Synthesis and anticancer activity of aminopropoxytriterpenoids

[1]  O. Kazakova,et al.  Synthesis and evaluation of 29-norcycloartane triterpenoids as α-glucosidase inhibitors , 2015, Medicinal Chemistry Research.

[2]  D. V. Kazakov,et al.  Synthesis of a Triterpenoid with a 1,2,4,5-Tetraoxane Fragment , 2015, Chemistry of Natural Compounds.

[3]  M. Mahmoudi,et al.  Ursolic acid induced apoptotic cell death following activation of caspases in isolated human melanoma cells , 2015, Cell biology international.

[4]  Zhenfeng Chen,et al.  Synthesis of oleanolic acid dimers linked at C-28 and evaluation of anti-tumor activity. , 2015, European journal of medicinal chemistry.

[5]  V. Poroikov,et al.  Synthesis and anticancer activity of quinopimaric and maleopimaric acids’ derivatives. , 2014, Bioorganic & medicinal chemistry.

[6]  O. Kazakova,et al.  One-pot Synthesis of Hollongdione from Dipterocarpol , 2014, Natural product communications.

[7]  Fernando J. Reyes-Zurita,et al.  Solid-phase library synthesis of bi-functional derivatives of oleanolic and maslinic acids and their cytotoxicity on three cancer cell lines. , 2014, ACS combinatorial science.

[8]  Vladimir Poroikov,et al.  Prediction of the Biological Activity Spectra of Organic Compounds Using the Pass Online Web Resource , 2014, Chemistry of Heterocyclic Compounds.

[9]  N. A. Zhukova,et al.  Synthesis of aminopropylamino derivatives of betulinic and oleanolic acids , 2013, Russian Journal of Bioorganic Chemistry.

[10]  D. V. Kazakov,et al.  Synthesis, structure, and pharmacological activity of (7R,8S)-epoxy-(13R,17R)-trioxolane abietic acid , 2013, Russian Journal of Bioorganic Chemistry.

[11]  B. Siewert,et al.  Synthesis of Antitumor‐Active Betulinic Acid‐Derived Hydroxypropargylamines by Copper‐Catalyzend Mannich Reactions , 2013, Archiv der Pharmazie.

[12]  B. Siewert,et al.  Cytotoxic betulin-derived hydroxypropargylamines trigger apoptosis. , 2013, Bioorganic & medicinal chemistry.

[13]  Y. Jing,et al.  Ursane-type pentacyclic triterpenoids as useful platforms to discover anticancer drugs. , 2012, Natural product reports.

[14]  G. Sethi,et al.  Targeted inhibition of tumor proliferation, survival, and metastasis by pentacyclic triterpenoids: potential role in prevention and therapy of cancer. , 2012, Cancer letters.

[15]  D. V. Kazakov,et al.  Anomalous ozonolysis product of 3β,28-di-O-acetyl-29-norlupan-20-one-O-methyloxime , 2011, Chemistry of Natural Compounds.

[16]  B. Cassels,et al.  Anti-HIV activity of natural triterpenoids and hemisynthetic derivatives 2004–2009 , 2011, Phytochemistry Reviews.

[17]  O. Kazakova,et al.  Synthesis of a-secomethylenamino- and substituted amidoximotriterpenoids , 2011, Russian Journal of Bioorganic Chemistry.

[18]  D. Ströhl,et al.  Improvement of the Cytotoxicity and Tumor Selectivity of Glycyrrhetinic Acid by Derivatization with Bifunctional Aminoacids , 2011, Archiv der Pharmazie.

[19]  Hongbin Sun,et al.  Synthesis, Biology and Clinical Significance of Pentacyclic Triterpenes: A Multi‐Target Approach to Prevention and Treatment of Metabolic and Vascular Diseases , 2011 .

[20]  O. Kazakova,et al.  Synthesis and antitumor activity of aminopropoxy derivatives of betulin, erythrodiol, and uvaol , 2011, Russian Journal of Bioorganic Chemistry.

[21]  G. Tolstikov,et al.  Synthetic transformations of higher terpenoids: XXIV. Synthesis of cyanoethyl derivatives of lupane triterpenoids and their transformation into 1,2,4-oxadiazoles , 2011 .

[22]  D. V. Kazakov,et al.  Chemiluminescence as a base for a new approach to the study of pharmacologically promising peroxide agents , 2011 .

[23]  D. V. Kazakov,et al.  Synthesis of triterpenoid-based 1,2,4-trioxolanes and 1,2,4-dioxazolidines by ozonolysis of allobetulin derivatives , 2011 .

[24]  B. Siewert,et al.  Synthesis, Encapsulation and Antitumor Activity of New Betulin Derivatives , 2011, Archiv der Pharmazie.

[25]  D. Ströhl,et al.  Synthesis, cytotoxicity and liposome preparation of 28-acetylenic betulin derivatives. , 2010, Bioorganic & medicinal chemistry.

