New and efficient synthesis of 3-arylquinazolin-4(1H)-ones and biologically important N-fused tetracycles based on N-(2-carboxyphenyl)oxalamide

[1]  S. Pollock Indian , 2021, How Literatures Begin.

[2]  S. Grimme,et al.  Acid‐Catalyzed Rearrangements of 3‐Aryloxirane‐2‐Carboxamides: Novel DFT Mechanistic Insights , 2020, ChemistryOpen.

[3]  A. Gubaidullin,et al.  Facile synthesis of 2-carboxanilido-3-arylquinazolin-4-ones from N1-(2-carboxyphenyl)-N2-(aryl)oxalamides , 2019, Tetrahedron Letters.

[4]  V. Mamedov,et al.  A new and efficient method for the synthesis of 3-(2-nitrophenyl)pyruvic acid derivatives and indoles based on the Reissert reaction , 2018, Tetrahedron Letters.

[5]  M. Ghavidel,et al.  A Domino Process for the Sustainable Synthesis of Quinazolin-4(3H)-ones with Direct Chemo- and Regioselective Bromination , 2018, Synlett.

[6]  Tun-Cheng Chien,et al.  Regioselective synthesis and biological evaluation of N-substituted 2-aminoquinazolin-4-ones. , 2018, Organic & biomolecular chemistry.

[7]  V. Mamedov,et al.  Simple synthesis of 3-hydroxyquinolines via Na2S2O4-mediated reductive cyclization of (2-(2-nitrophenyl)oxiran-1-yl)(aryl)methanones (o-nitrobenzalacetophenone oxides) , 2017 .

[8]  Indresh Kumar,et al.  Synthesis of Quinazolinones, Imidazo[1,2‐c]quinazolines and Imidazo[4,5‐c]quinolines through Tandem Reductive Amination of Aryl Halides and Oxidative Amination of C(sp3)–H Bonds , 2017 .

[9]  Tian-Qi Wei,et al.  I2/CHP‐Mediated Oxidative Coupling of 2‐Aminobenzamides and Isocyanides: Access to 2‐Aminoquinazolinones , 2016 .

[10]  S. Katsyuba,et al.  A novel acid-catalyzed rearrangement of 2-substituted-3-(2-nitrophenyl)oxiranes for the synthesis of di- and mono-oxalamides , 2016 .

[11]  Zhiyong Wang,et al.  Copper-catalyzed radical methylation/C-H amination/oxidation cascade for the synthesis of quinazolinones. , 2015, The Journal of organic chemistry.

[12]  Dinesh Kumar,et al.  Convenient synthesis of 2,3-disubstituted quinazolin-4(3H)-ones and 2-styryl-3-substituted quinazolin-4(3H)-ones: applications towards the synthesis of drugs , 2015 .

[13]  K. Gnanasekaran,et al.  Pyrazoloquinazolinones and pyrazolopyridopyrimidinones by a sequential N-acylation–SNAr reaction , 2015 .

[14]  M. Pal,et al.  Glyoxylic acid in the reaction of isatoic anhydride with amines: a rapid synthesis of 3-(un)substituted quinazolin-4(3H)-ones leading to rutaecarpine and evodiamine , 2014 .

[15]  H. Neumann,et al.  A convenient palladium-catalyzed carbonylative synthesis of 4(3H)-quinazolinones from 2-bromoformanilides and organo nitros with Mo(CO)6 as a multiple promoter , 2014 .

[16]  Ye-Gao Chen,et al.  Ammonium Chloride–Catalyzed One-Pot Synthesis of 4(3H)-Quinazolinones Under Solvent-Free Conditions , 2014 .

[17]  O. Jacquet,et al.  Complete Catalytic Deoxygenation of CO2 into Formamidine Derivatives , 2013 .

[18]  Hitesh B. Jalani,et al.  An efficient, greener, and solvent-free one-pot multicomponent synthesis of 3-substituted quinazolin-4(3H)ones and thienopyrimidin-4(3H)ones ☆ , 2012 .

[19]  Yongwen Jiang,et al.  Synthesis of 3-substituted and 2,3-disubstituted quinazolinones via Cu-catalyzed aryl amidation. , 2012, Organic letters.

[20]  Ke-Fang Yang,et al.  Green Synthesis of Quinazolinone Derivatives Catalyzed by Iodine in Ionic Liquid , 2012 .

[21]  Yuyuan Wang,et al.  Copper‐Catalyzed Domino Synthesis of Benzimidazo[2,1‐b]quin‐ azolin‐12(6H)‐ones Using Cyanamide as a Building Block , 2012 .

[22]  Tingting Zhang,et al.  Aluminium Nitrate–Catalyzed One-Pot Synthesis of 4(3H)-Quinazolinones by a Three-Component Coupling of Anthranilic Acid, Amines, and Ortho Esters , 2011 .

