Enantioselective synthesis of phosphinyl peptidomimetics via an asymmetric Michael reaction of phosphinic acids with acrylate derivatives

[1]  H. Cristau,et al.  A Convenient One-Pot Synthesis of Phosphino-Dipeptide Analogs , 2001 .

[2]  V. Dive,et al.  Convenient synthesis and diversification of dehydroalaninyl phosphinic peptide analogues. , 2001, Organic Letters.

[3]  Yves Dumond,et al.  Synthesis of Monosubstituted Phosphinic Acids: Palladium-Catalyzed Cross-Coupling Reactions of Anilinium Hypophosphite , 2001 .

[4]  T. Burke,et al.  Use of a Heck reaction for the synthesis of a new alpha-azido phosphotyrosyl mimetic suitably protected for peptide synthesis. , 2000, The Journal of organic chemistry.

[5]  P. Coric,et al.  Phosphinic derivatives as new dual enkephalin-degrading enzyme inhibitors: synthesis, biological properties, and antinociceptive activities. , 2000, Journal of medicinal chemistry.

[6]  V. Dive,et al.  Potent and selective inhibition of zinc aminopeptidase A (EC 3.4.11.7, APA) by glutamyl aminophosphinic peptides: importance of glutamyl aminophosphinic residue in the P1 position. , 2000, Biochemistry.

[7]  V. Dive,et al.  Protection of the Hydroxyphosphinyl Function of Phosphinic Dipeptides by Adamantyl. Application to the Solid-Phase Synthesis of Phosphinic Peptides. , 1996, The Journal of organic chemistry.

[8]  F. Checler,et al.  Development of the First Potent and Selective Inhibitor of the Zinc Endopeptidase Neurolysin Using a Systematic Approach Based on Combinatorial Chemistry of Phosphinic Peptides* , 1996, The Journal of Biological Chemistry.

[9]  M. Sibi,et al.  A new chiral oxazolidinone derived from diphenylalaninol. Aldol, alkylation, and diels-alder reactions , 1995 .

[10]  Paul A. Bartlett,et al.  Differential binding energy: a detailed evaluation of the influence of hydrogen-bonding and hydrophobic groups on the inhibition of thermolysin by phosphorus-containing inhibitors , 1991 .

[11]  K. James,et al.  A versatile route to substituted phosphinic acids , 1990 .

[12]  T. Shioiri,et al.  New Methods and Reagents in Organic Synthesis. 14. A Simple Efficient Preparation of Methyl Esters with Trimethylsilyldiazomethane (TMSCHN2) and Its Application to Gas Chromatographic Analysis of Fatty Acids , 1981 .

[13]  N. Hashimoto,et al.  有機合成の新しい方法と試薬 XIV トリメチルシリルジアゾメタン(TMSCHN 2 )を用いるメチルエステルの簡単で効果的な調製と,脂肪酸のガスクロマトグラフィー分析への応用 , 1981 .

[14]  Davidr . Evans,et al.  New Silicon-Phosphorus Reagents in Organic Synthesis. Carbonyl and Conjugate Addition Reactions of Silicon Phosphite Esters and Related Systems , 1978 .

[15]  S. J. Fitch Synthesis of Hypophosphite Esters from Orthocarbonyl Compounds , 1964 .

[16]  H. Schmidt Über eine neue Gruppe von organischen Phosphorverbindungen , 1948 .