Evaluation of N‐benzyl‐N‐[11C]methyl‐2‐ (7‐methyl‐8‐oxo‐2‐phenyl‐7,8‐dihydro‐9H‐purin‐9‐yl)acetamide ([11C]DAC) as a novel translocator protein (18 kDa) radioligand in kainic acid‐lesioned rat
暂无分享,去创建一个
Ming-Rong Zhang | O. Inoue | Kazutoshi Suzuki | Tomoteru Yamasaki | Joji Yui | K. Kawamura | K. Kumata | A. Hatori | M. Yamaguchi | Kazuhiko Yanamoto | Chika Odawara | KAZUHIKO YANAMOTO | TOMOTERU YAMASAKI | KATSUSHI KUMATA | JOJI YUI | CHIKA ODAWARA | KAZUNORI KAWAMURA | AKIKO HATORI | OSAMU INOUE | MASATOSHI YAMAGUCHI | KAZUTOSHI SUZUKI | MING-RONG ZHANG | Ming-Rong Zhang
[1] M. Imaizumi,et al. PET imaging with [ 11 C ] PBR 28 can localize and quantify upregulated peripheral benzodiazepine receptors associated with cerebral ischemia in rat , 2006 .
[2] Abraham Weizman,et al. Enigma of the peripheral benzodiazepine receptor. , 1999, Pharmacological reviews.
[3] Tetsuya Suhara,et al. Longitudinal, Quantitative Assessment of Amyloid, Neuroinflammation, and Anti-Amyloid Treatment in a Living Mouse Model of Alzheimer's Disease Enabled by Positron Emission Tomography , 2007, The Journal of Neuroscience.
[4] Philippe Hantraye,et al. 11C-DPA-713: A Novel Peripheral Benzodiazepine Receptor PET Ligand for In Vivo Imaging of Neuroinflammation , 2007, Journal of Nuclear Medicine.
[5] A. Gee,et al. The peripheral benzodiazepine receptor ligand PK11195 binds with high affinity to the acute phase reactant alpha1-acid glycoprotein: implications for the use of the ligand as a CNS inflammatory marker. , 2003, Nuclear medicine and biology.
[6] F. Yasuno,et al. Increased Binding of Peripheral Benzodiazepine Receptor in Alzheimer's Disease Measured by Positron Emission Tomography with [11C]DAA1106 , 2008, Biological Psychiatry.
[7] Yuji Nagai,et al. Novel peripheral benzodiazepine receptor ligand [11C]DAA1106 for PET: An imaging tool for glial cells in the brain , 2004, Synapse.
[8] B. Gulyás,et al. Brain Uptake and Plasma Metabolism of [11C]Vinpocetine: A Preliminary PET Study in a Cynomolgus Monkey , 1999, Journal of neuroimaging : official journal of the American Society of Neuroimaging.
[9] Ariel Miller,et al. Imaging brain inflammation Marco Rovaris, Massimo Filippi , 2001 .
[10] Akiko Hatori,et al. In vitro and ex vivo autoradiography studies on peripheral-type benzodiazepine receptor binding using [11C]AC-5216 in normal and kainic acid-lesioned rats , 2007, Neuroscience Letters.
[11] R. Anholt,et al. Peripheral-type benzodiazepine receptors: autoradiographic localization in whole-body sections of neonatal rats. , 1985, The Journal of pharmacology and experimental therapeutics.
[12] D. Nutt,et al. Translocator protein (18kDa): new nomenclature for the peripheral-type benzodiazepine receptor based on its structure and molecular function. , 2006, Trends in pharmacological sciences.
[13] S. Meikle,et al. Synthesis and in vivo evaluation of a novel peripheral benzodiazepine receptor PET radioligand. , 2005, Bioorganic & medicinal chemistry.
[14] S. Jan,et al. In vivo imaging of brain lesions with [11C]CLINME, a new PET radioligand of peripheral benzodiazepine receptors , 2007, Glia.
[15] T. Guilarte,et al. Cellular and Subcellular Localization of Peripheral Benzodiazepine Receptors After Trimethyltin Neurotoxicity , 2000, Journal of neurochemistry.
[16] Sami S Zoghbi,et al. Synthesis and evaluation in monkey of two sensitive 11C-labeled aryloxyanilide ligands for imaging brain peripheral benzodiazepine receptors in vivo. , 2008, Journal of medicinal chemistry.
[17] Ryuji Nakao,et al. Quantitative Analysis for Estimating Binding Potential of the Peripheral Benzodiazepine Receptor with [11C]DAA1106 , 2007, Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism.
[18] Denis Guilloteau,et al. DPA-714, a New Translocator Protein–Specific Ligand: Synthesis, Radiofluorination, and Pharmacologic Characterization , 2008, Journal of Nuclear Medicine.
