Synthesis of some pyrazolylaldehyde N-isonicotinoyl hydrazones and 2,5-disubstituted 1,3,4-oxadiazoles as DNA photocleaving agents

[1]  G. Gupta,et al.  Synthesis, docking study, and DNA photocleavage activity of some pyrimidinyl hydrazones and 3-(quinolin-3-yl)-5,7-dimethyl-1,2,4-triazolo[4,3-a]pyrimidine derivatives , 2015, Medicinal Chemistry Research.

[2]  Vasyl Kovalishyn,et al.  Design, synthesis and biological evaluation of novel isoniazid derivatives with potent antitubercular activity. , 2014, European journal of medicinal chemistry.

[3]  Anil Kumar Sharma,et al.  Isoxazoline containing natural products as anticancer agents: a review. , 2014, European journal of medicinal chemistry.

[4]  V. Saini,et al.  1,4-Diaryl-2-mercaptoimidazoles derivatives as a novel class of antimicrobial agents: design, synthesis, and computational studies , 2014, Medicinal Chemistry Research.

[5]  V. Beniwal,et al.  Synthesis, characterization and DNA photocleavage study of a novel dehydroacetic acid based hydrazone Schiff’s base and its metal complexes , 2014, Medicinal Chemistry Research.

[6]  D. Joshi,et al.  Synthesis and antimicrobial evaluation of 1,3,4-oxadiazole-based chalcone derivatives , 2014, Medicinal Chemistry Research.

[7]  Anil Kumar Sharma,et al.  Pyrazole containing natural products: synthetic preview and biological significance. , 2013, European journal of medicinal chemistry.

[8]  S. Sushanth Kumar,et al.  Developments in synthesis of the anti-inflammatory drug, celecoxib: a review. , 2013, Recent patents on inflammation & allergy drug discovery.

[9]  S. Bondock,et al.  Synthesis of some new 2-(3-pyridyl)-4,5-disubstituted thiazoles as potent antimicrobial agents. , 2013, European journal of medicinal chemistry.

[10]  H. Bhojya Naik,et al.  Synthesis, antimicrobial, DNA-binding and photonuclease studies of cobalt(III) and nickel(II) Schiff base complexes. , 2013, Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy.

[11]  Ghada S. Hassan,et al.  Substituted thiazoles VII. Synthesis and antitumor activity of certain 2-(substituted amino)-4-phenyl-1,3-thiazole analogs. , 2012, Bioorganic & medicinal chemistry letters.

[12]  Xianhai Lv,et al.  Design, synthesis, biological evaluation and molecular modeling of novel 1,3,4-oxadiazole derivatives based on Vanillic acid as potential immunosuppressive agents. , 2012, Bioorganic & medicinal chemistry.

[13]  M. Abdelaziz,et al.  Uses of Cyanoacetylhydrazine in Heterocyclic Synthesis: Novel Synthesis of Pyrazole Derivatives with Anti-tumor Activities , 2012, Molecules.

[14]  Hai-bin Gong,et al.  Synthesis, biological evaluation and molecular docking studies of 1,3,4-oxadiazole derivatives as potential immunosuppressive agents. , 2012, Bioorganic & medicinal chemistry.

[15]  J. Barbosa-Filho,et al.  Synthesis, Molecular Properties Prediction, and Anti-staphylococcal Activity of N-Acylhydrazones and New 1,3,4-Oxadiazole Derivatives , 2012, Molecules.

[16]  P. Yogeeswari,et al.  Synthesis of highly potent novel anti-tubercular isoniazid analogues with preliminary pharmacokinetic evaluation. , 2012, Bioorganic & medicinal chemistry letters.

[17]  Changlin Zhou,et al.  Synthesis and evaluation of anti-tubercular and antibacterial activities of new 4-(2,6-dichlorobenzyloxy)phenyl thiazole, oxazole and imidazole derivatives. Part 2. , 2012, European journal of medicinal chemistry.

[18]  P. Kumar An environmentally benign and solvent-free synthesis of 3-aryl[1,2,4]triazolo[4,3-a]pyridines and 1-aryl-5-methyl[1,2,4]triazolo[4,3-a]quinolines using phenyliodine bis(trifluoroacetate) or iodobenzene diacetate , 2012, Chemistry of Heterocyclic Compounds.

[19]  M. Ghodke,et al.  Synthesis of novel N-(2-substituted 4-oxothiazolidin-3-yl) isonicotinamide derivatives as anti mycobacterial agents , 2012 .

[20]  R. Kamble,et al.  Synthetic utility of sydnones: synthesis of pyrazolines derivatized with 1,2,4-triazoles as antihyperglymic, antioxidant agents and their DNA cleavage study , 2012, Medicinal Chemistry Research.

[21]  B. Narasimhan,et al.  Synthesis, antimycobacterial, antiviral, antimicrobial activities, and QSAR studies of isonicotinic acid-1-(substituted phenyl)-ethylidene/cycloheptylidene hydrazides , 2012, Medicinal Chemistry Research.

[22]  A. Deep,et al.  Synthesis of 2-(aryl)-5-(arylidene)-4-thiazolidinone derivatives with potential analgesic and anti-inflammatory activity , 2012, Medicinal Chemistry Research.

[23]  A. Deep,et al.  Synthesis, characterization and antimicrobial evaluation of novel derivatives of isoniazid , 2012, Medicinal Chemistry Research.

[24]  B. Narasimhan,et al.  Isoniazid: the magic molecule , 2012, Medicinal Chemistry Research.

[25]  S. Bősze,et al.  New series of isoniazid hydrazones linked with electron-withdrawing substituents. , 2011, European journal of medicinal chemistry.

