Drug-lipid interaction evaluation: why a 19th century solution?
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Miguel A R B Castanho | Manuel N Melo | N. Santos | M. Castanho | Nuno C Santos | Marta M B Ribeiro | Isa D Serrano | I. Serrano | M. Melo | M. M. B. Ribeiro
[1] James I. Wells,et al. Pharmaceutical preformulation : the physicochemical properties of drug substances , 1988 .
[2] J. Mocák,et al. Chemometrical study of the anaesthetical activity of alkoxyphenylcarbamic acid esters. , 2010, Die Pharmazie.
[3] Edward A Dennis,et al. Lipidomics joins the omics evolution , 2009, Proceedings of the National Academy of Sciences.
[4] Charles Tanford,et al. The Hydrophobic Effect: Formation of Micelles and Biological Membranes , 1991 .
[5] Marco M. Domingues,et al. Fold-unfold transitions in the selectivity and mechanism of action of the N-terminal fragment of the bactericidal/permeability-increasing protein (rBPI(21)). , 2009, Biophysical journal.
[6] Miguel A R B Castanho,et al. An overview of the biophysical applications of atomic force microscopy. , 2003, Biophysical chemistry.
[7] Hinrich W. H. Göhlmann,et al. Pharmaceutical R&D , 2009 .
[8] A. J. Staverman,et al. The entropy of liquid mixtures: I. The theory of Raoult's Law , 2010 .
[9] Bernard Testa,et al. Immobilized artificial membrane HPLC in drug research. , 2003, Journal of medicinal chemistry.
[10] S. Singer,et al. The Fluid Mosaic Model of the Structure of Cell Membranes , 1972, Science.
[11] S. Krämer,et al. The pH-Dependence in the Partitioning Behaviour of (RS)-[3H]Propranolol Between MDCK Cell Lipid Vesicles and Buffer , 1996, Pharmaceutical Research.
[12] H. Wu,et al. Binding of peptides with basic residues to membranes containing acidic phospholipids. , 1991, Biophysical journal.
[13] T. Hartmann,et al. Lipophilicity - beyond octanol/water: a short comparison of modern technologies. , 2004, Drug discovery today. Technologies.
[14] D. Müller. AFM: a nanotool in membrane biology. , 2008 .
[15] A. Ghose,et al. Prediction of Hydrophobic (Lipophilic) Properties of Small Organic Molecules Using Fragmental Methods: An Analysis of ALOGP and CLOGP Methods , 1998 .
[16] Jörg Keldenich,et al. Multilamellar Liposomes and Solid-Supported Lipid Membranes (TRANSIL): Screening of Lipid-Water Partitioning Toward a High-Throughput Scale , 2001, Pharmaceutical Research.
[17] R. Daniels,et al. Pharmaceutical Preformulation – The Physicochemical Properties of Drug Substances ‐ von James I. Wells, 227 S., 47 Abb., 99 Tab., Preis: £ 35.00, Ellis Horwood Limited, Chichester, England 1988 , 1989 .
[18] Caron,et al. Combined molecular lipophilicity descriptors and their role in understanding intramolecular effects. , 1999, Pharmaceutical science & technology today.
[19] Kerly F. M. Pasqualoto,et al. QSAR Modeling of a Set of Pyrazinoate Esters as Antituberculosis Prodrugs , 2010, Archiv der Pharmazie.
[20] C. Pidgeon,et al. Membrane partition coefficients chromatographically measured using immobilized artificial membrane surfaces. , 1995, Analytical chemistry.
[21] H. Meyer. Zur Theorie der Alkoholnarkose , 1899, Archiv für experimentelle Pathologie und Pharmakologie.
[22] Emilio Benfenati,et al. QSPR modeling of octanol/water partition coefficient of antineoplastic agents by balance of correlations. , 2010, European journal of medicinal chemistry.
[23] J. Richmond. The 3Rs - Past, Present and Future , 2000 .
[24] M. N. Melo,et al. Antimicrobial peptides: linking partition, activity and high membrane-bound concentrations , 2009, Nature Reviews Microbiology.
[25] W. Nernst. Verteilung eines Stoffes zwischen zwei Lösungsmitteln und zwischen Lösungsmittel und Dampfraum , 1891 .
[26] G. Hodges,et al. Practical methods for the measurement of logP for surfactants. , 2010, Ecotoxicology and environmental safety.
