Optimization of the potency and pharmacokinetic properties of a macrocyclic ghrelin receptor agonist (Part I): Development of ulimorelin (TZP-101) from hit to clinic.
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Martin Brassard | D. Veber | S. Beauchemin | A. Mathieu | M. Vezina | É. Marsault | M. L. Peterson | H. Hoveyda | R. Gagnon | A. Landry | Zhigang Wang | K. Benakli | S. Beaubien | C. Saint-Louis | M. Brassard | J. Pinault | L. Ouellet | S. Bhat | M. Ramaseshan | Xiaowen Peng | L. Foucher | Patrick Bhérer | G. Fraser | Shridhar Bhat | Daniel F Veber | Eric Marsault | Axel P Mathieu | Mark L Peterson | Hamid R Hoveyda | René Gagnon | Martin Vézina | Carl Saint-Louis | Annick Landry | Jean-François Pinault | Luc Ouellet | Sophie Beauchemin | Sylvie Beaubien | Kamel Benakli | Zhigang Wang | Mahesh Ramaseshan | Patrick Bhérer | Laurence Foucher | Xiaowen Peng | Graeme L Fraser | M. Peterson
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