Synthesis and evaluation of potent and selective human V1a receptor antagonists as potential ligands for PET or SPECT imaging.
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Craig F. Ferris | Michael J. Brownstein | Ned D. Heindel | C. Ferris | M. Brownstein | N. Simon | C. Guillon | Shi-fang Lu | Neal G. Simon | Christophe Guillon | Graham B Jones | Michael S Placzek | N. Heindel | Shi-fang Lu | Graham Jones | Michael Placzek | Karine Fabio | Carl J. Lacey | C. J. Lacey | Karine M Fabio
[1] D. Swaab,et al. Increased Arginine Vasopressin mRNA Expression in the Human Hypothalamus in Depression: A Preliminary Report , 2006, Biological Psychiatry.
[2] P. Joyce,et al. Reduction in basal afternoon plasma ACTH during early treatment of depression with fluoxetine , 2001, Psychopharmacology.
[3] F. Holsboer,et al. V1 vasopressin receptor antisense oligodeoxynucleotide into septum reduces vasopressin binding, social discrimination abilities, and anxiety-related behavior in rats , 1995, The Journal of neuroscience : the official journal of the Society for Neuroscience.
[4] Larry J Young,et al. Profound Impairment in Social Recognition and Reduction in Anxiety-Like Behavior in Vasopressin V1a Receptor Knockout Mice , 2004, Neuropsychopharmacology.
[5] H. Anisman,et al. Corticotropin-Releasing Hormone, Arginine Vasopressin, Gastrin-Releasing Peptide, and Neuromedin B Alterations in Stress-Relevant Brain Regions of Suicides and Control Subjects , 2006, Biological Psychiatry.
[6] H. Coenen,et al. Nucleophilic 18F-fluorination of heteroaromatic iodonium salts with no-carrier-added [18F]fluoride. , 2007, Journal of the American Chemical Society.
[7] O. Solin,et al. Radiosynthesis and evaluation of [18F]Selectfluor bis(triflate). , 2010, Angewandte Chemie.
[8] Li Di,et al. High throughput artificial membrane permeability assay for blood-brain barrier. , 2003, European journal of medicinal chemistry.
[9] J. Maffrand,et al. Nonpeptide vasopressin receptor antagonists: development of selective and orally active V1a, V2 and V1b receptor ligands. , 2002, Progress in brain research.
[10] Gary W. Caldwell,et al. Optimization In Drug Discovery In Vitro Methods , 2010 .
[11] T. Dinan,et al. Vasopressin as a target for antidepressant development: an assessment of the available evidence. , 2002, Journal of affective disorders.
[12] D. Swaab,et al. Increased number of vasopressin- and oxytocin-expressing neurons in the paraventricular nucleus of the hypothalamus in depression. , 1996, Archives of general psychiatry.
[13] A. Konings. FREE-RADICAL PATHOLOGY - AN INTRODUCTION , 1987 .
[14] R. Derijk,et al. Anxious–Retarded Depression: Relation with Plasma Vasopressin and Cortisol , 2003, Neuropsychopharmacology.
[15] R. Landgraf,et al. Born to be Anxious: Neuroendocrine and Genetic Correlates of Trait Anxiety in HAB Rats , 2003, Stress.
[16] I. Greguric,et al. Synthesis and evaluation of novel radioiodinated benzamides for malignant melanoma. , 2007, Journal of medicinal chemistry.
[17] N. Toschi,et al. Reduction of Hypothalamic Vasopressinergic Hyperdrive Contributes to Clinically Relevant Behavioral and Neuroendocrine Effects of Chronic Paroxetine Treatment in a Psychopathological Rat Model , 2003, Neuropsychopharmacology.
[18] M. Timsit-Berthier,et al. [Study of the stress response: role of anxiety, cortisol and DHEAs]. , 2002, L'Encephale.
[19] T. Insel,et al. Facilitation of Affiliation and Pair-Bond Formation by Vasopressin Receptor Gene Transfer into the Ventral Forebrain of a Monogamous Vole , 2001, The Journal of Neuroscience.
[20] B. Långström,et al. Synthesis of 3-[(2S)-azetidin-2-ylmethoxy]-5-[11C]-methylpyridine, an analogue of A-85380, via a Stille coupling , 2002 .
[21] P. Veinante,et al. Vasopressin and Oxytocin Excite Distinct Neuronal Populations in the Central Amygdala , 2005, Science.
