Tablet disintegration and drug dissolution in viscous media: paracetamol IR tablets.

[1]  Hans Lennernäs,et al.  The Effects of Food on the Dissolution of Poorly Soluble Drugs in Human and in Model Small Intestinal Fluids , 2005, Pharmaceutical Research.

[2]  J. Brasseur,et al.  A Novel in Vitro and Numerical Analysis of Shear-Induced Drug Release from Extended-Release Tablets in the Fed Stomach , 2005, Pharmaceutical Research.

[3]  Brahma N. Singh A quantitative approach to probe the dependence and correlation of food‐effect with aqueous solubility, dose/solubility ratio, and partition coefficient (Log P) for orally active drugs administered as immediate‐release formulations , 2005 .

[4]  J. Dressman,et al.  The delayed dissolution of paracetamol products in the canine fed stomach can be predicted in vitro but it does not affect the onset of plasma levels. , 2005, International journal of pharmaceutics.

[5]  P. Dickinson,et al.  An investigation of the disintegration of tablets in biorelevant media. , 2005, International journal of pharmaceutics.

[6]  B. Abrahamsson,et al.  Food effects on tablet disintegration. , 2004, European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences.

[7]  Clive G. Wilson,et al.  Comparison of the Rates of Disintegration, Gastric Emptying, and Drug Absorption Following Administration of a New and a Conventional Paracetamol Formulation, Using γ Scintigraphy , 2003, Pharmaceutical Research.

[8]  R. Krishna,et al.  On the assessment of effects of food on the pharmacokinetics of drugs in early development. , 2002, Biopharmaceutics & drug disposition.

[9]  W. J. Irwin,et al.  A New Rapidly Absorbed Paracetamol Tablet Containing Sodium Bicarbonate. II. Dissolution Studies and In Vitro/In Vivo Correlation , 2002, Drug development and industrial pharmacy.

[10]  G. Tucker,et al.  A New Rapidly Absorbed Paracetamol Tablet Containing Sodium Bicarbonate. I. A Four-Way Crossover Study to Compare the Concentration–Time Profile of Paracetamol from the New Paracetamol/Sodium Bicarbonate Tablet and a Conventional Paracetamol Tablet in Fed and Fasted Volunteers , 2002, Drug development and industrial pharmacy.

[11]  R. Schall,et al.  Comparison of the Pharmacokinetic Profiles of Soluble Aspirin and Solid Paracetamol Tablets in Fed and Fasted Volunteers , 2000, Current medical research and opinion.

[12]  Brahma N. Singh Effects of Food on Clinical Pharmacokinetics , 1999, Clinical pharmacokinetics.

[13]  D. Fleisher,et al.  Drug, Meal and Formulation Interactions Influencing Drug Absorption After Oral Administration , 1999, Clinical pharmacokinetics.

[14]  R. Löbenberg,et al.  Evaluation of Various Dissolution Media for Predicting In Vivo Performance of Class I and II Drugs , 1998, Pharmaceutical Research.

[15]  J. Dressman,et al.  Effect of elevated viscosity in the upper gastrointestinal tract on drug absorption in dogs. , 1998, European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences.

[16]  J. Dressman,et al.  Physiochemical and physiological mechanisms for the effects of food on drug absorption: the role of lipids and pH. , 1997, Journal of pharmaceutical sciences.

[17]  B. Nickel,et al.  The influence of different formula diets and different pharmaceutical formulations on the systemic availability of paracetamol, gallbladder size, and plasma glucose. , 1989, International journal of clinical pharmacology, therapy and toxicology.

[18]  A. C. Shah,et al.  Mass transport in dissolution kinetics. I: Convective diffusion to assess the role of fluid viscosity under forced flow conditions. , 1987, Journal of pharmaceutical sciences.

[19]  Michael A. Koupparis,et al.  Dissolution of 4 controlled-release theophylline formulations in milk , 1987 .

[20]  P. Maturu,et al.  Influence of a high fat breakfast on the bioavailability of theophylline controlled-release formulations: an in vitro demonstration of an in vivo observation. , 1986, Journal of pharmaceutical sciences.

[21]  P. Welling,et al.  Influence of food and fluid ingestion on aspirin bioavailability. , 1978, Journal of pharmaceutical sciences.

[22]  J. Jaffe,et al.  Effects of dietary components on GI absorption of acetaminophen tablets in man. , 1971, Journal of pharmaceutical sciences.

[23]  S. Ibrić,et al.  An attempt to establish an in vitro-in vivo correlation: case of paracetamol immediate-release tablets , 2010, European Journal of Drug Metabolism and Pharmacokinetics.

[24]  Eric Beyssac,et al.  A level A in vitro/in vivo correlation in fasted and fed states using different methods: applied to solid immediate release oral dosage form. , 2006, European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences.

[25]  L. Rumbach,et al.  Intraindividual variability of paracetamol absorption kinetics after a semi-solid meal in healthy volunteers , 1998, European Journal of Clinical Pharmacology.

[26]  H. Junginger,et al.  A new in vitro model to detect interactions between controlled release dosage forms and food , 1990 .

[27]  A. Karim,et al.  Food-Induced Theophylline Release/Absorption Changes from Controlled-Release Formulations: A Proposed In Vitro Model , 1988 .