Synthesis of [11C-methyl]-(-)-OSU6162, its regional brain distribution and some pharmacological effects of (-)-OSU6162 on the dopaminergic system studied in the rhesus monkey by positron emission tomography.

[1]  L. Hansson,et al.  On the quantitative structure-activity relationships of meta-substituted (S)-phenylpiperidines, a class of preferential dopamine D2 autoreceptor ligands: modeling of dopamine synthesis and release in vivo by means of partial least squares regression. , 1995, Journal of medicinal chemistry.

[2]  C. Sonesson,et al.  AN EFFICIENT SYNTHESIS OF THE NOVEL DOPAMINE AUTORECEPTOR ANTAGONIST S-(-)-OSU6162, VIA PALLADIUM CATALYZED CROSS-COUPLING REACTION , 1994 .

[3]  A. Carlsson,et al.  Substituted (S)-phenylpiperidines and rigid congeners as preferential dopamine autoreceptor antagonists: synthesis and structure-activity relationships. , 1994, Journal of medicinal chemistry.

[4]  J S Fowler,et al.  Striatal binding of the PET ligand 11C‐raclopride is altered by drugs that modify synaptic dopamine levels , 1993, Synapse.

[5]  Bruno Giros,et al.  Localization of dopamine D3 receptor mRNA in the rat brain using in situ hybridization histochemistry: comparison with dopamine D2 receptor mRNA , 1991, Brain Research.

[6]  David J. Brooks,et al.  A Two-Compartment Description and Kinetic Procedure for Measuring Regional Cerebral [11C]Nomifensine Uptake Using Positron Emission Tomography , 1990, Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism.

[7]  G. Antoni,et al.  Synthesis of L- and D-[methyl-11C]methionine. , 1987, Journal of nuclear medicine : official publication, Society of Nuclear Medicine.

[8]  G. Chiara,et al.  Haloperidol increases and apomorphine decreases striatal dopamine metabolism after destruction of striatal dopamine-sensitive adenylate cyclase by kainic acid , 1977, Brain Research.

[9]  M. Newman,et al.  The Conversion of Phenols to Thiophenols via Dialkylthiocarbamates1 , 1966 .