[26]  T. Mueller,et al.  Carbamate derivatives of betulinic acid and betulin with selective cytotoxic activity. , 2010, Bioorganic & medicinal chemistry letters.

[27]  N. Medvedeva,et al.  Synthesis, modification, and antimicrobial activity of the N-methylpiperazinyl amides of triterpenic acids , 2010, Russian Journal of Bioorganic Chemistry.

[28]  D. V. Kazakov,et al.  Synthesis of nontrivial quinopimaric acid derivatives by oxidation with dimethyldioxirane , 2010 .

[29]  Huiyuan Chen,et al.  Terpenoids induce cell cycle arrest and apoptosis from the stems of Celastrus kusanoi associated with reactive oxygen species. , 2010, Journal of agricultural and food chemistry.

[30]  Melanie N Laszczyk,et al.  Pentacyclic triterpenes of the lupane, oleanane and ursane group as tools in cancer therapy. , 2009, Planta medica.

[31]  W. Fang,et al.  Pentacyclic triterpenoids and their saponins with apoptosis-inducing activity. , 2009, Current topics in medicinal chemistry.

[32]  Keduo Qian,et al.  Plant-derived triterpenoids and analogues as antitumor and anti-HIV agents. , 2009, Natural product reports.

[33]  Marita Hernández,et al.  Natural Triterpenic Diols Promote Apoptosis in Astrocytoma Cells through ROS-Mediated Mitochondrial Depolarization and JNK Activation , 2009, PloS one.

[34]  G. Tolstikov,et al.  Synthesis of olean-18(19)-ene derivatives from betulin , 2009, Russian Journal of Bioorganic Chemistry.

[35]  S. Kwon,et al.  Anti-cancer effect of Betulin on a human lung cancer cell line: a pharmacoproteomic approach using 2 D SDS PAGE coupled with nano-HPLC tandem Mass Spectrometry. , 2009, Planta medica.

[36]  Vladimir Poroikov,et al.  Chapter 6:Probabilistic Approaches in Activity Prediction , 2008 .

[37]  H. Daniel,et al.  Erythrodiol, a natural triterpenoid from olives, has antiproliferative and apoptotic activity in HT-29 human adenocarcinoma cells. , 2008, Molecular nutrition & food research.

[38]  A. Pichette,et al.  Useful approach to access germanicanes from betulin , 2007 .

[39]  U. Pfüller,et al.  Solubility studies of oleanolic acid and betulinic acid in aqueous solutions and plant extracts of Viscum album L. , 2007, Planta medica.

[40]  C. Schempp,et al.  Physical, chemical and pharmacological characterization of a new oleogel-forming triterpene extract from the outer bark of birch (betulae cortex). , 2006, Planta medica.

[41]  R. Shoemaker.  The NCI60 human tumour cell line anticancer drug screen , 2006, Nature Reviews Cancer.

[42]  P. Džubák,et al.  Pharmacological activities of natural triterpenoids and their therapeutic implications. , 2006, Natural product reports.

[43]  K. Hata,et al.  Anti-leukemia activities of Lup-28-al-20(29)-en-3-one, a lupane triterpene. , 2003, Toxicology letters.

[44]  G. Tolstikov,et al.  Synthesis and Pharmacological Activity of Betulin Dinicotinate , 2002, Russian Journal of Bioorganic Chemistry.

[45]  J. Pezzuto,et al.  Synthesis of betulinic acid derivatives with activity against human melanoma. , 1998, Bioorganic & medicinal chemistry letters.

[46]  G. S. Johnson,et al.  An Information-Intensive Approach to the Molecular Pharmacology of Cancer , 1997, Science.

[47]  M. Boyd,et al.  Some practical considerations and applications of the national cancer institute in vitro anticancer drug discovery screen , 1995 .

[48]  M R Grever,et al.  The National Cancer Institute: cancer drug discovery and development program. , 1992, Seminars in oncology.

[49]  D. Scudiero,et al.  Feasibility of a high-flux anticancer drug screen using a diverse panel of cultured human tumor cell lines. , 1991, Journal of the National Cancer Institute.

[50]  D A Scudiero,et al.  Feasibility of drug screening with panels of human tumor cell lines using a microculture tetrazolium assay. , 1988, Cancer research.

[51]  T. Mosmann.  Rapid colorimetric assay for cellular growth and survival: application to proliferation and cytotoxicity assays. , 1983, Journal of immunological methods.

[52]  Liu Xiaokan.  Influence of betulin in proliferation and apoptosis of human colon cancer SW480 cells , 2015 .

[53]  D. A. Borisov,et al.  Chemiluminescence from the biomimetic reaction of 1,2,4-trioxolanes and 1,2,4,5-tetroxanes with ferrous ions , 2012 .

[54]  R. Geran,et al.  PROTOCOLS FOR SCREENING CHEMICAL AGENTS AND NATURAL PRODUCTS AGAINST ANIMAL TUMORS AND OTHER BIOLOGICAL SYSTEMS , 1972 .

[55]  S. A. Hiller,et al.  Syntheses of methyl-2-furylketones , 1967 .