Solid-Phase Synthesis of 2-Benzothiazolyl and 2-(Aminophenyl)benzothiazolyl Amino Acids and Peptides
暂无分享,去创建一个
[1] B. Shainyan,et al. Synthetic Approaches to Biologically Active C-2-Substituted Benzothiazoles , 2022, Molecules.
[2] T. Walsh,et al. Thiazole/Thiadiazole/Benzothiazole Based Thiazolidin-4-One Derivatives as Potential Inhibitors of Main Protease of SARS-CoV-2 , 2022, Molecules.
[3] C. Supuran,et al. Repurposing FDA-approved sulphonamide carbonic anhydrase inhibitors for treatment of Neisseria gonorrhoeae , 2021, Journal of enzyme inhibition and medicinal chemistry.
[4] M. Shahar Yar,et al. Recent advances and SAR study of 2-substituted benzothiazole scaffold based potent chemotherapeutic agents , 2021, Results in Chemistry.
[5] S. Mahajan,et al. Riluzole: A neuroprotective drug with potential as a novel anti-cancer agent (Review) , 2021, International journal of oncology.
[6] V. Chudasama,et al. Cysteine protecting groups: applications in peptide and protein science. , 2021, Chemical Society reviews.
[7] M. Kannavou,et al. Liposomes Decorated with 2-(4'-Aminophenyl)benzothiazole Effectively Inhibit Aβ1-42 Fibril Formation and Exhibit in Vitro Brain-Targeting Potential. , 2020, Biomacromolecules.
[8] Sumit,et al. Advancement in Pharmacological Activities of Benzothiazole and its Derivatives:An Up to Date Review. , 2020, Mini reviews in medicinal chemistry.
[9] Y. Mabkhot,et al. Benzothiazoles as potential antiviral agents , 2020, The Journal of pharmacy and pharmacology.
[10] M. Yar,et al. Free radical scavengers: An overview on heterocyclic advances and medicinal prospects. , 2020, European journal of medicinal chemistry.
[11] E. Pioro,et al. Real-world evidence of riluzole effectiveness in treating amyotrophic lateral sclerosis , 2020, Amyotrophic lateral sclerosis & frontotemporal degeneration.
[12] Tian-Yi Zhang,et al. Synthesis, biological evaluation of benzothiazole derivatives bearing a 1,3,4-oxadiazole moiety as potential anti-oxidant and anti-inflammatory agents. , 2020, Bioorganic & medicinal chemistry letters.
[13] Xiang Gao,et al. Recent Advances in Synthesis of Benzothiazole Compounds Related to Green Chemistry , 2020, Molecules.
[14] B. C. Uzuegbunam,et al. PET Radiopharmaceuticals for Alzheimer’s Disease and Parkinson’s Disease Diagnosis, the Current and Future Landscape , 2020, Molecules.
[15] Zhi‐Bing Dong,et al. A Review on Domino Condensation/Cyclization Reactions for the Synthesis of 2-Substituted 1,3-Benzothiazole Derivatives , 2020 .
[16] M. Yar,et al. Synthetic strategy and SAR studies of C-glucoside heteroaryls as SGLT2 inhibitor: A review. , 2019, European journal of medicinal chemistry.
[17] C. Supuran,et al. Benzothiazole derivatives as anticancer agents , 2019, Journal of enzyme inhibition and medicinal chemistry.
[18] A. Abadi,et al. Structure-activity relationships of thiazole and benzothiazole derivatives as selective cannabinoid CB2 agonists with in vivo anti-inflammatory properties. , 2019, European journal of medicinal chemistry.
[19] A. Husain,et al. Novel hybrids of benzothiazole-1,3,4-oxadiazole-4-thiazolidinone: Synthesis, in silico ADME study, molecular docking and in vivo anti-diabetic assessment. , 2019, Bioorganic chemistry.
[20] Dongyu Zhang,et al. Recent developments in benzothiazole-based iridium(Ⅲ) complexes for application in OLEDs as electrophosphorescent emitters , 2019, Organic Electronics.
[21] V. Psycharis,et al. Remarkable Brain Penetration of Cyclopentadienyl M(CO)3+ (M = 99mTc, Re) Derivatives of Benzothiazole and Benzimidazole Paves the Way for Their Application as Diagnostic, with Single-Photon-Emission Computed Tomography (SPECT), and Therapeutic Agents for Alzheimer's Disease. , 2019, Journal of medicinal chemistry.
[22] M. Amir,et al. Design, Synthesis, and Screening of Hybrid Benzothiazolyl-Oxadiazoles as Anticonvulsant Agents , 2018 .
[23] G. Loudos,et al. 2-(4'-Aminophenyl)benzothiazole Labeled with 99mTc-Cyclopentadienyl for Imaging β-Amyloid Plaques. , 2017, ACS medicinal chemistry letters.
[24] Mengchao Cui,et al. Recent progress in the development of metal complexes as β-amyloid imaging probes in the brain. , 2017, MedChemComm.
[25] M. Gioia,et al. One-pot synthesis of amides from carboxylic acids activated using thionyl chloride , 2016 .
[26] Y. Keum,et al. Chrysin-benzothiazole conjugates as antioxidant and anticancer agents. , 2015, Bioorganic & medicinal chemistry letters.
[27] Rangappa S. Keri,et al. A comprehensive review in current developments of benzothiazole-based molecules in medicinal chemistry. , 2015, European journal of medicinal chemistry.
[28] T. Pabst,et al. Short Synthesis of a Proline Amide Orexin Receptor Antagonist on the Pilot Plant Scale , 2014 .
[29] Rajesh H. Vekariya,et al. Recent advances in the synthesis of 2-substituted benzothiazoles: a review , 2014 .
