Discovery and structure-activity relationship of (1R)-8-chloro-2,3,4,5-tetrahydro-1-methyl-1H-3-benzazepine (Lorcaserin), a selective serotonin 5-HT2C receptor agonist for the treatment of obesity.
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Brian M. Smith | F. Menzaghi | P. Dosa | N. Beeley | Jeffrey M Smith | J. Tsai | J. Schultz | C. Gilson | Scott A. Estrada | Rita R Chen | Douglas M Park | Emily B Prieto | C. Gallardo | D. Sengupta | John Covel | Albert S. Ren | R. Webb | Michael Martin | Michael E. Morgan | S. Espitia | Hazel R Saldana | C. Bjenning | K. Whelan | A. Grottick | W. Thomsen