2-Aryl-3-(6-trifluoromethoxy)benzo[d]thiazole-based thiazolidinone hybrids as potential anti-infective agents: Synthesis, biological evaluation and molecular docking studies.

[1]  E. Giovannetti,et al.  Therapeutic Strategies To Counteract Antibiotic Resistance in MRSA Biofilm‐Associated Infections , 2020, ChemMedChem.

[2]  L. Jilla,et al.  Synthesis and antimicrobial agents of thiazolidinone derivatives from benzocyclohepetenone , 2020 .

[3]  M. Al-Omar,et al.  Synthesis of Novel Sulfamethaoxazole 4-Thiazolidinone Hybrids and Their Biological Evaluation , 2020, Molecules.

[4]  M. J. Ramaiah,et al.  Synthesis, in vitro and structural aspects of benzothiazole analogs as anti-oxidants and potential neuroprotective agents. , 2020, Environmental toxicology and pharmacology.

[5]  Maxwell Z. Wilson,et al.  A Dual-Mechanism Antibiotic Kills Gram-Negative Bacteria and Avoids Drug Resistance , 2020, Cell.

[6]  Tian-Yi Zhang,et al.  Synthesis, biological evaluation of benzothiazole derivatives bearing a 1,3,4-oxadiazole moiety as potential anti-oxidant and anti-inflammatory agents. , 2020, Bioorganic & medicinal chemistry letters.

[7]  K. N. Venugopala,et al.  Screening and Molecular Docking of Novel Benzothiazole Derivatives as Potential Antimicrobial Agents , 2020, Antibiotics.

[8]  E. Giovannetti,et al.  Thiazoles, Their Benzofused Systems, and Thiazolidinone Derivatives: Versatile and Promising Tools to Combat Antibiotic Resistance , 2020, Journal of medicinal chemistry.

[9]  D. Kaminskyy,et al.  Thiazole-Bearing 4-Thiazolidinones as New Anticonvulsant Agents , 2020, Scientia Pharmaceutica.

[10]  D. Carbone,et al.  Inhibitors of antibiotic resistance mechanisms: clinical applications and future perspectives. , 2020, Future medicinal chemistry.

[11]  C. Tratrat.  Novel Thiazole-Based Thiazolidinones as Potent Anti-Infective Agents: In silico PASS and Toxicity Prediction, Synthesis, Biological Evaluation and Molecular Modelling. , 2020, Combinatorial chemistry & high throughput screening.

[12]  G. Elgemeie,et al.  Efficient Synthesis and Docking Studies of Novel Benzothiazole-Based Pyrimidinesulfonamide Scaffolds as New Antiviral Agents and Hsp90α Inhibitors , 2020, ACS omega.

[13]  M. Haroun.  Novel Series of Benzothiazole-Based Pyrazolidinediones Targeting PPARγ. In Silico Studies, Synthesis and In Vivo Anti-Diabetic Activity. , 2019, Medicinal chemistry (Shariqah (United Arab Emirates)).

[14]  C. Supuran,et al.  Benzothiazole derivatives as anticancer agents , 2019, Journal of enzyme inhibition and medicinal chemistry.

[15]  A. Geronikaki,et al.  Novel Thiazolidin-4-ones as Potential Non-Nucleoside Inhibitors of HIV-1 Reverse Transcriptase , 2019, Molecules.

[16]  E. Giovannetti,et al.  2,6-Disubstituted imidazo[2,1-b][1,3,4]thiadiazole derivatives as potent staphylococcal biofilm inhibitors. , 2019, European journal of medicinal chemistry.

[17]  Yasser A. Bamarouf,et al.  Synthesis of benzothiazole derivatives as a potent α-glucosidase inhibitor. , 2019, Bioorganic chemistry.

[18]  M. Sarg,et al.  Design, Synthesis, and Anticancer Activity of Novel Benzothiazole Analogues , 2019, Journal of Heterocyclic Chemistry.

[19]  M. El-Magd,et al.  Design, synthesis, modeling studies and biological evaluation of thiazolidine derivatives containing pyrazole core as potential anti-diabetic PPAR-γ agonists and anti-inflammatory COX-2 selective inhibitors. , 2019, Bioorganic chemistry.

[20]  S. Saini.  Synthesis and Anticonvulsant Studies of Thiazolidinone and Azetidinone Derivatives from Indole Moiety , 2018, Drug Research.

[21]  S. Jagannath,et al.  Anti-mitotic Activity of the Benzothiazole-pyrazole Hybrid Derivatives , 2018, Anti-Infective Agents.

[22]  S. S. Kanwar,et al.  Benzothiazole-Based-Bioconjugates with Improved Antimicrobial, Anticancer and Antioxidant Potential , 2018, ChemistrySelect.

[23]  A. Geronikaki,et al.  5-Adamantan thiadiazole-based thiazolidinones as antimicrobial agents. Design, synthesis, molecular docking and evaluation. , 2018, Bioorganic & medicinal chemistry.

