS receiving mechanical ventilation

X. Pivot, O. Collange, Z. Huang, 2021, Journal of Controlled Release.