Facile synthesis of 2-carboxanilido-3-arylquinazolin-4-ones from N1-(2-carboxyphenyl)-N2-(aryl)oxalamides

[1]  Shiuh-Tzung Liu,et al.  Preparation of 4(3H)-quinazolinones from aryldiazonium salt, nitriles and 2-aminobenzoate via a cascade annulation , 2019, Tetrahedron.

[2]  Walid Fathalla,et al.  Synthesis and Antimicrobial Activity of Methyl 2‐(2‐(2‐Arylquinazolin‐4‐yl)oxy) Acetylamino Alkanoates , 2018, Journal of Heterocyclic Chemistry.

[3]  R. S. Gouhar,et al.  Synthesis and Reactions of Some New Quinazoline Derivatives forIn VitroEvaluation as Anticancer and Antimicrobial Agents , 2018, Journal of Heterocyclic Chemistry.

[4]  M. Mohamed,et al.  Synthesis and antitumor evaluation of trimethoxyanilides based on 4(3H)-quinazolinone scaffolds. , 2016, European journal of medicinal chemistry.

[5]  S. Katsyuba,et al.  A novel acid-catalyzed rearrangement of 2-substituted-3-(2-nitrophenyl)oxiranes for the synthesis of di- and mono-oxalamides , 2016 .

[6]  Haifeng Zhou,et al.  FeCl3-catalyzed tandem condensation/intramolecular nucleophilic addition/C–C bond cleavage: a concise synthesis of 2-substitued quinazolinones from 2-aminobenzamides and 1,3-diketones in aqueous media , 2016 .

[7]  A. Samigullina,et al.  Transformations of anilides of 3-aryl-2,3-epoxypropionic acids when exposed to acidic agents , 2015, Russian Chemical Bulletin.

[8]  U. A. Kshirsagar,et al.  Recent developments in the chemistry of quinazolinone alkaloids. , 2015, Organic & biomolecular chemistry.

[9]  C. Bundgaard,et al.  A Multifaceted GABAA Receptor Modulator: Functional Properties and Mechanism of Action of the Sedative-Hypnotic and Recreational Drug Methaqualone (Quaalude) , 2015, Molecular Pharmacology.

[10]  A. Gubaidullin,et al.  Metal-free intramolecular transannulation of N,3-diaryloxirane-2-carboxamides: a concise and versatile route to 3-arylquinolin-2(1H)-ones , 2015 .

[11]  B. Elmuradov,et al.  Tricyclic Quinazoline Alkaloids: Isolation, Synthesis, Chemical Modification, and Biological Activity , 2014, Chemistry of Natural Compounds.

[12]  S. Bari,et al.  Quinazolines: new horizons in anticonvulsant therapy. , 2014, European journal of medicinal chemistry.

[13]  M. Pines,et al.  The chemistry and biology of febrifugine and halofuginone. , 2014, Bioorganic & medicinal chemistry.

[14]  Jie Bao,et al.  Asperterrestide A, a cytotoxic cyclic tetrapeptide from the marine-derived fungus Aspergillus terreus SCSGAF0162. , 2013, Journal of natural products.

[15]  Zheng-chao Tu,et al.  Alkaloids from the deep-sea-derived fungus Aspergillus westerdijkiae DFFSCS013. , 2013, Journal of natural products.

[16]  Can Zhang,et al.  Novel oxazolo[4,5-g]quinazolin-2(1H)-ones: dual inhibitors of EGFR and Src protein tyrosine kinases. , 2012, European journal of medicinal chemistry.

[17]  A. El-Azab,et al.  Design and synthesis of novel 7-aminoquinazoline derivatives: antitumor and anticonvulsant activities. , 2012, Bioorganic & medicinal chemistry letters.

[18]  G. Marzaro,et al.  Quinazoline derivatives as potential anticancer agents: a patent review (2007 – 2010) , 2012, Expert opinion on therapeutic patents.

[19]  P. Evans,et al.  Dihydroxylation of vinyl sulfones: stereoselective synthesis of (+)- and (-)-febrifugine and halofuginone. , 2010, The Journal of organic chemistry.

[20]  S. Dakshanamurthy,et al.  Asymmetric synthesis of 2,3-dihydro-2-arylquinazolin-4-ones: methodology and application to a potent fluorescent tubulin inhibitor with anticancer activity. , 2008, Journal of medicinal chemistry.

[21]  N. Argade,et al.  The Chemistry of Recently Isolated Naturally Occurring Quinazolinone Alkaloids , 2006 .

