Discovery of a new potent inhibitor of mushroom tyrosinase (Agaricus bisporus) containing 4-(4-hydroxyphenyl)piperazin-1-yl moiety.

[1]  T. Langer,et al.  A Combination of Pharmacophore and Docking‐based Virtual Screening to Discover new Tyrosinase Inhibitors , 2020, Molecular informatics.

[2]  M. Rafiq,et al.  Hydroxyl substituted benzoic acid/cinnamic acid derivatives: Tyrosinase inhibitory kinetics, anti-melanogenic activity and molecular docking studies. , 2019, Bioorganic & medicinal chemistry letters.

[3]  A. Fishman,et al.  Exploiting the 1-(4-fluorobenzyl)piperazine fragment for the development of novel tyrosinase inhibitors as anti-melanogenic agents: Design, synthesis, structural insights and biological profile. , 2019, European journal of medicinal chemistry.

[4]  J. Choi,et al.  Phlorotannins with Potential Anti-Tyrosinase and Antioxidant Activity Isolated from the Marine Seaweed Ecklonia stolonifera , 2019, Antioxidants.

[5]  F. Delogu,et al.  Synthesis, molecular docking and cholinesterase inhibitory activity of hydroxylated 2-phenylbenzofuran derivatives. , 2019, Bioorganic chemistry.

[6]  Mahmud Tareq Hassan Khan,et al.  A comprehensive review on tyrosinase inhibitors , 2019, Journal of enzyme inhibition and medicinal chemistry.

[7]  V. Namasivayam,et al.  Inhibitors of Melanogenesis: An Updated Review. , 2018, Journal of medicinal chemistry.

[8]  Ximing Xu,et al.  Correction: design, synthesis and evaluation of cinnamic acid ester derivatives as mushroom tyrosinase inhibitors , 2018, MedChemComm.

[9]  A. Fishman,et al.  Targeting Tyrosinase: Development and Structural Insights of Novel Inhibitors Bearing Arylpiperidine and Arylpiperazine Fragments. , 2018, Journal of medicinal chemistry.

[10]  E. Pieroni,et al.  Novel 2-pheynlbenzofuran derivatives as selective butyrylcholinesterase inhibitors for Alzheimer’s disease , 2018, Scientific Reports.

[11]  Ximing Xu,et al.  Design, synthesis and evaluation of cinnamic acid ester derivatives as mushroom tyrosinase inhibitors. , 2018, MedChemComm.

[12]  S. Vilar,et al.  New insights into highly potent tyrosinase inhibitors based on 3-heteroarylcoumarins: Anti-melanogenesis and antioxidant activities, and computational molecular modeling studies. , 2017, Bioorganic & medicinal chemistry.

[13]  M. Kanteev,et al.  Chemical exploration of 4-(4-fluorobenzyl)piperidine fragment for the development of new tyrosinase inhibitors. , 2017, European journal of medicinal chemistry.

[14]  Fengyan Wu,et al.  Molecular docking studies and biological evaluation of 1,3,4-thiadiazole derivatives bearing Schiff base moieties as tyrosinase inhibitors. , 2016, Bioorganic chemistry.

[15]  S. Ferro,et al.  Searching for indole derivatives as potential mushroom tyrosinase inhibitors , 2015, Journal of enzyme inhibition and medicinal chemistry.

[16]  R. Shimmon,et al.  Development of hydroxylated naphthylchalcones as polyphenol oxidase inhibitors: Synthesis, biochemistry and molecular docking studies. , 2015, Bioorganic chemistry.

[17]  A. Scala,et al.  From NMDA receptor antagonists to discovery of selective σ₂ receptor ligands. , 2014, Bioorganic & medicinal chemistry.

[18]  Arbakariya B. Ariff,et al.  Depigmenting Effect of Kojic Acid Esters in Hyperpigmented B16F1 Melanoma Cells , 2012, Journal of biomedicine & biotechnology.

[19]  L. Mondello,et al.  Betula pendula leaves: polyphenolic characterization and potential innovative use in skin whitening products. , 2012, Fitoterapia.

[20]  B. Dijkstra,et al.  Crystal structure of Agaricus bisporus mushroom tyrosinase: identity of the tetramer subunits and interaction with tropolone. , 2011, Biochemistry.

[21]  R. Citraro,et al.  Development of 3-substituted-1H-indole derivatives as NR2B/NMDA receptor antagonists. , 2009, Bioorganic & medicinal chemistry.

[22]  R. Bentley From miso, saké and shoyu to cosmetics: a century of science for kojic acid. , 2006, Natural product reports.

[23]  S. Kim,et al.  Solid-phase synthesis of kojic acid-tripeptides and their tyrosinase inhibitory activity, storage stability, and toxicity. , 2004, Bioorganic & medicinal chemistry letters.

[24]  Alessandro Pedretti,et al.  VEGA – An open platform to develop chemo-bio-informatics applications, using plug-in architecture and script programming , 2004, J. Comput. Aided Mol. Des..

[25]  L. Xie,et al.  Inhibitory Effects of Some Flavonoids on the Activity of Mushroom Tyrosinase , 2003, Biochemistry (Moscow).

[26]  Y. Murata,et al.  Mushroom Tyrosinase Inhibitory Activity of Esculetin Isolated from Seeds of Euphorbia lathyris L. , 2003, Bioscience, biotechnology, and biochemistry.

[27]  M. Soni,et al.  Evaluation of health aspects of kojic acid in food. , 2001, Regulatory toxicology and pharmacology : RTP.

[28]  I. Kubo,et al.  Flavonols from Heterotheca inuloides: tyrosinase inhibitory activity and structural criteria. , 2000, Bioorganic & medicinal chemistry.

[29]  S. Rhee,et al.  Inhibition of tyrosinase by green tea components. , 1999, Life sciences.

[30]  J N Rodríguez-López,et al.  Tyrosinase: a comprehensive review of its mechanism. , 1995, Biochimica et biophysica acta.