论文信息 - Synthesis of irreversible HIV-1 protease inhibitors containing sulfonamide and sulfone as amide bond isosteres - 字舞流文

Synthesis of irreversible HIV-1 protease inhibitors containing sulfonamide and sulfone as amide bond isosteres

Ho-il Choi | J. Koh | W. Jung | N. Choy | Tae Gyu Lee | Sung Chun Kim | H. Yoon | C. Kim

[1] Sangsoo Kim,et al. DESIGN, SYNTHESIS, AND CHARACTERIZATION OF DIPEPTIDE ISOSTERE CONTAINING CIS-EPOXIDE FOR THE IRREVERSIBLE INACTIVATION OF HIV PROTEASE , 1996 .

[2] Ho-il Choi,et al. Rational design of irreversible, pseudo-C2-symmetric hiv-1 protease inhibitors , 1995 .

[3] U. Hacksell,et al. Stereoselective Epoxidation of Phe-Gly and Phe-Phe Vinyl Isosteres , 1994 .

[4] U. Hacksell,et al. Novel L-Phe-Gly mimetics , 1992 .

[5] C. Debouck,et al. The HIV-1 protease as a therapeutic target for AIDS. , 1992, AIDS research and human retroviruses.

[6] J. Huff,et al. HIV protease: a novel chemotherapeutic target for AIDS. , 1991, Journal of medicinal chemistry.

[7] E. Clercq,et al. Design of Anti-AIDS Drugs , 1990 .

[8] B. Dunn,et al. Viral proteinases: weakness in strength. , 1990, Biochimica et biophysica acta.

[9] Brian W. Metcalf,et al. Inhibition of HIV-1 protease in infected T-lymphocytes by synthetic peptide analogues , 1990, Nature.

[10] B. Ho,et al. Role of human immunodeficiency virus type 1-specific protease in core protein maturation and viral infectivity , 1989, Journal of virology.

[11] D. Rich,et al. An improved cathepsin-D substrate and assay procedure. , 1983, Analytical biochemistry.