[23]  J. Yadav,et al.  Eco‐friendly, solvent‐free novel one‐pot, three‐component synthesis of quinazolinones at ambient temperature catalyzed by silica gel‐supported phosphomolybdic acid , 2010 .

[24]  P. Molina,et al.  Preparation of Fused Tetracyclic Quinazolinones by Combinations of Aza‐Wittig Methodologies and CuI‐Catalysed Heteroarylation Processes , 2009 .

[25]  Michael G. Yang,et al.  Synthesis of 3-substituted-4(3H)-quinazolinones via HATU-mediated coupling of 4-hydroxyquinazolines with amines. , 2009, Organic letters.

[26]  A. de Meijere,et al.  ortho-Lithiophenyl isocyanide: a versatile precursor for 3H-quinazolin-4-ones and 3H-quinazolin-4-thiones. , 2009, Organic letters.

[27]  C. Rabia,et al.  A Microwave-Assisted and Heteropolyacids-Catalysed Cyclocondensation Reaction for the Synthesis of4(3H)-Quinazolinones , 2008, Molecules.

[28]  K. Lam,et al.  Microwave-mediated heterocyclization to benzimidazo[2,1-b]quinazolin-12(5H)-ones. , 2007, The Journal of organic chemistry.

[29]  K. Mukkanti,et al.  Silica gel/FeCl3: An efficient and recyclable heterogenous catalyst for one step synthesis of 4(3H)-quinazolinones under solvent free conditions , 2006 .

[30]  K. C. Mahesh,et al.  Lanthanum(III) nitrate hexahydrate or p-toluenesulfonic acid catalyzed one-pot synthesis of 4(3H)-quinazolinones under solvent-free conditions , 2006 .

[31]  K. Rad‐Moghadam,et al.  Convergent One‐Pot Synthesis of 3‐Substituted Quinazolin‐4(3H)‐ones under Solvent‐Free Conditions , 2006 .

[32]  I. Mohammadpoor‐Baltork,et al.  Bi(TFA)3–[nbp]FeCl4: a new, efficient and reusable promoter system for the synthesis of 4(3H)-quinazolinone derivatives , 2006 .

[33]  D. Shi,et al.  An efficient synthesis of quinazoline derivatives with the aid of low‐valent titanium reagent , 2005 .

[34]  Ruifang Chen,et al.  Synthesis of 3,4‐Dihydropyrimidine‐2(1H)‐thiones and Quinazolin‐4(3H)‐ones over Yb(III)‐Resin Catalyst Under Solvent‐free Conditions , 2005 .

[35]  M. Dabiri,et al.  One‐Pot Synthesis of Mono‐ and Disubstituted (3H)‐Quinazolin‐4‐ones in Dry Media Under Microwave Irradiation , 2005 .

[36]  D. Shi,et al.  Facile Synthesis of Substituted Quinazolin‐4‐(3H)‐ones Using Low‐Valence Titanium Reagent , 2004 .

[37]  K. Rad‐Moghadam,et al.  A CONVENIENT SYNTHESIS OF SUBSTITUTED QUINAZOLIN-4(3H)-ONES UNDER MICROWAVE AND SOLVENT-FREE CONDITIONS , 2004 .

[38]  J. Banerjee,et al.  Silica-supported Sodium Hydrogen Sulfate and Amberlyst-15 : Two Efficient Heterogeneous Catalysts for Single-step Synthesis of 4(3H)-Quinazolinones from Anthranilic Acid, Ortho Esters, and Amines under Solvent Free Conditions , 2004 .

[39]  W. Su,et al.  Pd2(dba)3/P(i-BuNCH2CH2)3N-catalyzed Stille cross-coupling of aryl chlorides. , 2004, Organic letters.

[40]  D. Shi,et al.  Synthesis of quinazolin-4(3H)-ones and 1,2-dihydroquinazolin-4(3H)-ones with the aid of a low-valent titanium reagent , 2003 .

[41]  Limin Wang,et al.  Yb(OTf)3-Catalyzed One-Pot Synthesis of Quinazolin-4(3H)-ones from Anthranilic­ Acid, Amines and Ortho Esters (or Formic Acid) in Solvent-Free Conditions , 2003 .

[42]  R. Houghten,et al.  A traceless approach for the parallel solid-phase synthesis of 2-(arylamino)quinazolinones. , 2002, The Journal of organic chemistry.

[43]  P. Knochel,et al.  Preparation of polyfunctional heterocycles using highly functionalized aminated arylmagnesium reagents as versatile scaffolds. , 2002, Organic letters.

[44]  Y. Yamauchi,et al.  Preparation of a Useful Synthetic Precursor, 2-Substituted 4(3H)-Quinazolinone: Directed Lithiation and N3-Deprotection of 3-t-Butoxycarbonyl-4(3H)-quinazolinone , 2002 .

[45]  A. Da Settimo,et al.  Synthesis, in vitro antiproliferative activity and DNA-interaction of benzimidazoquinazoline derivatives as potential anti-tumor agents. , 2001, Farmaco.

