Comparison of Succinimidyl [125I]Iodobenzoate with Iodogen Iodination Methods to Study Pharmacokinetics and ADME of Biotherapeutics
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[1] Hua Bai,et al. Pharmacokinetics, Tissue Distribution and Excretion of Recombinant Human Parathyroid Hormone 1–84 in Animals , 2013, Cell Biochemistry and Biophysics.
[2] J. Ozer,et al. Decreased Subcutaneous Bioavailability of an Oxyntomodulin Analog in a Controlled Release Formulation could be Caused by Skin Metabolism in Rats , 2012 .
[3] Afshin Safavi,et al. Ligand Binding Assays in the 21st Century Laboratory: Recommendations for Characterization and Supply of Critical Reagents , 2012, The AAPS Journal.
[4] Lee Goodwin,et al. Bioanalytical approaches to analyzing peptides and proteins by LC--MS/MS. , 2011, Bioanalysis.
[5] M. Khalil,et al. Molecular SPECT Imaging: An Overview , 2011, International journal of molecular imaging.
[6] Heather Myler,et al. Bioanalytical Approaches to Quantify “Total” and “Free” Therapeutic Antibodies and Their Targets: Technical Challenges and PK/PD Applications Over the Course of Drug Development , 2011, The AAPS Journal.
[7] Y. Vugmeyster,et al. Biodistribution of [125I]-labeled therapeutic proteins: application in protein drug development beyond oncology. , 2010, Journal of pharmaceutical sciences.
[8] D. Rajalingam,et al. Trichloroacetic acid‐induced protein precipitation involves the reversible association of a stable partially structured intermediate , 2009, Protein science : a publication of the Protein Society.
[9] B. Gorovits. Antidrug Antibody Assay Validation: Industry Survey Results , 2009, The AAPS Journal.
[10] M. Schlumberger,et al. 131I Effective Half-Life and Dosimetry in Thyroid Cancer Patients , 2008, Journal of Nuclear Medicine.
[11] Denise M O'Hara,et al. Critical ligand binding reagent preparation/selection: When specificity depends on reagents , 2007, The AAPS Journal.
[12] R. Aebersold,et al. Mass Spectrometry and Protein Analysis , 2006, Science.
[13] A. A. van Well,et al. Changes in the secondary structure of proteins labeled with 125I: CD spectroscopy and enzymatic activity studies , 2005 .
[14] Binodh DeSilva,et al. Recommendations for the Bioanalytical Method Validation of Ligand-Binding Assays to Support Pharmacokinetic Assessments of Macromolecules , 2003, Pharmaceutical Research.
[15] S. Jurisson,et al. Modification of the structure of a metallopeptide: Synthesis and biological evaluation of 111in-labeled DOTA-conjugated rhenium-cyclized α-MSH analogues , 2002 .
[16] S. Jurisson,et al. α–melanocyte‐stimulating hormone peptide analogs labeled with technetium‐99m and indium‐111 for malignant melanoma targeting , 2002, Cancer.
[17] S. Jurisson,et al. Modification of the structure of a metallopeptide: synthesis and biological evaluation of (111)In-labeled DOTA-conjugated rhenium-cyclized alpha-MSH analogues. , 2002, Journal of medicinal chemistry.
[18] A. Khalaj,et al. A new and simple synthesis of N‐succinimidyl‐4‐[127/125I]iodobenzoate involving a microwave ‐ accelerated iodination step , 2001 .
[19] G. V. van Dongen,et al. Optimal quality (131)I-monoclonal antibodies on high-dose labeling in a large reaction volume and temporarily coating the antibody with IODO-GEN. , 2001, Journal of nuclear medicine : official publication, Society of Nuclear Medicine.
[20] L. Potempa,et al. Biodistribution and clearance of 125I-labeled C-reactive protein and 125I-labeled modified C-reactive protein in CD-1 mice. , 1998, Drug metabolism and disposition: the biological fate of chemicals.
[21] M. Juweid,et al. Advantage of residualizing radiolabels for an internalizing antibody against the B-cell lymphoma antigen, CD22 , 1997, Cancer Immunology, Immunotherapy.
[22] S. Strand,et al. Optimization of radioiodination and biotinylation of monoclonal antibody chimeric BR96: an indirect labeling using N-succinimidyl-3-(tri-n-butylstannyl)benzoate conjugate. , 1996, Cancer biotherapy & radiopharmaceuticals.
[23] D. Wilbur,et al. Development of a stable radioiodinating reagent to label monoclonal antibodies for radiotherapy of cancer. , 1989, Journal of nuclear medicine : official publication, Society of Nuclear Medicine.
[24] M. Zalutsky,et al. Radiohalogenation of a monoclonal antibody using an N-succinimidyl 3-(tri-n-butylstannyl)benzoate intermediate. , 1988, Cancer research.
[25] R. Baughman,et al. Pharmacokinetics and tissue distribution of recombinant human tumor necrosis factor-alpha in mice. , 1988, Drug metabolism and disposition: the biological fate of chemicals.
[26] M. Zalutsky,et al. A method for the radiohalogenation of proteins resulting in decreased thyroid uptake of radioiodine. , 1987, International journal of radiation applications and instrumentation. Part A, Applied radiation and isotopes.
[27] V. Cody,et al. Rat liver iodothyronine monodeiodinase. Evaluation of the iodothyronine ligand-binding site. , 1986, The Journal of biological chemistry.
[28] L. Osterman. Methods of protein and nucleic acid research , 1984 .
[29] R. Coleman,et al. Comparison of iodine monochloride and modified chloramine-T radioiodination for in vivo protein studies. , 1977, Journal of Laboratory and Clinical Medicine.
[30] W. Hunter,et al. The labelling of proteins to high specific radioactivities by conjugation to a 125I-containing acylating agent. , 1973, The Biochemical journal.