[26]  A. Al-ayed Synthesis of New Substituted Chromen[4,3-c]pyrazol-4-ones and Their Antioxidant Activities , 2011, Molecules.

[27]  O. Prakash,et al.  A facile iodine(III)-mediated synthesis of 3-(3-aryl-1-phenyl-1H-pyrazol-4-yl)-[1,2,4]triazolo[4,3-a]pyridines via oxidation of 2-((3-aryl-1-phenyl-1H-pyrazol-4-yl)methylene)-1-(pyridin-2-yl)hydrazines and their antimicrobial evaluations , 2011, Organic and medicinal chemistry letters.

[28]  B. Narasimhan,et al.  Synthesis, antimycobacterial, antiviral, antimicrobial activities, and QSAR studies of isonicotinic acid-1-(substituted phenyl)-ethylidene/cycloheptylidene hydrazides , 2011, Medicinal Chemistry Research.

[29]  K. R. Desai,et al.  Synthesis and anti-tubercular activity of novel pyrazol-5(H)-one derivatives , 2011 .

[30]  P. Yogeeswari,et al.  Microwave assisted one-pot synthesis of highly potent novel isoniazid analogues. , 2011, Bioorganic & medicinal chemistry letters.

[31]  N. Golla,et al.  Synthesis, characterization and biological activities of 2,5-disubstituted 1,3,4-oxadiazoles , 2011 .

[32]  E. Sausville,et al.  Synthesis, Characterization and Evaluation of Isoniazid Analogues as Potent Anticancer Agents , 2011 .

[33]  S. S. Rajput,et al.  A NOVEL METHOD FOR THE SYNTHESIS OF FORMYL PYRAZOLES USING VILSMEIER-HAACK REACTION , 2011 .

[34]  Jagadish Singh,et al.  Synthesis of some novel 3,5-disubstituted 1,3,4-oxadiazole derivatives and anticancer activity on EAC animal model , 2011, Medicinal Chemistry Research.

[35]  V. Revankar,et al.  Synthesis, characterization, antibiogram and DNA binding studies of novel Co(II), Ni(II), Cu(II), and Zn(II) complexes of Schiff base ligands with quinoline core , 2011, Medicinal Chemistry Research.

[36]  A. Kulkarni,et al.  DNA cleavage and antimicrobial investigation of Co(II), Ni(II), and Cu(II) complexes with triazole Schiff bases: synthesis and spectral characterization , 2011, Medicinal Chemistry Research.

[37]  Abdul Samad,et al.  Molecular properties prediction, synthesis and antimicrobial activity of some newer oxadiazole derivatives. , 2010, European journal of medicinal chemistry.

[38]  P. L. Lobo,et al.  Synthesis and biological evaluation of some 1,3,4-oxadiazole derivatives. , 2010, European journal of medicinal chemistry.

[39]  Priyanka Singh,et al.  Design, synthesis and biological evaluation of 1,3,4-oxadiazole derivatives. , 2010, European journal of medicinal chemistry.

[40]  R. Kumar,et al.  Hypervalent iodine(III) mediated synthesis of novel unsymmetrical 2,5-disubstituted 1,3,4-oxadiazoles as antibacterial and antifungal agents. , 2010, European journal of medicinal chemistry.

[41]  P. Shetty,et al.  Synthesis, characterization and biological activity of some new 1,3,4-oxadiazole bearing 2-flouro-4-methoxy phenyl moiety. , 2010, European journal of medicinal chemistry.

[42]  M. Deodhar,et al.  Synthesis and analgesic activity of new pyridine-based heterocyclic derivatives , 2010, Medicinal Chemistry Research.

[43]  Alaa A. Hassan,et al.  Synthesis of novel pyrazole derivatives and evaluation of their antidepressant and anticonvulsant activities. , 2009, European journal of medicinal chemistry.

[44]  A. Bekhit,et al.  Synthesis and biological evaluation of novel pyrazole derivatives as anti-inflammatory antimicrobial agents. , 2009, Medicinal chemistry (Shariqah (United Arab Emirates)).

[45]  V. Zhdankin Hypervalent iodine(III) reagents in organic synthesis , 2009 .

[46]  S. Rostamizadeh,et al.  A mild and facile method for one pot synthesis of 2,5-di-substituted 1,3,4-oxadiazoles at room temperature , 2008 .

[47]  R. Kumar,et al.  A facile and rapid one-pot synthesis of 1,4-diaryl-2-mercaptoimidazoles under solvent-free conditions , 2007 .

[48]  N. Raman,et al.  DNA cleavage, structural elucidation and anti-microbial studies of three novel mixed ligand Schiff base complexes of copper(II) , 2007 .

[49]  Vinod Kumar,et al.  Synthesis and antibacterial activity of some new 1-heteroaryl-5-amino-4-phenyl-3-trifluoromethylpyrazoles. , 2005, European journal of medicinal chemistry.

[50]  D. Richardson,et al.  Crystal and molecular structure of 2-hydroxy-1-naphthaldehyde isonicotinoyl hydrazone (NIH) and its iron(III) complex: an iron chelator with anti-tumour activity , 1999, JBIC Journal of Biological Inorganic Chemistry.

[51]  A. Varvoglis Chemical Transformations Induced by Hypervalent Iodine Reagents , 1997 .

[52]  Alan R. Katritzky,et al.  Comprehensive Heterocyclic Chemistry IV , 1996 .

[53]  L. Dai,et al.  Hypervalent iodine oxidation of N-acylhydrazones and N- phenylsemicarbazone: An efficient method for the synthesis of derivatives of 1,3,4-oxadiazoles and △^3-1,3,4- oxadiazolines , 1993 .