Current progress toward synthetic routes and medicinal significance of quinoline

[1]  M. Zaki,et al.  Mechanochemical Synthesis and Molecular Docking Studies of New Azines Bearing Indole as Anticancer Agents , 2023, Molecules.

[2]  Sasidhar B. Somappa,et al.  An insight into the recent developments in anti-infective potential of indole and associated hybrids , 2022, Journal of Molecular Structure.

[3]  K. Lestari,et al.  Potential of Quinine Sulfate for COVID-19 Treatment and Its Safety Profile: Review , 2021, Clinical pharmacology : advances and applications.

[4]  I. Eissa,et al.  Design, synthesis, docking, and anticancer evaluations of phthalazines as VEGFR‐2 inhibitors , 2021, Archiv der Pharmazie.

[5]  S. Mouneir,et al.  Synthesis, DFT calculation, pharmacological evaluation, and catalytic application in the synthesis of diverse pyrano[2,3-c]pyrazole derivatives. , 2021, Bioorganic chemistry.

[6]  S. Mouneir,et al.  Recent advances in chemistry and pharmacological aspects of 2-pyridone scaffolds , 2021, Journal of Saudi Chemical Society.

[7]  Atukuri Dorababu.  Quinoline: A Promising Scaffold in Recent Antiprotozoal Drug Discovery , 2021, ChemistrySelect.

[8]  Kapil Kumar,et al.  Synthetic and medicinal perspective of quinolines as antiviral agents , 2021, European Journal of Medicinal Chemistry.

[9]  Raviraj S. Pattanashettar,et al.  A comprehensive review on the biological interest of quinoline and its derivatives. , 2020, Bioorganic & medicinal chemistry.

[10]  Vishant C. Patel,et al.  A green perspective: Synthesis of 2-chloro-3-formylquinolines and its derivatives , 2020 .

[11]  F. A. Saddique,et al.  Recent synthetic methodologies for the tricyclic fused-quinoline derivatives , 2020 .

[12]  V. Bobade,et al.  Synthesis and antimycobacterial screening of new 4‐(4‐ (1‐benzyl‐1H ‐1,2,3‐triazol‐4‐yl)‐ 1‐phenyl‐1H ‐pyrazol‐3‐yl)quinoline derivatives , 2020, Journal of Heterocyclic Chemistry.

[13]  Uma S. Dubey,et al.  Quinoline Glycoconjugates as Potentially Anticancer and Anti‐Inflammatory Agents: An Investigation Involving Synthesis, Biological Screening, and Docking , 2020 .

[14]  R. Eswaramoorthy,et al.  Synthesis and Antibacterial, Antioxidant, and Molecular Docking Analysis of Some Novel Quinoline Derivatives , 2020 .

[15]  S. Gaonkar,et al.  SYNTHESIS, ANTIOXIDANT AND ANTICANCER ACTIVITY OF NEW QUINOLINE-[1, 2, 4]-TRIAZOLE HYBRIDS , 2020 .

[16]  P. Taslimi,et al.  Quinoline‐based promising anticancer and antibacterial agents, and some metabolic enzyme inhibitors , 2020, Archiv der Pharmazie.

[17]  Endale Mulugeta,et al.  Recent advances in the synthesis of biologically and pharmaceutically active quinoline and its analogues: a review , 2020, RSC advances.

[18]  T. Eren,et al.  Decision making for promising quinoline‐based anticancer agents through combined methodology , 2020, Journal of biochemical and molecular toxicology.

[19]  K. N. Venugopala,et al.  Cytotoxicity and Antimycobacterial Properties of Pyrrolo[1,2-a]quinoline Derivatives: Molecular Target Identification and Molecular Docking Studies , 2020, Antibiotics.

[20]  D. Raoult,et al.  New insights on the antiviral effects of chloroquine against coronavirus: what to expect for COVID-19? , 2020, International Journal of Antimicrobial Agents.

[21]  M. Assy,et al.  An efficient synthesis and antimicrobial activity of N-bridged triazolo[3,4-b]thiadiazine and triazolo[3,4-b]thiadiazole derivatives under microwave irradiation , 2020, Synthetic Communications.

[22]  Wu Zhong,et al.  Remdesivir and chloroquine effectively inhibit the recently emerged novel coronavirus (2019-nCoV) in vitro , 2020, Cell Research.

[23]  El-Sayed R. El-Sayed,et al.  Semi-continuous production of the anticancer drug taxol by Aspergillus fumigatus and Alternaria tenuissima immobilized in calcium alginate beads , 2020, Bioprocess and Biosystems Engineering.

