Synthesis and dopamine receptor binding of sulfur-containing aporphines.
暂无分享,去创建一个
[1] R. Baldessarini,et al. Synthesis and neuropharmacological evaluation of R(-)-N-alkyl-11-hydroxynoraporphines and their esters. , 2004, Bioorganic & medicinal chemistry.
[2] M. Tóth,et al. Synthesis of sulfide-and disulfide-type bisaporphines from thebaine , 2004 .
[3] F. Tarazi,et al. Role of Dopamine D4 Receptors in Motor Hyperactivity Induced by Neonatal 6-Hydroxydopamine Lesions in Rats , 2001, Neuropsychopharmacology.
[4] S. Lal,et al. Apomorphine and the dopamine hypothesis of schizophrenia: a dilemma? , 2001, Journal of psychiatry & neuroscience : JPN.
[5] C. Csutoras,et al. A SIMPLE, ONE-POT PROCEDURE FOR THE PREPARATION OF DOPAMINERGIC ALKYLTHIOAPOMORPHINES , 1998 .
[6] J. Kebabian,et al. RBI-257: a highly potent dopamine D4 receptor-selective ligand. , 1997, European journal of pharmacology.
[7] C. Csutoras,et al. A new and efficient one-pot synthesis of apomorphine and its ring-A halogenated derivatives , 1996 .
[8] C. Csutoras,et al. Regioselective O-Demethylation of Aporphines with Methanesulfonic Acid / Methionine: An Efficient One-Pot Transformation of Thebaine to (R)(-)-2-Methoxyapomorphine , 1995 .
[9] J. Clemens,et al. Synthesis and dopamine antagonist activity of 2-thioether derivatives of the ergoline ring system. , 1993, Journal of medicinal chemistry.
[10] R. Baldessarini,et al. Prolonged D2 antidopaminergic activity of alkylating and nonalkylating derivatives of spiperone in rat brain. , 1992, Molecular pharmacology.
[11] R. Baldessarini,et al. Synthesis and dopamine receptor affinity of (R)-(-)-2-fluoro-N-n-propylnorapomorphine: a highly potent and selective dopamine D2 agonist. , 1990, Journal of medicinal chemistry.
[12] R. Baldessarini,et al. Synthesis and dopamine receptor affinities of enantiomers of 2-substituted apomorphines and their N-n-propyl analogues. , 1990, Journal of medicinal chemistry.
[13] L. Szilágyi,et al. Formation of a new polycyclic heteroring system by the acid-catalyzed rearrangement of thebaine in the presence of thiosalicylic acid , 2002 .
[14] B. Kiss,et al. Synthesis and neuropharmacological evaluation of new (R)-(-) and (S)-(+)-2-(alkylthio)aporphine derivatives , 1997 .
[15] S. Berényi,et al. Rearrangement of morphinandienes in methanesulfonic acid , 1993 .
[16] S. Hosztafi,et al. A new efficient method for the preparation of 2-fluoro-N-propylnorapomorphine , 1992 .
[17] R. Baldessarini,et al. R and S enantiomers of 11-hydroxy- and 10,11-dihydroxy-N-allylnoraporphine: synthesis and affinity for dopamine receptors in rat brain tissue. , 1991, Journal of medicinal chemistry.