[46]  A. Kamal,et al.  Chemoenzymatic synthesis of pyrrolo[2,1-b]quinazolinones: lipase-catalyzed resolution of vasicinone. , 2001, The Journal of organic chemistry.

[47]  M. Zaki,et al.  REACTION OF ISATOIC ANHYDRIDE WITH BIFUNCTIONAL REAGENTS: SYNTHESIS OF SOME NEW QUINAZOLONE FUSED HETEROCYCLES, 2-SUBSTITUTED ANILINOHETEROCYCLIC DERIVATIVES AND OTHER RELATED COMPOUNDS , 2001 .

[48]  J. Bergman,et al.  Synthesis and Reactions of some 2-Vinyl-3H-quinazolin-4-ones , 2000 .

[49]  Rui Yang,et al.  A concise and efficient solid-phase synthesis of 2-amino-4(3H)-quinazolinones , 2000 .

[50]  O. Leoni,et al.  Reactivity Range of a Chiral 1,3-Oxazolidine-2-thione Obtained from Vegetable Source through Chemo-enzymatic Processing , 2000 .

[51]  Minakata,et al.  Lactone synthesis based on atom transfer carbonylation , 2000, Organic letters.

[52]  O. Leoni,et al.  Chemo-enzymatic preparation from renewable resources of enantiopure 1,3-oxazolidine-2-thiones , 1999 .

[53]  M. Ueno,et al.  Catalytic asymmetric synthesis of febrifugine and isofebrifugine , 1999 .

[54]  D. Obrecht,et al.  Solid-Phase Synthesis of 3H-Quinazolin-4-ones Based on an Aza Wittig-Mediated annulation Strategy , 1998 .

[55]  S. S. Ibrahim,et al.  Synthesis and Biological Activities of Some New Fully Fused Quinazoline Derivatives. , 1998 .

[56]  B. Roth,et al.  Novel nonpeptide CCK-B antagonists: design and development of quinazolinone derivatives as potent, selective, and orally active CCK-B antagonists. , 1998, Journal of medicinal chemistry.

[57]  X. Dai,et al.  Synthesis and Resolution of Quinazolinone Atropisomeric Phosphine Ligands(,). , 1998, The Journal of organic chemistry.

[58]  N. Liverton,et al.  Nonpeptide glycoprotein IIb/IIIa inhibitors: substituted quinazolinediones and quinazolinones as potent fibrinogen receptor antagonists. , 1998, Bioorganic & medicinal chemistry letters.

[59]  C. Lamberth,et al.  Regio- and Stereoselective Alkoxycarbonylmethylenation of Partially Saturated Heterobicyclic Compounds: First Synthesis of 2-Substituted Quinazoline-8-acetic Acid Esters , 1998 .

[60]  Y. Kurogi,et al.  Synthesis and hypolipidemic activities of novel 2-[4-[diethoxyphosphoryl)methyl]phenyl]quinazolines and 4(3H)-quinazolinones. , 1996, Journal of medicinal chemistry.

[61]  M. Sato,et al.  Studies on antiulcer agents. IV. Antiulcer effects of 2-benzylthio5,6,7,8-tetrahydro-4(3H)-quinazolinones and related compounds. , 1995, Chemical & pharmaceutical bulletin.

[62]  J. F. Wolfe,et al.  Synthesis and anticonvulsant activity of some new 2-substituted 3-aryl-4(3H)-quinazolinones. , 1990, Journal of medicinal chemistry.

[63]  C. Bird,et al.  The thermal rearrangement of 2-aryl-1-cyanoindazol-3-ones , 1987 .

[64]  J. Baldwin,et al.  Rules for ring closure. , 1977, Ciba Foundation symposium.

[65]  R. W. Harper,et al.  Benzimidazo[2,1-b]quinazolin-12-ones. A new class of potent immunosuppressive compounds. , 1971, Journal of medicinal chemistry.

[66]  R. W. Harper,et al.  Methods for preparing benzimidazo[2,1-b] quinazolin-12-ones and related compounds , 1971 .

[67]  D. J. Brown,et al.  The Dimroth rearrangement. XI. Simple examples in the quinazoline series , 1968 .

[68]  C. W. Bird The rearrangement of 2-cyano-1-phenylpyrazole derivatives , 1965 .

[69]  B. R. Baker,et al.  AN ANTIMALARIAL ALKALOID FROM HYDRANGEA. XVIII. DERIVATIVES OF 4-PYRIMIDONE , 1953 .

[70]  S. Gordon,et al.  AN ANTIMALARIAL ALKALOID FROM HYDRANGEA. II. ISOLATION , 1952 .

[71]  J. Mead,et al.  An alkaloid with high antimalarial activity from Dichroa febrifuga. , 1947, Journal of the American Chemical Society.

[72]  T. Chou,et al.  Ch'ang Shan, a Chinese Antimalarial Herb. , 1946, Science.