[24]  P. Diana,et al.  Bacterial Biofilm Inhibition in the Development of Effective Anti-Virulence Strategy , 2018, The open medicinal chemistry journal.

[25]  Petrou Anthi,et al.  Design, synthesis and antimicrobial activity of usnic acid derivatives. , 2018, MedChemComm.

[26]  Riham F. George,et al.  Synthesis and biological evaluation of 2-aminothiazole-thiazolidinone conjugates as potential antitubercular agents. , 2018, Future medicinal chemistry.

[27]  Danish Idrees,et al.  Design, synthesis and biological evaluation of novel pyridine-thiazolidinone derivatives as anticancer agents: Targeting human carbonic anhydrase IX. , 2018, European journal of medicinal chemistry.

[28]  S. Okafor,et al.  Novel anti-inflammatory and analgesic agents: synthesis, molecular docking and in vivo studies , 2018, Journal of enzyme inhibition and medicinal chemistry.

[29]  Ki Duk Park,et al.  Indole-Substituted Benzothiazoles and Benzoxazoles as Selective and Reversible MAO-B Inhibitors for Treatment of Parkinson's Disease. , 2017, ACS chemical neuroscience.

[30]  D. Kaminskyy,et al.  Study of novel anticancer 4-thiazolidinone derivatives. , 2017, Chemico-biological interactions.

[31]  Juan Rodrigo Salazar,et al.  Novel 5-aminosalicylic derivatives as anti-inflammatories and myeloperoxidase inhibitors evaluated in silico, in vitro and ex vivo , 2017 .

[32]  K. Ramasamy,et al.  4-Thiazolidinone derivatives: synthesis, antimicrobial, anticancer evaluation and QSAR studies , 2016 .

[33]  A. Saxena,et al.  Design, synthesis and biological evaluation of new substituted 5-benzylideno-2-adamantylthiazol[3,2-b][1,2,4]triazol-6(5H)ones. Pharmacophore models for antifungal activity , 2016 .

[34]  M. Al-agamy,et al.  Design, Synthesis, Antimicrobial Evaluation and Molecular Modeling Study of 1,2,4-Triazole-Based 4-Thiazolidinones , 2016, Molecules.

[35]  M. Rosales-Hernández,et al.  Evaluation of a new benzothiazole derivative with antioxidant activity in the initial phase of acetaminophen toxicity , 2016 .

[36]  G. Özhan,et al.  Indole-based hydrazide-hydrazones and 4-thiazolidinones: synthesis and evaluation as antitubercular and anticancer agents , 2015, Journal of enzyme inhibition and medicinal chemistry.

[37]  T. Singh.  » SYNTHESIS OF THIAZOLIDINE-4-ONE FOR THEIR ANTHELMINTIC ACTIVITY , 2014 .

[38]  Rangappa S. Keri,et al.  Design, synthesis and neuroprotective evaluation of novel tacrine-benzothiazole hybrids as multi-targeted compounds against Alzheimer's disease. , 2013, Bioorganic & medicinal chemistry.

[39]  C. G. Mohan,et al.  Identification of hotspot regions of MurB oxidoreductase enzyme using homology modeling, molecular dynamics and molecular docking techniques , 2011, Journal of molecular modeling.

[40]  Christoph Helma,et al.  Lazy structure-activity relationships (lazar) for the prediction of rodent carcinogenicity and Salmonella mutagenicity , 2006, Molecular Diversity.

[41]  R. Levesque,et al.  Structure and function of the Mur enzymes: development of novel inhibitors , 2002, Molecular microbiology.

[42]  H. T. Ho,et al.  4-Thiazolidinones: novel inhibitors of the bacterial enzyme MurB. , 2000, Bioorganic & medicinal chemistry letters.

[43]  W. El‐Sayed,et al.  Design, synthesis and anti-inflammatory vel 5-(Indol-3-yl)thiazolidinone derivatives as COX-2 inhibitors. , 2020 .

[44]  M. Attimarad,et al.  Design, Synthesis, Evaluation of Antimicrobial Activity and Docking Studies of New Thiazole-based Chalcones. , 2019, Current topics in medicinal chemistry.

[45]  E. Giovannetti,et al.  Synthetic small molecules as anti-biofilm agents in the struggle against antibiotic resistance. , 2019, European journal of medicinal chemistry.

[46]  K. Arora,et al.  Synthesis, Computational Studies and Anticonvulsant Activity of Novel Benzothiazole Coupled Sulfonamide Derivatives , 2019, Iranian journal of pharmaceutical research : IJPR.

[47]  M. Attimarad,et al.  New Benzothiazole-based Thiazolidinones as Potent Antimicrobial Agents. Design, synthesis and Biological Evaluation. , 2018, Current topics in medicinal chemistry.

[48]  S. Bari,et al.  Exploring Anti-inflammatory Potential of Thiazolidinone Derivatives of Benzenesulfonamide via Synthesis, Molecular Docking and Biological Evaluation. , 2016, Anti-Inflammatory & Anti-Allergy Agents in Medicinal Chemistry.