[22] B. Faller,et al. High-throughput permeability pH profile and high-throughput alkane/water log P with artificial membranes. , 2001, Journal of medicinal chemistry.
[23] Nicolas Singewald,et al. A Hypomorphic Vasopressin Allele Prevents Anxiety-Related Behavior , 2009, PloS one.
[24] C. Nemeroff,et al. Psychoneuroendocrinology of depression. Hypothalamic-pituitary-adrenal axis. , 1998, The Psychiatric clinics of North America.
[25] F. Holsboer,et al. Endocrine disturbances in depression , 2005, Journal of endocrinological investigation.
[26] G. Kerkhof,et al. Weak 24-h periodicity of body temperature and increased plasma vasopressin in melancholic depression , 2001, European Neuropsychopharmacology.
[27] Gary W. Caldwell,et al. Optimization in Drug Discovery , 2014, Methods in Pharmacology and Toxicology.
[28] D. Rujescu,et al. Candidate genes of anxiety-related behavior in HAB/LAB rats and mice: Focus on vasopressin and glyoxalase-I , 2007, Neuroscience & Biobehavioral Reviews.
[29] J. Hooker,et al. Synthesis of [11C]SSR149415 and preliminary imaging studies using positron emission tomography. , 2010, Bioorganic & medicinal chemistry letters.
[30] S. Volpi,et al. Vasopressinergic Regulation of the Hypothalamic Pituitary Adrenal Axis and Stress Adaptation , 2004, Stress.
[31] R. Landgraf. The involvement of the vasopressin system in stress-related disorders. , 2006, CNS & neurological disorders drug targets.
[32] C. Ferris,et al. Azetidinones as vasopressin V1a antagonists. , 2007, Bioorganic & medicinal chemistry.
[33] F. Zufall,et al. Social motivation is reduced in vasopressin 1b receptor null mice despite normal performance in an olfactory discrimination task , 2004, Hormones and Behavior.
[34] K. Zwinderman,et al. Depression with above-normal plasma vasopressin: Validation by relations with family history of depression and mixed anxiety and retardation , 2006, Psychiatry Research.
[35] N. Meanwell. Synopsis of some recent tactical application of bioisosteres in drug design. , 2011, Journal of medicinal chemistry.
[36] T. Dinan,et al. Anatomy of melancholia: focus on hypothalamic–pituitary–adrenal axis overactivity and the role of vasopressin , 2005, Journal of anatomy.
[37] R. Ring. The central vasopressinergic system: examining the opportunities for psychiatric drug development. , 2005, Current pharmaceutical design.
[38] S. Adelstein,et al. [125I/127I]iodoHoechst 33342: synthesis, DNA binding, and biodistribution. , 1996, Journal of medicinal chemistry.
[39] Praveen Kulkarni,et al. Imaging the neural circuitry and chemical control of aggressive motivation , 2008, BMC Neuroscience.
[40] C. Ferris,et al. Orally active vasopressin V1a receptor antagonist, SRX251, selectively blocks aggressive behavior , 2006, Pharmacology Biochemistry and Behavior.
[41] F. Holsboer,et al. Glucocorticoids and depression. , 1999, Bailliere's best practice & research. Clinical endocrinology & metabolism.
[42] V. Wiegant,et al. Plasma Levels of Arginine Vasopressin Elevated in Patients with Major Depression , 1997, Neuropsychopharmacology.
[43] M. Thibonnier,et al. Molecular cloning, sequencing, and functional expression of a cDNA encoding the human V1a vasopressin receptor. , 1994, The Journal of biological chemistry.
[44] Shuiyu Lu,et al. Fast and high-yield microreactor syntheses of ortho-substituted [(18)F]fluoroarenes from reactions of [(18)F]fluoride ion with diaryliodonium salts. , 2010, The Journal of organic chemistry.
[45] F. Holsboer,et al. Alterations in Central Neuropeptide Expression, Release, and Receptor Binding in Rats Bred for High Anxiety: Critical Role of Vasopressin , 2004, Neuropsychopharmacology.
[46] C. Wotjak,et al. Septal vasopressin modulates anxiety-related behaviour in rats , 1996, Neuroscience Letters.
[47] Dennis K. Taylor,et al. 1,2-dioxines containing tethered hydroxyl functionality as convenient precursors for pyran syntheses. , 2005, The Journal of organic chemistry.