[24]  M. Assy,et al.  Cyclization of N ‐benzyl cyanoacetamide: Novel synthesis and biological activity of pyrrole, pyrimidine, and pyran derivatives , 2020 .

[25]  J. Sangshetti,et al.  Quinoline Based Monocarbonyl Curcumin Analogs as Potential Antifungal and Antioxidant Agents: Synthesis, Bioevaluation and Molecular Docking Study , 2019, Chemistry & biodiversity.

[26]  M. Assy,et al.  An Efficient and Green Synthesis of Highly SubstitutedN‐Amino‐2‐oxo‐nicotinonitriles and Their Sulfonamide Derivatives under Ultrasonic and Microwave Irradiation , 2019, ChemistrySelect.

[27]  A. Bhaumik,et al.  An Efficient Mesoporous Cu‐Organic Nanorod for Friedländer Synthesis of Quinoline and Click Reactions , 2019, ChemCatChem.

[28]  Liang‐Hua Zou,et al.  Copper-Catalyzed Ring-Opening/Reconstruction of Anthranils with Oxo-Compounds: Synthesis of Quinoline Derivatives. , 2019, The Journal of organic chemistry.

[29]  H. Togo,et al.  Preparation of 2-arylquinolines from β-arylpropionitriles with aryllithiums and NIS through iminyl radical-mediated cyclization. , 2019, Organic and biomolecular chemistry.

[30]  Rakesh Kumar,et al.  Catalyst-Free Synthesis of 2-Anilinoquinolines and 3-Hydroxyquinolines via Three-Component Reaction of Quinoline N-Oxides, Aryldiazonium Salts, and Acetonitrile. , 2019, The Journal of organic chemistry.

[31]  M. Akhter,et al.  Green recipes to quinoline: A review. , 2019, European journal of medicinal chemistry.

[32]  A. Chaturvedi,et al.  Visible light catalyzed synthesis of quinolines from (aza)-Morita-Baylis-Hillman adducts. , 2018, Organic and biomolecular chemistry.

[33]  Rakesh Kumar,et al.  Rh(III)-Catalyzed C(8)-H Functionalization of Quinolines via Simultaneous C-C and C-O Bond Formation: Direct Synthesis of Quinoline Derivatives with Antiplasmodial Potential. , 2018, The Journal of organic chemistry.

[34]  R. Krüger,et al.  Current advances of pharmacological properties of 7-chloro-4-(phenylselanyl) quinoline: Prevention of cognitive deficit and anxiety in Alzheimer's disease model. , 2018, Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie.

[35]  A. Amr,et al.  Chemistry of 4,6-diaryl(heteroaryl)-2-oxonicotinonitriles and their fused heterocyclic systems , 2018, Synthetic Communications.

[36]  Xingmin Sun,et al.  Facilely accessible quinoline derivatives as potent antibacterial agents. , 2018, Bioorganic & medicinal chemistry.

[37]  Xia Chen,et al.  Highly efficient Brønsted acid and Lewis acid catalysis systems for the Friedländer Quinoline synthesis , 2018 .

[38]  Mei Zhao,et al.  An efficient and green synthesis of ferrocenyl-quinoline conjugates via a TsOH-catalyzed three-component reaction in water , 2018, RSC advances.

[39]  Jing Sun,et al.  An Efficient Synthesis of Spiropyrroloquinolines by the Domino Reaction of α‐Dicarbonyl Compounds and Anilinosuccinimides , 2017 .

[40]  Zhi Xu,et al.  Quinoline hybrids and their antiplasmodial and antimalarial activities. , 2017, European journal of medicinal chemistry.

[41]  Z. Chao,et al.  Heterogeneous catalytic synthesis of quinoline compounds from aniline and C1–C4 alcohols over zeolite-based catalysts , 2017 .

[42]  G. Cheng,et al.  Chloroquine, a FDA-approved Drug, Prevents Zika Virus Infection and its Associated Congenital Microcephaly in Mice , 2017, EBioMedicine.

[43]  Zi‐Xuan Wang,et al.  Divergent Synthesis of Functionalized Quinolines from Aniline and Two Distinct Amino Acids. , 2017, The Journal of organic chemistry.

[44]  Wei Zhang,et al.  One-pot and catalyst-free synthesis of pyrroloquinolinediones and quinolinedicarboxylates , 2017 .

