Switching reaction pathways of trifluoromethylated thiobenzanilides by choice of different oxidative systems

[1]  Haibo Xie,et al.  Diastereoselective silver-catalyzed 1,3-dipolar cycloaddition of azomethine ylides with fluorinated imine. , 2010, The Journal of organic chemistry.

[2]  Ri‐Yuan Tang,et al.  Copper-catalyzed thiolation annulations of 1,4-dihalides with sulfides leading to 2-trifluoromethyl benzothiophenes and benzothiazoles. , 2010, The Journal of organic chemistry.

[3]  Haibo Xie,et al.  A new strategy for the synthesis of poly-substituted 3-H, 3-fluoro, or 3-trifluoromethyl pyridines via the tandem C-F bond cleavage protocol. , 2010, Organic letters.

[4]  Haibo Xie,et al.  Efficient Synthesis of 2‐Fluoromethylated Quinolines via Copper‐Catalyzed Alkynylation and Cyclization of Fluorinated Imidoyl Iodides , 2010 .

[5]  Haibo Xie,et al.  Copper(I)-Catalyzed Synthesis of Novel 4-(Trifluoromethyl)-[1,2,3]triazolo[1,5-a]quinoxalines via Cascade Reactions of N-(o-Haloaryl)alkynylimine with Sodium Azide , 2010 .

[6]  Devender Singh,et al.  Metal‐Free Air Oxidation of Thiols in Recyclable Ionic Liquid: A Simple and Efficient Method for the Synthesis of Disulfides , 2010 .

[7]  Haibo Xie,et al.  A general and straightforward method for the synthesis of 2-trifluoromethylbenzothiazoles. , 2010, Organic letters.

[8]  Haibo Xie,et al.  Palladium catalyzed synthesis of 2-trifluoromethylquinolines through a domino Sonogashira-alkyne carbocyclization process. , 2010, Chemical communications.

[9]  Xin Lv,et al.  Synthesis of N-Substituted-2-Aminobenzothiazoles by Ligand-Free Copper(I)-Catalyzed Cross-Coupling Reaction of 2-Haloanilines with Isothiocyanates , 2009 .

[10]  B. Patel,et al.  Copper(I)‐Catalyzed Cascade Synthesis of 2‐Substituted 1,3‐Benzothiazoles: Direct Access to Benzothiazolones , 2009 .

[11]  Hoyun Lee,et al.  Hybrid pharmacophore design and synthesis of isatin-benzothiazole analogs for their anti-breast cancer activity. , 2009, Bioorganic & medicinal chemistry.

[12]  R. Batey,et al.  Heterocycle formation via palladium-catalyzed intramolecular oxidative C-H bond functionalization: an efficient strategy for the synthesis of 2-aminobenzothiazoles. , 2009, Organic letters.

[13]  Peng Xue,et al.  Efficient and economical access to substituted benzothiazoles: copper-catalyzed coupling of 2-haloanilides with metal sulfides and subsequent condensation. , 2009, Angewandte Chemie.

[14]  Haibo Xie,et al.  Synthesis of 2-fluoroalkylbenzimidazoles via copper(I)-catalyzed tandem reactions. , 2009, Chemical communications.

[15]  Scott P. Brown,et al.  Synthesis and evaluation of benzothiazole-based analogues as novel, potent, and selective fatty acid amide hydrolase inhibitors. , 2009, Journal of medicinal chemistry.

[16]  T. Doi,et al.  Palladium-catalyzed synthesis of 2-substituted benzothiazoles via a C-H functionalization/intramolecular C-S bond formation process. , 2008, Organic letters.

[17]  N. Downer-Riley,et al.  Conversion of thiobenzamides to benzothiazoles via intramolecular cyclization of the aryl radical cation , 2008 .

[18]  K. Bahrami,et al.  Mild and highly efficient method for the synthesis of 2-arylbenzimidazoles and 2-arylbenzothiazoles. , 2008, The Journal of organic chemistry.