[19] O. Inoue,et al. Synthesis and evaluation of11C-PK 11195 forin vivo study of peripheral-type benzodiazepine receptors using position emission tomography , 1989 .
[20] J Versijpt,et al. PET visualization of microglia in multiple sclerosis patients using [11C]PK11195 , 2003, European journal of neurology.
[21] Tetsuya Suhara,et al. [(11)C]DAA1106: radiosynthesis and in vivo binding to peripheral benzodiazepine receptors in mouse brain. , 2003, Nuclear medicine and biology.
[22] G. Paxinos,et al. The Rat Brain in Stereotaxic Coordinates , 1983 .
[23] D. Duverger,et al. Imaging of primary and remote ischaemic and excitotoxic brain lesions. An autoradiographic study of peripheral type benzodiazepine binding sites in the rat and cat , 1988, Brain Research.
[24] Ryuji Nakao,et al. Quantitative analyses of 18F-FEDAA1106 binding to peripheral benzodiazepine receptors in living human brain. , 2006, Journal of nuclear medicine : official publication, Society of Nuclear Medicine.
[25] Sylvain Houle,et al. Radiosynthesis and initial evaluation of [18F]-FEPPA for PET imaging of peripheral benzodiazepine receptors. , 2008, Nuclear medicine and biology.
[26] B. Agranoff,et al. Barbiturate-enhanced detection of brain lesions by carbon-14-labeled 2-deoxyglucose autoradiography. , 1983, Science.
[27] C. Carter,et al. Peripheral type benzodiazepine binding sites are a sensitive indirect index of neuronal damage , 1987, Brain Research.
[28] T. Guilarte,et al. Peripheral benzodiazepine receptor imaging in CNS demyelination: functional implications of anatomical and cellular localization. , 2004, Brain : a journal of neurology.
[29] Hervé Boutin,et al. Nuclear imaging of neuroinflammation: a comprehensive review of [11C]PK11195 challengers , 2008, European Journal of Nuclear Medicine and Molecular Imaging.
[30] C. Wiley,et al. The Positron Emission Tomography Ligand DAA1106 Binds With High Affinity to Activated Microglia in Human Neurological Disorders , 2008, Journal of neuropathology and experimental neurology.
[31] M. Petit-Taboué,et al. Brain kinetics and specific binding of [11C]PK 11195 to omega 3 sites in baboons: positron emission tomography study. , 1991, European journal of pharmacology.
[32] S. Kurumiya,et al. Antianxiety and antidepressant‐like effects of AC‐5216, a novel mitochondrial benzodiazepine receptor ligand , 2004, British journal of pharmacology.
[33] V. Perry,et al. Differential Blood–Brain Barrier Breakdown and Leucocyte Recruitment Following Excitotoxic Lesions in Juvenile and Adult Rats , 1998, Experimental Neurology.
[34] Tetsuya Suhara,et al. 11C-AC-5216: A Novel PET Ligand for Peripheral Benzodiazepine Receptors in the Primate Brain , 2007, Journal of Nuclear Medicine.
[35] S. Hume,et al. Synthesis of the enantiomers of [N-methyl-11C]PK 11195 and comparison of their behaviours as radioligands for PK binding sites in rats. , 1994, Nuclear medicine and biology.
[36] F. Fazio,et al. Labeling and evaluation of N-[11C]methylated quinoline-2-carboxamides as potential radioligands for visualization of peripheral benzodiazepine receptors. , 2001, Journal of medicinal chemistry.
[37] O. Inoue,et al. Synthesis and evaluation of 11C-PK 11195 for in vivo study of peripheral-type benzodiazepine receptors using positron emission tomography. , 1989, Annals of nuclear medicine.
[38] M. Grégoire,et al. Synthesis and biological evaluation of substituted [18F]imidazo[1,2-a]pyridines and [18F]pyrazolo[1,5-a]pyrimidines for the study of the peripheral benzodiazepine receptor using positron emission tomography. , 2008, Journal of medicinal chemistry.
[40] Robert B. Innis,et al. PET imaging with [11C]PBR28 can localize and quantify upregulated peripheral benzodiazepine receptors associated with cerebral ischemia in rat , 2007, Neuroscience Letters.
[41] Yen F. Tai,et al. Imaging microglial activation in Huntington's disease , 2007, Brain Research Bulletin.
[42] Jordi Llop,et al. Imaging Brain Inflammation with [11C]PK11195 by PET and Induction of the Peripheral-Type Benzodiazepine Receptor after Transient Focal Ischemia in Rats , 2007, Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism.
[43] Tetsuya Suhara,et al. Development of a new radioligand, N-(5-fluoro-2-phenoxyphenyl)-N-(2-[18F]fluoroethyl-5-methoxybenzyl)acetamide, for pet imaging of peripheral benzodiazepine receptor in primate brain. , 2004, Journal of medicinal chemistry.
[44] B. Wipf,et al. Computer controlled large scale production of , 1994 .