Identification and biological evaluation of 4-(3-trifluoromethylpyridin-2-yl)piperazine-1-carboxylic acid (5-trifluoromethylpyridin-2-yl)amide, a high affinity TRPV1 (VR1) vanilloid receptor antagonist.
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N. Carruthers | A. Dubin | Sui-Po Zhang | S. Chaplan | Leon Chang | M. Rizzolio | J. Breitenbucher | K. Hoey | B. Lord | M. Bogenstaetter | C. Mazur | Devin M. Swanson | C. Shah | N. Nasser | E. Codd | S. Dax | Changlu Liu | M. Jetter | D. H. Lee | L. Gonzales