One-step radiosynthesis of 4-nitrophenyl 2-[(18) F]fluoropropionate ([(18) F]NFP); improved preparation of radiolabeled peptides for PET imaging.
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R. Hicks | A. Katsifis | J. Karas | C. Hutton | P. Roselt | C. Wichmann | Wayne Noonan | M. Haskali
[1] H. Maecke,et al. Radiolabeled Peptides: Valuable Tools for the Detection and Treatment of Cancer , 2012, Theranostics.
[2] H. Maecke,et al. Radiopharmaceutical development of radiolabelled peptides , 2012, European Journal of Nuclear Medicine and Molecular Imaging.
[3] Rhona A. Berganos,et al. First Experience with Clinical-Grade [18F]FPP(RGD)2: An Automated Multi-step Radiosynthesis for Clinical PET Studies , 2012, Molecular Imaging and Biology.
[4] Xiaoyuan Chen,et al. Comparison study of [18F]FAl-NOTA-PRGD2, [18F]FPPRGD2, and [68Ga]Ga-NOTA-PRGD2 for PET imaging of U87MG tumors in mice. , 2011, Bioconjugate chemistry.
[5] R. Kimura,et al. PET Imaging of Integrin Positive Tumors Using 18F Labeled Knottin Peptides , 2011, Theranostics.
[6] Rhona A. Berganos,et al. Pilot pharmacokinetic and dosimetric studies of (18)F-FPPRGD2: a PET radiopharmaceutical agent for imaging α(v)β(3) integrin levels. , 2011, Radiology.
[7] Xiaoyuan Chen,et al. 18F-Labeled GRPR Agonists and Antagonists: A Comparative Study in Prostate Cancer Imaging , 2011, Theranostics.
[8] M. Schwaiger,et al. PET Imaging of Integrin αVβ3 Expression , 2011, Theranostics.
[9] D E Olberg,et al. Labeling strategies of peptides with ¹⁸F for positron emission tomography. , 2010, Current topics in medicinal chemistry.
[10] Kai Chen,et al. 18F-Labeled Galacto and PEGylated RGD Dimers for PET Imaging of αvβ3 Integrin Expression , 2010, Molecular Imaging and Biology.
[11] R. Valkema,et al. Somatostatin-receptor-based imaging and therapy of gastroenteropancreatic neuroendocrine tumors. , 2010, Endocrine-related cancer.
[12] A. Cuthbertson,et al. One step radiosynthesis of 6-[(18)F]fluoronicotinic acid 2,3,5,6-tetrafluorophenyl ester ([(18)F]F-Py-TFP): a new prosthetic group for efficient labeling of biomolecules with fluorine-18. , 2010, Journal of medicinal chemistry.
[13] Shuang Liu. Radiolabeled cyclic RGD peptides as integrin alpha(v)beta(3)-targeted radiotracers: maximizing binding affinity via bivalency. , 2009, Bioconjugate chemistry.
[14] R. Valkema,et al. Tumor imaging and therapy using radiolabeled somatostatin analogues. , 2009, Accounts of chemical research.
[15] B. Felding-Habermann,et al. Activation of tumor cell integrin αvβ3 controls angiogenesis and metastatic growth in the brain , 2009, Proceedings of the National Academy of Sciences.
[16] H. Kessler,et al. Ligands for mapping alphavbeta3-integrin expression in vivo. , 2009, Accounts of chemical research.
[17] H. Wester,et al. Molecular imaging targeting peptide receptors. , 2009, Methods.
[18] J. Reubi,et al. Peptide-Based Probes for Cancer Imaging , 2008, Journal of Nuclear Medicine.
[19] Markus Schwaiger,et al. [18F]Galacto-RGD Positron Emission Tomography for Imaging of αvβ3 Expression on the Neovasculature in Patients with Squamous Cell Carcinoma of the Head and Neck , 2007, Clinical Cancer Research.
[20] W. Cai,et al. 18F-labeled mini-PEG spacered RGD dimer (18F-FPRGD2): synthesis and microPET imaging of αvβ3 integrin expression , 2007, European Journal of Nuclear Medicine and Molecular Imaging.
[21] M. Schwaiger,et al. Biodistribution and pharmacokinetics of the alphavbeta3-selective tracer 18F-galacto-RGD in cancer patients. , 2005, Journal of nuclear medicine : official publication, Society of Nuclear Medicine.
[22] M. Schwaiger,et al. Radiolabeled carbohydrated somatostatin analogs: a review of the current status. , 2004, Cancer biotherapy & radiopharmaceuticals.
[23] J. Reubi. Peptide receptors as molecular targets for cancer diagnosis and therapy. , 2003, Endocrine reviews.
[24] Milind Rajopadhye,et al. Tumor targeting with radiolabeled alpha(v)beta(3) integrin binding peptides in a nude mouse model. , 2002, Cancer research.
[25] Sibylle Ziegler,et al. Noninvasive Imaging of αvβ3 Integrin Expression Using 18F-labeled RGD-containing Glycopeptide and Positron Emission Tomography , 2001 .
[26] J W Smith,et al. Integrin activation controls metastasis in human breast cancer. , 2001, Proceedings of the National Academy of Sciences of the United States of America.
[27] Horst Kessler,et al. Radiolabeled αvβ3 Integrin Antagonists: A New Class of Tracers for Tumor Targeting , 1999 .
[28] W. Eckelman,et al. One-step synthesis of 18F labeled [18F]-N-succinimidyl 4-(fluoromethyl)benzoate for protein labeling. , 1994, Applied radiation and isotopes : including data, instrumentation and methods for use in agriculture, industry and medicine.
[29] H. Coenen,et al. Fluoroacylation agents based on small n.c.a. [18F]fluorocarboxylic acids , 1994 .
[30] H. Coenen,et al. N.C.A. 18F-fluoroacylation via fluorocarboxylic acid esters , 1988 .
[31] David A. Cheresh,et al. Integrins in cancer: biological implications and therapeutic opportunities , 2010, Nature Reviews Cancer.
[32] J. Katzenellenbogen,et al. Facile nucleophilic fluorination reactions using tert-alcohols as a reaction medium: significantly enhanced reactivity of alkali metal fluorides and improved selectivity. , 2008, The Journal of organic chemistry.
[33] S. Gambhir,et al. Quantitative PET Imaging of Tumor Integrin αvβ3 Expression with 18F-FRGD2 , 2006 .
[34] M. Schwaiger,et al. [18F]Galacto-RGD: synthesis, radiolabeling, metabolic stability, and radiation dose estimates. , 2004, Bioconjugate chemistry.