Development of an efficient and selective radioligand for bradykinin B1 receptor occupancy studies.

[1]  F. Marceau,et al.  Bradykinin receptor ligands: therapeutic perspectives , 2004, Nature Reviews Drug Discovery.

[2]  M. Bock,et al.  Pharmacological characterization and radioligand binding properties of a high-affinity, nonpeptide, bradykinin B1 receptor antagonist. , 2004, European journal of pharmacology.

[3]  M. Bock,et al.  Generation and Characterization of a Human Bradykinin Receptor B1 Transgenic Rat as a Pharmacodynamic Model , 2004, Journal of Pharmacology and Experimental Therapeutics.

[4]  M. Bock,et al.  Discovery of a potent, non-peptide bradykinin B1 receptor antagonist. , 2003, Journal of the American Chemical Society.

[5]  Tsing-Bau Chen,et al.  Benzodiazepines as potent and selective bradykinin B1 antagonists. , 2003, Journal of medicinal chemistry.

[6]  J. Calixto,et al.  The use of kinin B1 and B2 receptor knockout mice and selective antagonists to characterize the nociceptive responses caused by kinins at the spinal level , 2002, Neuropharmacology.

[7]  R. Couture,et al.  Kinin receptors in pain and inflammation. , 2001, European journal of pharmacology.

[8]  Q. Ma,et al.  Basal expression of bradykinin B1 receptor in peripheral sensory ganglia in the rat , 2000, Neuroreport.

[9]  J. Winter,et al.  Bradykinin B1 receptor is constitutively expressed in the rat sensory nervous system , 2000, Neuroscience Letters.

[10]  M. Bock,et al.  Bradykinin antagonists: new opportunities. , 2000, Current opinion in chemical biology.

[11]  T. Walther,et al.  Hypoalgesia and altered inflammatory responses in mice lacking kinin B1 receptors. , 2000, Proceedings of the National Academy of Sciences of the United States of America.

[12]  C. Strader,et al.  Expression of B1 and B2 bradykinin receptor mRNA and their functional roles in sympathetic ganglia and sensory dorsal root ganglia neurones from wild-type and B2 receptor knockout mice , 1997, Neuropharmacology.

[13]  J. Hess,et al.  Partial agonists and full antagonists at the human and murine bradykinin B1 receptors. , 1997, Canadian journal of physiology and pharmacology.

[14]  F. Marceau Kinin B1 receptors: a review. , 1995, Immunopharmacology.

[15]  D. Regoli,et al.  Pharmacology of bradykinin and related kinins. , 1980, Advances in experimental medicine and biology.

[16]  E. Perl,et al.  The molecular basis of pain induction , 1999 .