Binding Method for Detection of Muscarinic Acetylcholine Receptors in Receptor’s Natural Environment
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K. Sada | T. Masuoka | T. Taniguchi | I. Muramatsu | J. Uwada | M. Nishio | H. Yoshiki | Junsuke Uwada
[1] M. Kainoh,et al. Pharmacologically distinct phenotypes of α1B‐adrenoceptors: variation in binding and functional affinities for antagonists , 2014, British journal of pharmacology.
[2] T. Masuoka,et al. Intracellular localization of the M1 muscarinic acetylcholine receptor through clathrin-dependent constitutive internalization is mediated by a C-terminal tryptophan-based motif , 2014, Journal of Cell Science.
[3] N. Matsuki,et al. Novel contribution of cell surface and intracellular M1‐muscarinic acetylcholine receptors to synaptic plasticity in hippocampus , 2013, Journal of neurochemistry.
[4] Arthur Christopoulos,et al. Bridging the gap: bitopic ligands of G-protein-coupled receptors. , 2013, Trends in pharmacological sciences.
[5] H. Ikeuchi,et al. M1 is a major subtype of muscarinic acetylcholine receptors on mouse colonic epithelial cells , 2013, Journal of Gastroenterology.
[6] A. Nishimune,et al. Regional quantification of muscarinic acetylcholine receptors and β‐adrenoceptors in human airways , 2012, British journal of pharmacology.
[7] A. Nishimune,et al. Phenotype pharmacology of lower urinary tract α1‐adrenoceptors , 2012, British journal of pharmacology.
[8] A. Nishimune,et al. Re-Evaluation of Nicotinic Acetylcholine Receptors in Rat Brain by a Tissue-Segment Binding Assay , 2011, Front. Pharmacol..
[9] A. Nishimune,et al. Influence of Tissue Integrity on Pharmacological Phenotypes of Muscarinic Acetylcholine Receptors in the Rat Cerebral Cortex , 2011, Journal of Pharmacology and Experimental Therapeutics.
[10] A. Nishimune,et al. Intracellular distribution of functional M1‐muscarinic acetylcholine receptors in N1E‐115 neuroblastoma cells , 2011, Journal of neurochemistry.
[11] D. Bylund,et al. Radioligand binding methods for membrane preparations and intact cells. , 2011, Methods in molecular biology.
[12] Laurence J. Miller,et al. Seven Transmembrane Receptors as Shapeshifting Proteins: The Impact of Allosteric Modulation and Functional Selectivity on New Drug Discovery , 2010, Pharmacological Reviews.
[13] A. Anisuzzaman,et al. Identification of M(1) muscarinic receptor subtype in rat stomach using a tissue segment binding method, and the effects of immobilization stress on the muscarinic receptors. , 2008, European journal of pharmacology.
[14] A. Anisuzzaman,et al. Different affinities of native alpha1B-adrenoceptors for ketanserin between intact tissue segments and membrane preparations. , 2008, European journal of pharmacology.
[15] J A Peters,et al. Guide to Receptors and Channels (GRAC), 3rd edition , 2008, British journal of pharmacology.
[16] H. Akino,et al. Assessment of muscarinic receptor subtypes in human and rat lower urinary tract by tissue segment binding assay. , 2008, Journal of Pharmacological Sciences.
[17] S. Hill,et al. Multiple GPCR conformations and signalling pathways: implications for antagonist affinity estimates , 2007, Trends in pharmacological sciences.
[18] R A John Challiss,et al. "Phenotypic" pharmacology: the influence of cellular environment on G protein-coupled receptor antagonist and inverse agonist pharmacology. , 2007, Biochemical pharmacology.
[19] S. Morishima,et al. Pharmacological evaluation of plasma membrane beta-adrenoceptors in rat hearts using the tissue segment binding method. , 2006, Life sciences.
[20] A. Anisuzzaman,et al. Quantifying receptor properties: the tissue segment binding method - a powerful tool for the pharmacome analysis of native receptors. , 2005, Journal of pharmacological sciences.
[21] Takashi Tanaka,et al. Identification of α-1L Adrenoceptor in Rabbit Ear Artery , 2004, Journal of Pharmacology and Experimental Therapeutics.
[22] Li Zhang,et al. Alpha‐1 adrenoceptors: evaluation of receptor subtype‐binding kinetics in intact arterial tissues and comparison with membrane binding , 2004, British journal of pharmacology.
[23] C. V. van Koppen,et al. Regulation of muscarinic acetylcholine receptor signaling. , 2003, Pharmacology & therapeutics.
[24] J. Faber,et al. Expression of α-Adrenoceptor Subtypes by Smooth Muscle Cells and Adventitial Fibroblasts in Rat Aorta and in Cell Culture , 2001 .
[25] J. Balligand,et al. Dynamin mediates caveolar sequestration of muscarinic cholinergic receptors and alteration in NO signaling , 2000, The EMBO journal.
[26] A. Ford,et al. Characterization of an atypical muscarinic cholinoceptor mediating contraction of the guinea‐pig isolated uterus , 1998, British journal of pharmacology.
[27] J. Pennefather,et al. Pharmacological characterization of muscarinic receptors in the uterus of oestrogen‐primed and pregnant rats , 1998, British journal of pharmacology.
[28] J. Edwardson,et al. Intracellular trafficking of the muscarinic acetylcholine receptor: importance of subtype and cell type. , 1996, Molecular pharmacology.
[29] T. Kenakin,et al. On the importance of the "antagonist assumption" to how receptors express themselves. , 1995, Biochemical pharmacology.
[30] F. Ehlert,et al. Regional distribution of M1, M2 and non-M1, non-M2 subtypes of muscarinic binding sites in rat brain. , 1990, The Journal of pharmacology and experimental therapeutics.
[31] A. Michel,et al. Affinity of muscarinic receptor antagonists for three putative muscarinic receptor binding sites , 1989, British journal of pharmacology.
[32] R. Sherman-Gold. Neurotransmitter receptor binding, 2nd edn: edited by Henry I. Yamamura, S. J. Enna and Michael J. Kuhar, Raven Press, 1985. US$58.00 (xiv + 242 pages), ISBN 0 88167 027 8 , 1985 .
[33] J. Galper,et al. The biphasic response of muscarinic cholinergic receptors in cultured heart cells to agonists. Effects on receptor number and affinity in intact cells and homogenates. , 1982, The Journal of biological chemistry.
[34] R. Alexander,et al. Regulation of the Postsynaptic α‐Adrenergic Receptor in Rat Mesenteric Artery: Effects of Chemical Sympathectomy and Epinephrine Treatment 1981 , 1981, Circulation research.
[35] J. Schwartz,et al. Pharmacological specificity of brain histamine H2-receptors differs in intact cells and cell-free preparations , 1980, Nature.
[36] H. Rang,et al. The uptake of atropine and related drugs by intestinal smooth muscle of the guinea-pig in relation to acetylcholine receptors , 1965, Proceedings of the Royal Society of London. Series B. Biological Sciences.