Diastereoselective Ugi reaction without chiral amines: the synthesis of chiral pyrroloketopiperazines

[1]  M. Mironov Design of Multi‐Component Reactions: From Libraries of Compounds to Libraries of Reactions , 2006 .

[2]  Alexander Dömling,et al.  Recent developments in isocyanide based multicomponent reactions in applied chemistry. , 2006, Chemical reviews.

[3]  S. Sollis Short and novel stereospecific synthesis of trisubstituted 2,5-diketopiperazines. , 2005, The Journal of organic chemistry.

[4]  Andrea Basso,et al.  A novel highly selective chiral auxiliary for the asymmetric synthesis of L- and D-alpha-amino acid derivatives via a multicomponent Ugi reaction. , 2005, The Journal of organic chemistry.

[5]  Alexey P. Ilyn,et al.  AN EFFICIENT SYNTHESIS OF 3-OXO-1,2,3,4-TETRAHYDROPYRROLO[1,2-α]PYRAZINE-1-CARBOXAMIDES USING NOVEL MODIFICATION OF UGI CONDENSATION , 2005 .

[6]  Jieping Zhu Recent Developments in the Isonitrile‐Based Multicomponent Synthesis of Heterocycles , 2003 .

[7]  I. Ugi,et al.  Stereoselective U-4CRS with 1-amino-5-desoxy-5-thio-2,3,4-O-isobutanoyl-β-d-xylopyranose: an effective and selectively removable chiral auxiliary , 2002 .

[8]  R. Nutt,et al.  Concise total synthesis of the prolyl endopeptidase inhibitor eurystatin A via a novel Passerini reaction–deprotection–acyl migration strategy , 2001 .

[9]  C. Willis,et al.  Ugi four component condensations using aldehydes with an asymmetric centre at C-2 , 2000 .

[10]  I. Ugi,et al.  Multicomponent Reactions with Isocyanides. , 2000, Angewandte Chemie.

[11]  T. Ziegler,et al.  PASSERINI AND UGI REACTIONS OF BENZYL AND ACETYL PROTECTED ISOCYANOGLUCOSES , 1999 .

[12]  W. Herlihy,et al.  Unique Structures Generated by Ugi 3CC Reactions Using Bifunctional Starting Materials Containing Aldehyde and Carboxylic Acid. , 1999, The Journal of organic chemistry.

[13]  M. Murata,et al.  Novel, highly potent aldose reductase inhibitors: (R)-(-)-2-(4-bromo-2-fluorobenzyl)-1,2,3,4- tetrahydropyrrolo[1,2-a]pyrazine -4-spiro-3'-pyrrolidine-1,2',3,5'-tetrone (AS-3201) and its congeners. , 1998, Journal of medicinal chemistry.

[14]  T. Ziegler,et al.  PASSERINI AND UGI REACTIONS OF ANOMERIC GLUCOSYL ISONITRILES , 1998 .

[15]  H. Kunz,et al.  Asymmetric synthesis on carbohydrate templates: stereoselective Ugi-synthesis of .alpha.-amino acid derivatives , 1988 .

[16]  H. Kunz,et al.  Diastereoselective Strecker Synthesis of α‐Aminonitriles on Carbohydrate Templates , 1987 .

[17]  T. Chan,et al.  1,4-Dichloro-1,4-dimethoxybutane as a mild reagent for the conversion of primary amines to pyrroles. Synthesis of a pyrrole compound from tobacco , 1983 .

[18]  G. Olah,et al.  Synthetic methods and reactions. 62. Transformations with chlorotrimethylsilane/sodium iodide, a convenient in situ iodotrimethylsilane reagent , 1979 .

[19]  R. C. Erickson,et al.  Semisynthetic cephalosporins. Synthesis and structure-activity relationships of 7-(1-pyrryl)- and 7-(1-indolyl)acetamidocephalosporin derivatives. , 1978, Journal of medicinal chemistry.

[20]  I. Ugi,et al.  Stereoselective syntheses. V. Isonitriles. XXIV. Stereoselective four-component condensations of .alpha.-ferrocenylethylamine and its absolute configuration , 1970 .

[21]  I. Ugi,et al.  Stereoselektive Synthesen, III. Die Umsetzung von (S)‐α‐Phenyläthylamin und Isobutyraldehyd mit Benzoesäure und tert.‐Butyl‐isocyanid als Modellreaktion für stereoselektive Peptid‐Synthesen mittels Vierkomponenten‐Kondensationen , 1967 .

[22]  Ivar Ugi,et al.  Stereoselektive Synthesen, IV. Der Reaktionsmechanismus stereoselektiver Vierkomponenten‐Kondensationen , 1967 .