论文信息 - Solvent-free preparation of primary imines from (2-hydroxyaryl)ketones - 字舞流文

Solvent-free preparation of primary imines from (2-hydroxyaryl)ketones

Primary imines can be readily prepared from (2-hydroxyaryl)ketones by reaction with ammonium iodide and piperidine under solvent-free conditions.

P. Perlmutter | Neeranat Thienthong | Y. Bergman

[1] Y. Mizuno,et al. Process development of potassium channel opener, TCV-295, based on convenient ring formation of 2H-1,3-benzoxazine and selective N-oxidation of the pyridyl moiety , 2001 .

[2] G. Rothenberg,et al. Understanding solid/solid organic reactions. , 2001, Journal of the American Chemical Society.

[3] S. Yamamoto,et al. Synthesis and biological activity of novel 1,3-benzoxazine derivatives as K+ channel openers. , 1996, Chemical and pharmaceutical bulletin.

[4] M. Poiana,et al. Ketimines From Ketones and Ammonia , 1988 .

[5] B. Davis. The syntheses of 4‐aminobutanoic acid‐2,2‐2H2 and ‐4,4‐2H2 and progabide‐2,2‐2H2 and ‐4,4‐2H2 , 1987 .

[6] T. Heffner,et al. 1,3-Dialkyl-4-(iminoarylmethyl)-1H-pyrazol-5-ols. A series of novel potential antipsychotic agents. , 1987, Journal of medicinal chemistry.

[7] K. Shepard,et al. Imino-bridged heterocycles. IV: A facile synthesis of sulfenimines derived from diaryl ketones , 1985 .

[8] K. Grellmann,et al. The photochemical formation of ketimines from aromatic ketoximes , 1975 .

[9] A. Schönberg,et al. Darstellung von Iminen durch Einwirkung von flüssigem Ammoniak auf geminale Dihalogenide , 1966 .