Discovery of a new potent inhibitor of mushroom tyrosinase (Agaricus bisporus) containing 4-(4-hydroxyphenyl)piperazin-1-yl moiety.
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A. Fais | F. Pintus | S. Vittorio | M. P. Germanò | R. Gitto | A. Rapisarda | L. De Luca | M. R. Buemi | Salvatore Mirabile | Maria R Buemi
[1] T. Langer,et al. A Combination of Pharmacophore and Docking‐based Virtual Screening to Discover new Tyrosinase Inhibitors , 2020, Molecular informatics.
[2] M. Rafiq,et al. Hydroxyl substituted benzoic acid/cinnamic acid derivatives: Tyrosinase inhibitory kinetics, anti-melanogenic activity and molecular docking studies. , 2019, Bioorganic & medicinal chemistry letters.
[3] A. Fishman,et al. Exploiting the 1-(4-fluorobenzyl)piperazine fragment for the development of novel tyrosinase inhibitors as anti-melanogenic agents: Design, synthesis, structural insights and biological profile. , 2019, European journal of medicinal chemistry.
[4] J. Choi,et al. Phlorotannins with Potential Anti-Tyrosinase and Antioxidant Activity Isolated from the Marine Seaweed Ecklonia stolonifera , 2019, Antioxidants.
[5] F. Delogu,et al. Synthesis, molecular docking and cholinesterase inhibitory activity of hydroxylated 2-phenylbenzofuran derivatives. , 2019, Bioorganic chemistry.
[6] Mahmud Tareq Hassan Khan,et al. A comprehensive review on tyrosinase inhibitors , 2019, Journal of enzyme inhibition and medicinal chemistry.
[7] V. Namasivayam,et al. Inhibitors of Melanogenesis: An Updated Review. , 2018, Journal of medicinal chemistry.
[8] Ximing Xu,et al. Correction: design, synthesis and evaluation of cinnamic acid ester derivatives as mushroom tyrosinase inhibitors , 2018, MedChemComm.
[9] A. Fishman,et al. Targeting Tyrosinase: Development and Structural Insights of Novel Inhibitors Bearing Arylpiperidine and Arylpiperazine Fragments. , 2018, Journal of medicinal chemistry.
[10] E. Pieroni,et al. Novel 2-pheynlbenzofuran derivatives as selective butyrylcholinesterase inhibitors for Alzheimer’s disease , 2018, Scientific Reports.
[11] Ximing Xu,et al. Design, synthesis and evaluation of cinnamic acid ester derivatives as mushroom tyrosinase inhibitors. , 2018, MedChemComm.
[12] S. Vilar,et al. New insights into highly potent tyrosinase inhibitors based on 3-heteroarylcoumarins: Anti-melanogenesis and antioxidant activities, and computational molecular modeling studies. , 2017, Bioorganic & medicinal chemistry.
[13] M. Kanteev,et al. Chemical exploration of 4-(4-fluorobenzyl)piperidine fragment for the development of new tyrosinase inhibitors. , 2017, European journal of medicinal chemistry.
[14] Fengyan Wu,et al. Molecular docking studies and biological evaluation of 1,3,4-thiadiazole derivatives bearing Schiff base moieties as tyrosinase inhibitors. , 2016, Bioorganic chemistry.
[15] S. Ferro,et al. Searching for indole derivatives as potential mushroom tyrosinase inhibitors , 2015, Journal of enzyme inhibition and medicinal chemistry.
[16] R. Shimmon,et al. Development of hydroxylated naphthylchalcones as polyphenol oxidase inhibitors: Synthesis, biochemistry and molecular docking studies. , 2015, Bioorganic chemistry.
[17] A. Scala,et al. From NMDA receptor antagonists to discovery of selective σ₂ receptor ligands. , 2014, Bioorganic & medicinal chemistry.
[18] Arbakariya B. Ariff,et al. Depigmenting Effect of Kojic Acid Esters in Hyperpigmented B16F1 Melanoma Cells , 2012, Journal of biomedicine & biotechnology.
[19] L. Mondello,et al. Betula pendula leaves: polyphenolic characterization and potential innovative use in skin whitening products. , 2012, Fitoterapia.
[20] B. Dijkstra,et al. Crystal structure of Agaricus bisporus mushroom tyrosinase: identity of the tetramer subunits and interaction with tropolone. , 2011, Biochemistry.
[21] R. Citraro,et al. Development of 3-substituted-1H-indole derivatives as NR2B/NMDA receptor antagonists. , 2009, Bioorganic & medicinal chemistry.
[22] R. Bentley. From miso, saké and shoyu to cosmetics: a century of science for kojic acid. , 2006, Natural product reports.
[23] S. Kim,et al. Solid-phase synthesis of kojic acid-tripeptides and their tyrosinase inhibitory activity, storage stability, and toxicity. , 2004, Bioorganic & medicinal chemistry letters.
[24] Alessandro Pedretti,et al. VEGA – An open platform to develop chemo-bio-informatics applications, using plug-in architecture and script programming , 2004, J. Comput. Aided Mol. Des..
[25] L. Xie,et al. Inhibitory Effects of Some Flavonoids on the Activity of Mushroom Tyrosinase , 2003, Biochemistry (Moscow).
[26] Y. Murata,et al. Mushroom Tyrosinase Inhibitory Activity of Esculetin Isolated from Seeds of Euphorbia lathyris L. , 2003, Bioscience, biotechnology, and biochemistry.
[27] M. Soni,et al. Evaluation of health aspects of kojic acid in food. , 2001, Regulatory toxicology and pharmacology : RTP.
[28] I. Kubo,et al. Flavonols from Heterotheca inuloides: tyrosinase inhibitory activity and structural criteria. , 2000, Bioorganic & medicinal chemistry.
[29] S. Rhee,et al. Inhibition of tyrosinase by green tea components. , 1999, Life sciences.
[30] J N Rodríguez-López,et al. Tyrosinase: a comprehensive review of its mechanism. , 1995, Biochimica et biophysica acta.