Diastereoselective Synthesis of the Acid Part of a New Muscarinic M3 Receptor Antagonist

[1]  Y. Ogino,et al.  Discovery of a muscarinic M3 receptor antagonist with high selectivity for M3 over M2 receptors among 2-[(1S,3S)-3-sulfonylaminocyclopentyl]phenylacetamide derivatives. , 2000, Bioorganic & medicinal chemistry.

[2]  M. Shindo,et al.  1,1,4,7,10-10-Hexamethyltriethylenetetramine: a reagent to enhance the rate of alkylation reaction of the lithium enolate of 1-tetralone with alkyl halides , 1999 .

[3]  Y. Ogino,et al.  Stereoselective synthesis of a new muscarinic M3 receptor antagonist, J-104129. , 1999, Bioorganic & medicinal chemistry letters.

[4]  B. Lipshutz,et al.  A convenient, efficient method for conjugate reductions using catalytic quantities of Cu(I) , 1998 .

[5]  S. Takano,et al.  Enantiocontrolled Synthesis of Two Amino Acids; (S)-Glutamic Acid and (S)-2-Aminoadipic Acid , 1994 .

[6]  S. Takano,et al.  Non-hazardous preparation of 3-acetoxy- and 3-oxodicyclopentadienes , 1994 .

[7]  K. Inomata,et al.  Concise enatio- and stereo-controlled synthesis of (+)-equilenin using chiral cyclopentadienone synthon , 1990 .

[8]  E. Keinan,et al.  Highly chemoselective palladium-catalyzed conjugate reduction of .alpha.,.beta.-unsaturated carbonyl compounds with silicon hydrides and zinc chloride cocatalyst , 1986 .

[9]  D. Seebach,et al.  (α-Alkylation of α-heterosubstituted carboxylic acids without racemization : EPC-syntheses of tertiary alcohols and thiols☆☆☆ , 1984 .

[10]  T. Saegusa,et al.  Synthesis of .alpha.,.beta.-unsaturated carbonyl compounds by palladium(II)-catalyzed dehydrosilylation of silyl enol ethers , 1978 .