[22]  H. Fuwa,et al.  Synthetic studies on 3-arylquinazolin-4-ones: intramolecular nucleophilic aromatic substitution reaction of 2-carboxamido-3-arylquinazolin-4-ones and its application to the synthesis of secondary aryl amines , 2005 .

[23]  M. Döring,et al.  Double Anion Capture Reactions of Anthranilic Esters with Oxaldiimidoyl Dichlorides − Efficient Synthesis of 2,2′-Biquinazoline-4,4′(3H,3′H)-diones , 2001 .

[24]  S. Kuo,et al.  6-Alkylamino- and 2,3-dihydro-3'-methoxy-2-phenyl-4-quinazolinones and related compounds: their synthesis, cytotoxicity, and inhibition of tubulin polymerization. , 2000, Journal of medicinal chemistry.

[25]  M. Kurosu.  Expeditious amide-forming reactions using thiol esters , 2000 .

[26]  M. Döring,et al.  Efficient Synthesis of Quinazolin-4-ones and Axially Chiral 2,2′-Bisquinazolin-4-ones by Reaction of Anthranilic Acid Derived Nucleophiles with Oxalic Acid-Bis(imidoyl)chlorides , 1999 .

[27]  K. Rad‐Moghadam,et al.  One-pot Synthesis of Substituted Quinazolin-4(3H)-ones under Microwave Irradiation , 1998 .

[28]  B. Bandgar.  Synthesis of Quinazolin-4-(3h)-ones from O-Amidobenzonitriles Using Urea-hydrogen Peroxide1 , 1997 .

[29]  L. Őrfi,et al.  Heterocondensed quinazolones: synthesis and protein-tyrosine kinase inhibitory activity of 3,4-dihydro-1H,6H-[1,4] oxazino-[3,4-b]quinazolin-6-one derivatives. , 1996, Bioorganic & medicinal chemistry.

[30]  T. Saeki,et al.  Cyclic GMP phosphodiesterase inhibitors. 2. Requirement of 6-substitution of quinazoline derivatives for potent and selective inhibitory activity. , 1994, Journal of medicinal chemistry.

[31]  N. Peet,et al.  3-(1H-tetrazol-5-yl)-4(3H)-quinazolinone sodium salt (MDL 427): a new antiallergic agent. , 1986, Journal of medicinal chemistry.

[32]  S. Johne,et al.  Chinazolincarbonsäuren. XII. Mitteilung. Synthese von [2-(Ethoxycarbonyl)-3,4-dihydro-4-oxochinazolin-3-yl]-, [2-(Ethoxycarbonyl)chinazolin-4-yloxy]- und (5,6,7,8-Tetrahydro-2-phenylchinazolin-4-ylthio)alkansäure-estern† , 1986 .

[33]  Y. Yamada,et al.  Synthesis of the metabolites of afloqualone and related compounds. , 1983, Chemical & pharmaceutical bulletin.

[34]  S. Ozawa,et al.  Aldol Reaction of Aluminium Enolate Resulting from 1,4-Addition of R2AlX to α,β-Unsaturated Carbonyl Compound. A 1-Acylethenyl Anion Equivalent , 1981 .

[35]  M. Badr,et al.  Studies on Synthesis of 6-Bromo-2,3-disubstituted 4(3H)-Quinazolinones and Their Thiones , 1980 .

[36]  S. Weinreb,et al.  A mild, general method for conversion of esters to amides , 1978 .

[37]  J. Taylor,et al.  Synthesis and central nervous system activity of quinazolones related to 2-methyl-3-(o-tolyl)-4(3H)-quinazolone (methaqualone). , 1977, Journal of medicinal chemistry.

[38]  T. Hisano.  RECENT STUDIES ON THE MODIFIED NIEMENTOWSKI 4-QUINAZOLONE SYNTHESIS. A REVIEW , 1973 .

[39]  B. R. Baker,et al.  Nonclassical Antimetabolites. X.1,2 A Facile Synthesis of 4-Quinazolone-2-carboxylic Acid and the Structure of Bogert's Ammonium Salt , 1962 .

[40]  Friedrich Uhlig.  Polyphosphorsäure ‐ ein neues Cyclisierungsmittel in der präparativen organischen Chemie , 1954 .

[41]  J. F. Morgan,et al.  Phosphazo Compounds and their Use in Preparing Amides , 1946 .

[42]  S. Niementowski.  Synthesen von Chinazolinverbindungen , 1894 .