[27] Pickett,et al. Computational methods for the prediction of 'drug-likeness' , 2000, Drug discovery today.
[28] Michael R. Yeaman,et al. Mechanisms of Antimicrobial Peptide Action and Resistance , 2003, Pharmacological Reviews.
[29] J. Seelig,et al. Correlation of membrane/water partition coefficients of detergents with the critical micelle concentration. , 2000, Biophysical journal.
[30] D. Marsh,et al. Cholesterol-induced fluid membrane domains: a compendium of lipid-raft ternary phase diagrams. , 2009, Biochimica et biophysica acta.
[31] Manuel Prieto,et al. Quantifying molecular partition into model systems of biomembranes: an emphasis on optical spectroscopic methods. , 2003, Biochimica et biophysica acta.
[32] D. Sargent,et al. Membrane lipid phase as catalyst for peptide-receptor interactions. , 1986, Proceedings of the National Academy of Sciences of the United States of America.
[33] H. Riezman,et al. Lipid pickup and delivery , 2004, Nature Cell Biology.
[34] I. Bronshtein,et al. On the Correlation Between Hydrophobicity, Liposome Binding and Cellular Uptake of Porphyrin Sensitizers , 2006, Photochemistry and photobiology.
[35] H. Mewes,et al. Can we estimate the accuracy of ADME-Tox predictions? , 2006, Drug discovery today.
[36] R. Austin,et al. Partitioning of ionizing molecules between aqueous buffers and phospholipid vesicles. , 1995, Journal of pharmaceutical sciences.
[37] M Balls,et al. Replacement of animal procedures: alternatives in research, education and testing , 1994, Laboratory animals.
[38] N. Santos,et al. Interaction of peptides with biomembranes assessed by potential‐sensitive fluorescent probes , 2008, Journal of peptide science : an official publication of the European Peptide Society.
[39] F. Szoka,et al. Comparative properties and methods of preparation of lipid vesicles (liposomes). , 1980, Annual review of biophysics and bioengineering.
[40] A. Fedorov,et al. Lipidic Membranes Are Potential “Catalysts” in the Ligand Activity of the Multifunctional Pentapeptide Neokyotorphin , 2005, Chembiochem : a European journal of chemical biology.
[41] Alan E Mark,et al. University of Groningen Alternative Mechanisms for the Interaction of the Cell-Penetrating Peptides Penetratin and the TAT Peptide with Lipid Bilayers Yesylevskyy, , 2009 .
[42] M. Khaledi,et al. Interaction of Basic Drugs with Lipid Bilayers Using Liposome Electrokinetic Chromatography , 2004, Pharmaceutical Research.
[43] I. Belostotsky,et al. Mitochondrial targeting for photochemotherapy. Can selective tumor cell killing be predicted based on n-octanol/water distribution coefficients? , 2011, Biotechnic & histochemistry : official publication of the Biological Stain Commission.
[44] M. Castanho,et al. Lipid membrane-induced optimization for ligand–receptor docking: recent tools and insights for the “membrane catalysis” model , 2005, European Biophysics Journal.
[45] E. Ikonen,et al. Functional rafts in cell membranes , 1997, Nature.
[46] E. Blout,et al. Conformation of gramicidin A in phospholipid vesicles: circular dichroism studies of effects of ion binding, chemical modification, and lipid structure. , 1981, Biochemistry.
[47] S. Schreier,et al. EPR STUDY OF MEMBRANE PARTITIONING, ORIENTATION, AND MEMBRANE-MODULATED ALKALINE HYDROLYSIS OF A SPIN-LABELED BENZOIC ACID ESTER , 1991 .
[48] S. H. Lin,et al. Membrane-buffer partition coefficients of tetracaine for liquid-crystal and solid-gel membranes estimated by direct ultraviolet spectrophotometry. , 1988, Biochimica et biophysica acta.
[49] L. Mayer,et al. Vesicles of variable sizes produced by a rapid extrusion procedure. , 1986, Biochimica et biophysica acta.
[50] E. Gratton,et al. Lipid--protein interactions revealed by two-photon microscopy and fluorescence correlation spectroscopy. , 2005, Accounts of chemical research.
[51] Frédéric Pincet,et al. Giant vesicles formed by gentle hydration and electroformation: a comparison by fluorescence microscopy. , 2005, Colloids and surfaces. B, Biointerfaces.
[52] S. Semrau,et al. Membrane heterogeneity – from lipid domains to curvature effects , 2009 .