[45]  J. Nanubolu,et al.  An Efficient One-Pot Synthesis of Densely Functionalized Fused-Quinolines via Sequential Ugi4CC and Acid-Mediated Povarov-Type Reaction. , 2017, ACS Combinatorial Science.

[46]  Mustapha Mandewale,et al.  A review on quinoline hydrazone derivatives as a new class of potent antitubercular and anticancer agents , 2017 .

[47]  E. V. Van der Eycken,et al.  Temperature switchable Brønsted acid-promoted selective syntheses of spiro-indolenines and quinolines. , 2017, Chemical communications.

[48]  Manoj Kumar,et al.  Polythiophene-Encapsulated Bimetallic Au-Fe3O4 Nano-Hybrid Materials: A Potential Tandem Photocatalytic System for Nondirected C(sp2)–H Activation for the Synthesis of Quinoline Carboxylates , 2017 .

[49]  D. Pathak,et al.  Comprehensive review on current developments of quinoline-based anticancer agents , 2016 .

[50]  Bryan J Cowen,et al.  Recent Advances in Metal-Free Quinoline Synthesis , 2016, Molecules.

[51]  Xiaomin Xie,et al.  Visible-Light-Induced Photocatalytic Aerobic Oxidation/Povarov Cyclization Reaction: Synthesis of Substituted Quinoline-Fused Lactones. , 2016, The Journal of organic chemistry.

[52]  Mustapha Mandewale,et al.  Synthesis, structural studies and antituberculosis evaluation of new hydrazone derivatives of quinoline and their Zn(II) complexes , 2016 .

[53]  A. Zarghi,et al.  Design, Synthesis and Biological Evaluation of4-(Imidazolylmethyl)-2-(4-methylsulfonyl phenyl)-Quinoline Derivatives as Selective COX-2 Inhibitors and In-vitro Anti-breast Cancer Agents , 2016, Iranian journal of pharmaceutical research : IJPR.

[54]  Vinod Kumar,et al.  Synthesis of quinoline based heterocyclic compounds for blue lighting application , 2015 .

[55]  D. Jung,et al.  Quinolines Formation by Condensation of Heteroaromatic Ketones and 2‐Aminobenzophenones under MW Irradiation , 2015 .

[56]  Stéphanie Vandekerckhove,et al.  Quinoline-based antimalarial hybrid compounds. , 2015, Bioorganic & medicinal chemistry.

[57]  M. Tobe,et al.  The chemistry and biological activity of heterocycle-fused quinolinone derivatives: A review. , 2015, European journal of medicinal chemistry.

[58]  R. Kumar,et al.  A review on anticancer potential of bioactive heterocycle quinoline. , 2015, European journal of medicinal chemistry.

[59]  S. Bharate,et al.  Metal-free domino one-pot protocols for quinoline synthesis , 2015 .

[60]  Chavis A. Stackhouse,et al.  Investigation of prototypal MOFs consisting of polyhedral cages with accessible Lewis-acid sites for quinoline synthesis. , 2015, Chemical communications.

[61]  Shouyun Yu,et al.  Synthesis of Fused Quinoline and Quinoxaline Derivatives Enabled by Domino Radical Triple Bond Insertions , 2014 .

[62]  S. Tu,et al.  Highly diastereoselective synthesis of quinoline-2,5-diones and pyrazolo[3,4-b]pyridin-6(7H)-ones under microwave irradiation , 2014 .

[63]  Rangappa S. Keri,et al.  Quinoline: a promising antitubercular target. , 2014, Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie.

[64]  M. Heravi,et al.  Recent Applications of Doebner, Doebner-von Miller and Knoevenagel-Doebner Reactions in Organic Syntheses , 2014 .

[65]  Rajesh H. Vekariya,et al.  Recent advances in the synthesis of quinolines: a review , 2014 .

[66]  Vladimir Poroikov,et al.  Prediction of the Biological Activity Spectra of Organic Compounds Using the Pass Online Web Resource , 2014, Chemistry of Heterocyclic Compounds.

[67]  Shouyun Yu,et al.  Visible-light-mediated fluoroalkylation of isocyanides with ethyl bromofluoroacetates: unified synthesis of mono- and difluoromethylated phenanthridine derivatives. , 2014, Organic letters.

[68]  D. Browning.  Pharmacology of Chloroquine and Hydroxychloroquine , 2014, Hydroxychloroquine and Chloroquine Retinopathy.

[69]  S. Tu,et al.  A Facile and Expeditious Microwave‐Assisted Synthesis of Furo[3,4‐b]indeno[2,1‐f]quinolin‐1‐one Derivatives via Multicomponent Reaction , 2013 .

