Inhibition of gamma-secretase by the CK1 inhibitor IC261 does not depend on CK1delta.
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[1] K. Baumann,et al. NSAID-derived gamma-secretase modulators. Part III: Membrane anchoring. , 2009, Bioorganic & medicinal chemistry letters.
[2] H. Jacobsen,et al. Alzheimer's disease: from pathology to therapeutic approaches. , 2009, Angewandte Chemie.
[3] Wei Zhang,et al. Functionalized 3-benzylidene-indolin-2-ones: inducers of NAD(P)H-quinone oxidoreductase 1 (NQO1) with antiproliferative activity. , 2009, Bioorganic & medicinal chemistry.
[4] Birgit Dümpelfeld,et al. Purification, pharmacological modulation, and biochemical characterization of interactors of endogenous human gamma-secretase. , 2009, Biochemistry.
[5] M. Botta,et al. Synthesis, modeling, and RET protein kinase inhibitory activity of 3- and 4-substituted beta-carbolin-1-ones. , 2008, Journal of medicinal chemistry.
[6] S. D’Mello,et al. Synthesis and Structure-Activity Relationship Studies of 3-Substituted Indolin-2-ones as Effective Neuroprotective Agents , 2008, Experimental biology and medicine.
[7] Alessandra Gianoncelli,et al. Identification of novel protein kinase CK1 delta (CK1delta) inhibitors through structure-based virtual screening. , 2008, Bioorganic & medicinal chemistry letters.
[8] E. Mandelkow,et al. Curcumin‐Derived Pyrazoles and Isoxazoles: Swiss Army Knives or Blunt Tools for Alzheimer's Disease? , 2008, ChemMedChem.
[9] P. Greengard,et al. Regulation of Alzheimer's disease amyloid-β formation by casein kinase I , 2007, Proceedings of the National Academy of Sciences.
[10] C. Haass,et al. Scaffold of the cyclooxygenase-2 (COX-2) inhibitor carprofen provides Alzheimer gamma-secretase modulators. , 2006, Journal of medicinal chemistry.
[11] P. Renard,et al. Studies towards the conception of new selective PPARβ/δ ligands , 2006 .
[12] Ping-Chiang Lyu,et al. Indol-1-yl acetic acids as peroxisome proliferator-activated receptor agonists: design, synthesis, structural biology, and molecular docking studies. , 2006, Journal of medicinal chemistry.
[13] E. Ongini,et al. Non‐steroidal anti‐inflammatory drugs (NSAIDs) in Alzheimer's disease: old and new mechanisms of action , 2004, Journal of neurochemistry.
[14] Rong Wang,et al. Purification and characterization of the human gamma-secretase complex. , 2004, Biochemistry.
[15] S. Weggen,et al. Evidence That Nonsteroidal Anti-inflammatory Drugs Decrease Amyloid β42 Production by Direct Modulation of γ-Secretase Activity* , 2003, Journal of Biological Chemistry.
[16] C. Dvorak,et al. A new class of diamine-based human histamine H3 receptor antagonists: 4-(aminoalkoxy)benzylamines. , 2003, Journal of medicinal chemistry.
[17] T. Iwatsubo,et al. Sulindac Sulfide Is a Noncompetitive γ-Secretase Inhibitor That Preferentially Reduces Aβ42 Generation* , 2003, The Journal of Biological Chemistry.
[18] T. Hunter,et al. The Protein Kinase Complement of the Human Genome , 2002, Science.
[19] D. Beher,et al. Generation of C‐terminally truncated amyloid‐β peptides is dependent on γ‐secretase activity , 2002 .
[20] Rong Wang,et al. A subset of NSAIDs lower amyloidogenic Aβ42 independently of cyclooxygenase activity , 2001, Nature.
[21] Graeme Irvine Stevenson,et al. L-685,458, an Aspartyl Protease Transition State Mimic, Is a Potent Inhibitor of Amyloid β-Protein Precursor γ-Secretase Activity , 2000 .
[22] Martin Egli,et al. Crystal Structure of a Conformation-selective Casein Kinase-1 Inhibitor* , 2000, The Journal of Biological Chemistry.
[23] Min Xu,et al. Presenilin 1 is linked with gamma-secretase activity in the detergent solubilized state. , 2000, Proceedings of the National Academy of Sciences of the United States of America.
[24] J. Ozga,et al. Effect of halogen substitution of indole-3-acetic acid on biological activity in pea fruit , 1995 .
[25] C. Haass,et al. N-Substituted carbazolyloxyacetic acids modulate Alzheimer associated γ-secretase , 2007 .