[19]  D. Muralidharan,et al.  Oxidative cyclization of thiophenolic and phenolic Schiff's bases promoted by PCC: a new oxidant for 2-substituted benzothiazoles and benzoxazoles , 2008 .

[20]  K. Belfield,et al.  A New Water-Soluble Near-Neutral Ratiometric Fluorescent pH Indicator , 2007 .

[21]  T. Itoh,et al.  A novel practical synthesis of benzothiazoles via Pd-catalyzed thiol cross-coupling. , 2007, Organic letters.

[22]  Wencong Lu,et al.  One-pot synthesis of 2-trifluoromethyl and 2-difluoromethyl substituted benzo-1,3-diazoles , 2007 .

[23]  B. Srikanth,et al.  Synthesis of 2-Arylbenzothiazoles by DDQ-Promoted Cyclization of Thioformanilides; A Solution-Phase Strategy for Library Synthesis , 2007 .

[24]  M. Idrees,et al.  A convenient access to substituted benzothiazole scaffolds via intramolecular cyclization of thioformanilides , 2007 .

[25]  M. Idrees,et al.  Hypervalent iodine mediated intramolecular cyclization of thioformanilides: expeditious approach to 2-substituted benzothiazoles. , 2006, The Journal of organic chemistry.

[26]  R. Batey,et al.  Parallel synthesis of a library of benzoxazoles and benzothiazoles using ligand-accelerated copper-catalyzed cyclizations of ortho-halobenzanilides. , 2006, The Journal of organic chemistry.

[27]  E. Stone,et al.  Antitumor benzothiazoles. 26.(1) 2-(3,4-dimethoxyphenyl)-5-fluorobenzothiazole (GW 610, NSC 721648), a simple fluorinated 2-arylbenzothiazole, shows potent and selective inhibitory activity against lung, colon, and breast cancer cell lines. , 2006, Journal of medicinal chemistry.

[28]  J. Zou,et al.  Mn(III)-Promoted cyclization of substituted thioformanilides under microwave irradiation: a new reagent for 2-substituted benzothiazoles , 2005 .

[29]  E. De Clercq,et al.  Synthesis and antileishmanial activity of (1,3-benzothiazol-2-yl) amino-9-(10H)-acridinone derivatives. , 2004, European journal of medicinal chemistry.

[30]  R. Batey,et al.  Copper- and palladium-catalyzed intramolecular C-S bond formation: a convenient synthesis of 2-aminobenzothiazoles. , 2004, Chemical communications.

[31]  C. Claver,et al.  Synthesis of 2-substituted-benzothiazoles by palladium-catalyzed intramolecular cyclization of o-bromophenylthioureas and o-bromophenylthioamides , 2003 .

[32]  E. Sausville,et al.  DNA damage and cell cycle arrest induced by 2-(4-amino-3-methylphenyl)-5-fluorobenzothiazole (5F 203, NSC 703786) is attenuated in aryl hydrocarbon receptor deficient MCF-7 cells , 2003, British Journal of Cancer.

[33]  K. Paull,et al.  2-(4-Aminophenyl)benzothiazoles: novel agents with selective profiles of in vitro anti-tumour activity. , 1998, British Journal of Cancer.

[34]  M. Soufiaoui,et al.  Nouvelle Voie de Synthèse des 2-Arylbenzothiazoles Transfert d'Electrons Activé par Micro-ondes , 1997 .

[35]  S Wrigley,et al.  Antitumor benzothiazoles. 3. Synthesis of 2-(4-aminophenyl)benzothiazoles and evaluation of their activities against breast cancer cell lines in vitro and in vivo. , 1996, Journal of medicinal chemistry.

[36]  D. Davies,et al.  Structural studies on bioactive compounds. 23. Synthesis of polyhydroxylated 2-phenylbenzothiazoles and a comparison of their cytotoxicities and pharmacological properties with genistein and quercetin. , 1994, Journal of medicinal chemistry.

[37]  P. Jacobson.  Ueber Bildung von Anhydroverbindungen des Orthoamidophenylmercaptans aus Thioaniliden , 1886 .