[30] A. McNeil,et al. Enzyme-triggered gelation: targeting proteases with internal cleavage sites. , 2014, Chemical communications.
[31] Y. Kimura,et al. Novel Synthetic Method for the Vilsmeier-Haack Reagent and Green Routes to Acid Chlorides, Alkyl Formates, and Alkyl Chlorides , 2013 .
[32] Xiaopeng Hu,et al. Zopolrestat as a Human Glyoxalase I Inhibitor and Its Structural Basis , 2013, ChemMedChem.
[33] Andreas F. M. Kilbinger,et al. Tuning the solubility of hepta(p-benzamide)s via the monomer sequence , 2013 .
[34] T. Kawase,et al. An Effective Synthesis of N,N-Dimethylamides from Carboxylic Acids and a New Route from N,N-Dimethylamides to 1,2-Diaryl-1,2-diketones. , 2011 .
[35] T. Kawase,et al. An effective synthesis of N,N-dimethylamides from carboxylic acids and a new route from N,N-dimethylamides to 1,2-diaryl-1,2-diketones , 2010 .
[36] F. Albericio,et al. PyOxP and PyOxB: the Oxyma-based novel family of phosphonium salts. , 2010, Organic & biomolecular chemistry.
[37] D. Gatos,et al. Synthesis of the very acid-sensitive Fmoc-Cys(Mmt)-OH and its application in solid-phase peptide synthesis. , 2009, International journal of peptide and protein research.
[38] T. Singh,et al. Synthesis of New Thiazolylthiazolidinylbenzothiazoles and Thiazolylazetidinylbenzothiazoles as Potential Insecticidal, Antifungal, and Antibacterial Agents , 2006, Archiv der Pharmazie.
[39] P. K. Basniwal,et al. 2-(4-aminophenyl) benzothiazole: a potent and selective pharmacophore with novel mechanistic action towards various tumour cell lines. , 2006, Mini reviews in medicinal chemistry.
[40] A. Westwell,et al. The development of the antitumour benzothiazole prodrug, Phortress, as a clinical candidate. , 2004, Current medicinal chemistry.
[41] M. Stevens,et al. Antitumor benzothiazoles. 16. Synthesis and pharmaceutical properties of antitumor 2-(4-aminophenyl)benzothiazole amino acid prodrugs. , 2002, Journal of medicinal chemistry.
[42] S. Mourtas,et al. Solid phase synthesis of benzothiazolyl compounds , 2001 .
[43] D. Gatos,et al. Convergent Peptide Synthesis , 2000 .
[44] G. Dozeman,et al. Chemical Development of a Pilot Scale Process for the ACAT Inhibitor 2, 6-Diisopropylphenyl ((2,4,6-Triisopropylphenyl)acetyl)sulfamate. , 1997 .
[45] S Wrigley,et al. Antitumor benzothiazoles. 3. Synthesis of 2-(4-aminophenyl)benzothiazoles and evaluation of their activities against breast cancer cell lines in vitro and in vivo. , 1996, Journal of medicinal chemistry.
[46] L. A. Carpino. 1-Hydroxy-7-azabenzotriazole. An efficient peptide coupling additive , 1993 .
[47] F. Higashi,et al. Direct polyamidation with thionyl chloride in N‐methyl‐pyrrolidone , 1986 .
[48] P. M. Hardy. PROTECTING GROUPS IN PEPTIDE SYNTHESIS , 1980 .
[49] N. Semenov,et al. A New Look at the Chalcogen Bond: π-Hole-based Chalcogen (Se, Te) Bonding Which Does Not Include a σ-Hole Interaction , 2023, Inorganic Chemistry Frontiers.
[50] R. Liu,et al. Panchromatic luminescent D-π-A benzothiazoles with different π-bridging modulation: design, synthesis and application in WLEDs devices , 2023, Materials Chemistry Frontiers.
[51] A. Cherkasov,et al. Metal-involving C···dz2-PtII Tetrel Bonding as a Principal Component of Stacking Interaction between Arenes and the Platinum(II) Square-plane , 2023, Inorganic Chemistry Frontiers.
[52] É. Tóth,et al. Metal complexes for the visualisation of amyloid peptides , 2022, Sensors & Diagnostics.
[53] E. Rathi,et al. A review on anticancer potentials of benzothiazole derivatives. , 2019, Mini reviews in medicinal chemistry.
[54] Ashish A. Gawai,et al. Synthesis, Preliminary Pharmacological and Acute Toxicity Studies of a New Series of 7-(2-(Benzo[d]thiazol-2-ylamino)ethoxy)-4-methyl-2H-chromen-2-one Derivatives with Atypical Antipsychotic Activity , 2019, Indian Journal of Pharmaceutical Sciences.
[55] C. P. Rao,et al. Synthesis, characterization and biological evaluation of benzothiazole derivatives as potential antimicrobial and analgesic agents , 2017 .
[56] S. Mourtas,et al. Resin-bound aminothiols: synthesis and application , 2003 .
[57] W. Chan,et al. Fmoc Solid Phase Peptide Synthesis: A Practical Approach (Practical Approach Series) , 2019 .
[58] B. Merrifield,et al. Concept and early development of solid-phase peptide synthesis. , 1997, Methods in enzymology.
[59] E. Giralt,et al. Convergent solid-phase peptide synthesis. , 1997, Methods in enzymology.
[60] B. Mylari,et al. Novel, potent aldose reductase inhibitors: 3,4-dihydro-4-oxo-3-[[5-(trifluoromethyl)-2-benzothiazolyl] methyl]-1-phthalazineacetic acid (zopolrestat) and congeners. , 1991, Journal of medicinal chemistry.