4-(Alkylthio)- and 4-(arylthio)-benzonitrile derivatives as androgen receptor antagonists for the topical suppression of sebum production.
暂无分享,去创建一个
Danielle E. Dettling | D. Pocalyko | C. Kostlan | Z. Wang | L. Hu | L. Mitchell | D. Du | Kimberly Wade | M. Carroll
[1] Danielle E. Dettling,et al. (1R,2S)-4-(2-cyano-cyclohexyl-oxy)-2-trifluoromethyl-benzonitrile, a potent androgen receptor antagonist for stimulating hair growth and reducing sebum production. , 2007, Bioorganic & medicinal chemistry letters.
[2] Danielle E. Dettling,et al. Synthesis and biological evaluation of amino-pyridines as androgen receptor antagonists for stimulating hair growth and reducing sebum production. , 2007, Bioorganic & Medicinal Chemistry Letters.
[3] Danielle E. Dettling,et al. Preparation of 4-aryl-2-trifluoromethylbenzonitrile derivatives as androgen receptor antagonists for topical suppression of sebum production. , 2007, Bioorganic & medicinal chemistry letters.
[4] J. Dalton,et al. Chemistry and structural biology of androgen receptor. , 2005, Chemical reviews.
[5] D. Thiboutot. Regulation of human sebaceous glands. , 2004, The Journal of investigative dermatology.
[6] Y. Fradet. Bicalutamide (Casodex®) in the treatment of prostate cancer , 2004, Expert review of anticancer therapy.
[7] N. Bodor,et al. Designing safer (soft) drugs by avoiding the formation of toxic and oxidative metabolites , 2004, Molecular biotechnology.
[8] G. Heinze,et al. Topical cyproterone acetate treatment in women with acne: a placebo-controlled trial. , 1998, Archives of dermatology.
[9] W. Bergfeld,et al. Treatment of androgenic disorders in women: acne, hirsutism, and alopecia. , 1990, Cleveland Clinic journal of medicine.
[10] F. Wojnarowska,et al. Anti‐androgen treatment in women with acne: a controlled trial , 1986, The British journal of dermatology.
[11] Marcus Low,et al. EFFECT OF TOPICAL CYPROTERONE ACETATE ON SEBUM EXCRETION IN MAN , 1979, The Lancet.