论文信息 - Squaric acid derivatives as VLA-4 integrin antagonists. - 字舞流文

Squaric acid derivatives as VLA-4 integrin antagonists.

SAR studies aimed at improving the rate of clearance by the incorporation of a 3,4-diamino-3-cyclobutene-1,2-dione group as an amino acid isostere in a series of VLA-4 integrin antagonists are described.

David Critchley | John R Porter | Sarah C Archibald | Kirstie Childs | John C Head | Ted A H Parton | Martyn K Robinson | Anthony Shock | Graham J Warrellow | Richard J Taylor | Janeen M Linsley | Rikki P Alexander | Barry Langham

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