Regioselective formylation of 1,3-disubstituted benzenes through in situ lithiation

[1]  D. B. Collum,et al.  Regioselective lithium diisopropylamide-mediated ortholithiation of 1-chloro-3-(trifluoromethyl)benzene: role of autocatalysis, lithium chloride catalysis, and reversibility. , 2011, Journal of the American Chemical Society.

[2]  E. Fillion,et al.  Sc(OTf)3-catalyzed conjugate allylation of alkylidene Meldrum's acids. , 2009, Organic letters.

[3]  P. Jeschke,et al.  alpha-fluorinated ethers as "exotic" entity in medicinal chemistry. , 2007, Mini reviews in medicinal chemistry.

[4]  J. Findlay,et al.  Benzothienyloxy phenylpropanamines, novel dual inhibitors of serotonin and norepinephrine reuptake. , 2004, Bioorganic & medicinal chemistry letters.

[5]  Antonio Ramirez,et al.  Formation of benzynes from 2,6-dihaloaryllithiums: mechanistic basis of the regioselectivity. , 2004, Journal of the American Chemical Society.

[6]  Y. Itoh,et al.  Fluorinated carbonyl and olefinic compounds: basic character and asymmetric catalytic reactions. , 2004, Chemical reviews.

[7]  Anne‐Sophie Castanet,et al.  Selectivities in reactions of organolithium reagents with unprotected 2-halobenzoic acids. , 2003, Organic letters.

[8]  J. Mortier,et al.  ortho-metalation of unprotected 3-bromo and 3-chlorobenzoic acids with hindered lithium dialkylamides. , 2003, The Journal of organic chemistry.

[9]  A. Scott.  Biosynthesis: Aromatic Polyketides, Isoprenoids, Alkaloids. Topics in Current Chemistry. Vol. 209 Edited by Finian J. Leeper (University of Cambridge) and John C. Vederas (University of Alberta). Springer-Verlag: Berlin, Heidelberg, New York. 2000. viii + 247 pp. $159.00. ISBN 3-540-66573-0. , 2000 .

[10]  D. B. Collum,et al.  Are n-BuLi/TMEDA-Mediated Arene Ortholithiations Directed? Substituent-Dependent Rates, Substituent-Independent Mechanisms , 2000 .

[11]  W. Dmowski,et al.  A site selective functionalisation of 1,3-bis(trifluoromethyl)benzene , 1998 .

[12]  D. B. Collum,et al.  Is N,N,N',N'-tetramethylethylenediamine a good ligand for lithium? , 1992 .

[13]  A. Bridges,et al.  Fluorine as an ortho-directing group in aromatic metalation: A two step preparation of substituted benzo[b]thiophene-2-carboxylates , 1992 .

[14]  Victor Snieckus,et al.  Directed ortho metalation. Tertiary amide and O-carbamate directors in synthetic strategies for polysubstituted aromatics , 1990 .

[15]  J. Stadelhofer,et al.  Industrial Aromatic Chemistry , 1988 .