Evaluation of small-molecule modulators of the luteinizing hormone/choriogonadotropin and thyroid stimulating hormone receptors: structure-activity relationships and selective binding patterns.
暂无分享,去创建一个
Gerd Krause | Stefano Costanzi | Susanne Neumann | Gunnar Kleinau | Ralf Paschke | Susanna Moore | Jian-kang Jiang | R. Paschke | B. Raaka | G. Krause | M. Gershengorn | S. Neumann | S. Costanzi | G. Kleinau | Craig J. Thomas | A. Colson | Craig J Thomas | Jian-Kang Jiang | Bruce M Raaka | Marvin C Gershengorn | Holger Jaeschke | John Childress | Anny Colson | H. Jaeschke | S. Moore | John Childress
[1] H. Krishnamurthy,et al. Thyroid-Stimulating Hormone and Thyroid-Stimulating Hormone Receptor Structure-Function Relationships , 2002 .
[2] C. Timmers,et al. The First Orally Active Low Molecular Weight Agonists for the LH Receptor: Thienopyr(im)idines with Therapeutic Potential for Ovulation Induction , 2002, Chembiochem : a European journal of chemical biology.
[3] T. Guo. Small molecule agonists and antagonists for the LH and FSH receptors , 2005 .
[4] J. Ballesteros,et al. [19] Integrated methods for the construction of three-dimensional models and computational probing of structure-function relations in G protein-coupled receptors , 1995 .
[5] C. Kappe. Recent Advances in the Biginelli Dihydropyrimidine Synthesis. New Tricks from an Old Dog , 2001 .
[6] Ruben Abagyan,et al. ICM—A new method for protein modeling and design: Applications to docking and structure prediction from the distorted native conformation , 1994, J. Comput. Chem..
[7] C. Timmers,et al. Identification of substituted 6-amino-4-phenyltetrahydroquinoline derivatives: potent antagonists for the follicle-stimulating hormone receptor. , 2005, Journal of medicinal chemistry.
[8] M. Parmentier,et al. Cloning, sequencing and expression of the human thyrotropin (TSH) receptor: evidence for binding of autoantibodies. , 1989, Biochemical and biophysical research communications.
[9] R. Paschke,et al. Identification of a Novel Epitope in the Thyroid-stimulating Hormone Receptor Ectodomain Acting as Intramolecular Signaling Interface*[boxs] , 2004, Journal of Biological Chemistry.
[10] K. Jacobson,et al. Architecture of P2Y nucleotide receptors: structural comparison based on sequence analysis, mutagenesis, and homology modeling. , 2004, Journal of medicinal chemistry.
[11] M. Quon,et al. Hormone Signaling , 2002, Endocrine Updates.
[12] R. Paschke,et al. Role of the third intracellular loop for the activation of gonadotropin receptors. , 1999, Molecular endocrinology.
[13] Adam J Pawson,et al. Gonadotropin-releasing hormone receptors. , 2004, Endocrine reviews.
[14] C. Holmes,et al. Agonists of the follicle stimulating hormone receptor from an encoded thiazolidinone library. , 2004, Journal of combinatorial chemistry.
[15] R. Paschke,et al. A Low Molecular Weight Agonist Signals by Binding to the Transmembrane Domain of Thyroid-stimulating Hormone Receptor (TSHR) and Luteinizing Hormone/Chorionic Gonadotropin Receptor (LHCGR)* , 2006, Journal of Biological Chemistry.