[70]  M. Pal,et al.  Quinolines: a new hope against inflammation. , 2013, Drug discovery today.

[71]  Lizhen Fang,et al.  A simple one-pot synthesis of quinoline-4-carboxylic acid derivatives by Pfitzinger reaction of isatin with ketones in water , 2013, Monatshefte für Chemie - Chemical Monthly.

[72]  D. Bahnemann,et al.  Arenesulfonic Acid-Functionalized Mesoporous Silica Decorated with Titania: A Heterogeneous Catalyst for the One-Pot Photocatalytic Synthesis of Quinolines from Nitroaromatic Compounds and Alcohols , 2013 .

[73]  Xiaodong Jia,et al.  Radical cation salt induced Povarov reaction between iminoethyl glyoxylate and N-vinylamides: synthesis of quinoline-2-carboxylate derivatives , 2012 .

[74]  S. Gogoi,et al.  A microwave promoted solvent-free approach to steroidal quinolines and their in vitro evaluation for antimicrobial activities , 2012, Steroids.

[75]  S. Tu,et al.  Multicomponent synthesis of polysubstituted dihydroquinoline derivatives , 2012 .

[76]  S. Tangestaninejad,et al.  Efficient and environmentally-benign three-component synthesis of quinolines and bis-quinolines catalyzed by recyclable potassium dodecatungstocobaltate trihydrate under microwave irradiation , 2012 .

[77]  R. K. Verma,et al.  InCl3-driven regioselective synthesis of functionalized/annulated quinolines: scope and limitations. , 2012, Chemistry, an Asian journal.

[78]  Yongping Liang,et al.  Electrophile-driven regioselective synthesis of functionalized quinolines. , 2011, Organic letters.

[79]  Xiao-Ling Liu,et al.  Efficient Friedländer Synthesis of Quinoline Derivatives from 2-Aminoarylketones and Carbonyl Compounds Mediated by Recyclable PEG-Supported Sulfonic Acid , 2009 .

[80]  Li-Ming Zhao,et al.  Design and synthesis of 5-alkoxy-[1,2,4]triazolo[4,3-a]quinoline derivatives with anticonvulsant activity. , 2009, European journal of medicinal chemistry.

[81]  H. Tokuyama,et al.  Auto-tandem catalysis in the synthesis of substituted quinolines from aldimines and electron-rich olefins: cascade Povarov-hydrogen-transfer reaction. , 2008, The Journal of organic chemistry.

[82]  S. Yamashkin,et al.  Traditional and Modern Approaches to the Synthesis of Quinoline Systems by the Skraup and Doebner—Miller Methods , 2007 .

[83]  S. Yamashkin,et al.  Traditional and modern approaches to the synthesis of quinoline systems by the Skraup and Doebner-Miller methods. (Review) , 2006 .

[84]  C. Kappe,et al.  Microwaves in Organic and Medicinal Chemistry: KAPPE:MICROWAVES 2E O-BK , 2005 .

[85]  L. Caparrotta,et al.  Mannich bases of 3H-pyrrolo[3,2-f]quinoline having vasorelaxing activity. , 2002, European journal of medicinal chemistry.

[86]  N. P. Buu‐Hoï,et al.  The Pfitzinger Reaction in the Synthesis of Quinoline Derivatives , 1953 .

[87]  V. Kouznetsov,et al.  The direct C–H alkenylation of quinoline N-oxides as a suitable strategy for the synthesis of promising antiparasitic drugs , 2020 .

[88]  V. Ximenes,et al.  Facile Synthesis and Photophysical Characterization of New Quinoline Dyes , 2016, Journal of Fluorescence.

[89]  M. Pervaiz,et al.  Microwave Assisted Gould-Jacobs Reaction for Synthesis of 3-Acetyl-4-hydroxyquinoline Derivatives , 2015 .

[90]  L. C. Silva‐Filho,et al.  Synthesis of Quinoline Derivatives by Multicomponent Reaction Using Niobium Pentachloride as Lewis Acid , 2015 .

[91]  Omprakash Tanwar,et al.  Quinoline: A versatile heterocyclic. , 2013, Saudi pharmaceutical journal : SPJ : the official publication of the Saudi Pharmaceutical Society.

[92]  Thokhir Basha Shaik,et al.  Synthesis and anticancer activity of 4β-alkylamidochalcone and 4β-cinnamido linked podophyllotoxins as apoptotic inducing agents. , 2012, European journal of medicinal chemistry.