Improved synthesis of some commonly used PET radioligands by the use of [11C]methyl triflate.

[1]  A. Brownell,et al.  Substituted 3-phenyltropane analogs of cocaine: synthesis, inhibition of binding at cocaine recognition sites, and positron emission tomography imaging. , 1993, Journal of medicinal chemistry.

[2]  C. Halldin,et al.  [11C] beta-CIT, a cocaine analogue. Preparation, autoradiography and preliminary PET investigations. , 1993, Nuclear medicine and biology.

[3]  Alan A. Wilson,et al.  Synthesis of a radiotracer for studying dopamine uptake sites in vivo using PET: 2β‐carbomethoxy‐3β‐(4‐fluorophenyl)‐[N‐11C‐methyl]tropane ([11C]CFT or [11C]WIN‐35,428) , 1993 .

[4]  D. Jewett,et al.  A simple synthesis of [11C]methyl triflate. , 1992, International journal of radiation applications and instrumentation. Part A, Applied radiation and isotopes.

[5]  P B Hoffer,et al.  [123I]-2 beta-carbomethoxy-3 beta-(4-iodophenyl)tropane: high-affinity SPECT radiotracer of monoamine reuptake sites in brain. , 1991, Journal of medicinal chemistry.

[6]  K. Någren,et al.  Preparation of the antioestrogenic compound N-[methyl-11C]-toremifene for the study of oestrogen-receptor positive tumors in vivo , 1991 .

[7]  F I Carroll,et al.  Synthesis, ligand binding, QSAR, and CoMFA study of 3 beta-(p-substituted phenyl)tropane-2 beta-carboxylic acid methyl esters. , 1991, Journal of medicinal chemistry.

[8]  J. Neumeyer,et al.  Synthesis and receptor binding of N-substituted tropane derivatives. High-affinity ligands for the cocaine receptor. , 1991, Journal of medicinal chemistry.

[9]  M. Schwaiger,et al.  Synthesis and preliminary evaluation of carbon-11-meta-hydroxyephedrine: a false transmitter agent for heart neuronal imaging. , 1990, Journal of nuclear medicine : official publication, Society of Nuclear Medicine.

[10]  B. Långström,et al.  The preparation of 11C-methyl iodide and its use in the synthesis of 11C-methyl-L-methionine. , 1976, The International journal of applied radiation and isotopes.

[11]  R. L. Clarke,et al.  Compounds affecting the central nervous system. 4. 3 Beta-phenyltropane-2-carboxylic esters and analogs. , 1973, Journal of medicinal chemistry.

[12]  P. N. Craig,et al.  3-Substituted Tropane Derivatives. I. The Synthesis and Stereochemistry of the Tropane-3-carboxylic Acids and Their Esters. A Comparison of Positional Isomers in the Tropane Series1 , 1962 .

[13]  G. Sedvall,et al.  Synthesis of carbon-11 labelled SCH 39166, a new selective dopamine D-1 receptor ligand, and preliminary PET investigations. , 1991, International journal of radiation applications and instrumentation. Part A, Applied radiation and isotopes.

[14]  G. Sedvall,et al.  Carbon-11 labelling of eticlopride in two different positions--a selective high-affinity ligand for the study of dopamine D-2 receptors using PET. , 1990, International journal of radiation applications and instrumentation. Part A, Applied radiation and isotopes.

[15]  A. Wolf,et al.  Synthesis of suicide inhibitors of monoamine oxidase: Carbon‐11 labeled clorgyline, L‐deprenyl and D‐deprenyl , 1988 .

[16]  D. Comar,et al.  Synthesis of methyl iodide-11 C and formaldehyde-11 C. , 1977, The International journal of applied radiation and isotopes.