Preclinical studies on [11C]TMSX for mapping adenosine A2A receptors by positron emission tomography
暂无分享,去创建一个
Yuichi Kimura | Kiichi Ishiwata | Kenji Ishii | Kazunori Kawamura | K. Ishii | Y. Kimura | K. Ishiwata | K. Kawamura | Wei-Fang Wang | Wei-fang Wang
[1] M. Kiyosawa,et al. Evaluation of carbon-11 labeled KF15372 and its ethyl and methyl derivatives as a potential CNS adenosine A1 receptor ligand. , 1997, Nuclear medicine and biology.
[2] M. Kiyosawa,et al. Carbon-11-labeled KF21213: a highly selective ligand for mapping CNS adenosine A(2A) receptors with positron emission tomography. , 2000, Nuclear medicine and biology.
[3] M. Senda,et al. Myocardial adenosine A2a receptor imaging of rabbit by PET with [11C]KF17837 , 1997, Annals of nuclear medicine.
[4] E. Fuse,et al. Adenosine A1 antagonists. 3. Structure-activity relationships on amelioration against scopolamine- or N6-((R)-phenylisopropyl)adenosine-induced cognitive disturbance. , 1993, Journal of medicinal chemistry.
[5] M. Senda,et al. 11C-labeled KF18446: a potential central nervous system adenosine A2a receptor ligand. , 2000, Journal of nuclear medicine : official publication, Society of Nuclear Medicine.
[6] Mauro Papotti,et al. Immunohistochemical localization of adenosine A1 receptors in human brain regions , 2001, Neuroscience Letters.
[7] M. Avoli,et al. Upregulation of A1 adenosine receptors in human temporal lobe epilepsy: A quantitative autoradiographic study , 1993, Neuroscience Letters.
[8] S. Synder,et al. Autoradiographic localization of adenosine receptors in rat brain using [3H]cyclohexyladenosine , 1982, The Journal of neuroscience : the official journal of the Society for Neuroscience.
[9] R. Faull,et al. Alzheimer's disease: Changes in hippocampal N-methyl-d-aspartate, quisqualate, neurotensin, adenosine, benzodiazepine, serotonin and opioid receptors—an autoradiographic study , 1990, Neuroscience.
[10] T. Dunwiddie,et al. The Role and Regulation of Adenosine in the Central Nervous System , 2022 .
[11] G Burnstock,et al. Nomenclature and Classification of Purinoceptors* , 2005 .
[12] C. Cotman,et al. Reduced density of adenosine A1 receptors and preserved coupling of adenosine A1 receptors to G proteins in alzheimer hippocampus: A quantitative autoradiographic study , 1993, Neuroscience.
[13] D. Lubitz. Adenosine in the treatment of stroke: yes, maybe, or absolutely not? , 2001 .
[14] E. Broussolle,et al. Contributions of PET and SPECT to the understanding of the pathophysiology of Parkinson’s disease , 2001, Neurophysiologie Clinique/Clinical Neurophysiology.
[15] F Suzuki,et al. (E)-1,3-dialkyl-7-methyl-8-(3,4,5-trimethoxystyryl)xanthines: potent and selective adenosine A2 antagonists. , 1992, Journal of medicinal chemistry.
[16] J. Fastbom,et al. Adenosine A1 receptors in the human brain: A quantitative autoradiographic study , 1987, Neuroscience.
[17] E. Wolters,et al. IBZM- and CIT-SPECT of the dopaminergic system in parkinsonism. , 1997, Journal of neural transmission. Supplementum.
[18] B. Fredholm,et al. Further characterization of the binding of the adenosine receptor agonist [3H]CGS 21680 to rat brain using autoradiography , 1995, Neuropharmacology.
[19] H Toyama,et al. Synthesis and preliminary evaluation of [11C]KF17837, a selective adenosine A2A antagonist. , 1996, Applied radiation and isotopes : including data, instrumentation and methods for use in agriculture, industry and medicine.
[20] B. Fredholm,et al. Pharmacology of adenosine A2A receptors. , 1996, Trends in pharmacological sciences.
[21] H. Kase,et al. Photoisomerization of a potent and selective adenosine A2 antagonist, (E)-1,3-Dipropyl-8-(3,4-dimethoxystyryl)-7-methylxanthine. , 1993, Journal of medicinal chemistry.
[22] M. E. Lewis,et al. Autoradiographic visualization of rat brain adenosine receptors using N6-cyclohexyl [3H]adenosine. , 1981, European journal of pharmacology.
[23] S. Schiffmann,et al. Striatal Restricted Adenosine A2 Receptor (RDC8) Is Expressed by Enkephalin but Not by Substance P Neurons: An In Situ Hybridization Histochemistry Study , 1991, Journal of neurochemistry.
[24] Helmut L. Haas,et al. Functions of neuronal adenosine receptors , 2000, Naunyn-Schmiedeberg's Archives of Pharmacology.
[25] H Toyama,et al. A PET study of adenosine A1 receptor in anesthetized monkey brain. , 2000, Nuclear medicine and biology.
[26] M. Senda,et al. Evaluation of carbon-11-labeled KF17837: a potential CNS adenosine A2a receptor ligand. , 1998, Journal of nuclear medicine : official publication, Society of Nuclear Medicine.
[27] G. Wooten,et al. Differential localization of A2a adenosine receptor mRNA with D1 and D2 dopamine receptor mRNA in striatal output pathways following a selective lesion of striatonigral neurons , 1993, Brain Research.
[28] M. Senda,et al. Synthesis and in vivo evaluation of [11C]semotiadil, a benzothiazine calcium antagonist. , 1994, Applied radiation and isotopes : including data, instrumentation and methods for use in agriculture, industry and medicine.
[29] K. Ishiwata,et al. Synthesis and radiation dosimetry of 4-borono-2-[18F]fluoro-D,L-phenylalanine: a target compound for PET and boron neutron capture therapy. , 1991, International journal of radiation applications and instrumentation. Part A, Applied radiation and isotopes.
[30] J. Fastbom,et al. The distribution of adenosine a1 receptors and 5'-nucleotidase in the brain of some commonly used experimental animals , 1987, Neuroscience.
[31] Keiichi Oda,et al. Adenosine A2A receptor imaging with [11C]KF18446 PET in the rat brain after quinolinic acid lesion: Comparison with the dopamine receptor imaging , 2002, Annals of nuclear medicine.
[32] M. Senda,et al. Synthesis and preliminary evaluation of [11C]KF17837, a selective adenosine A2A antagonist. , 1996, Applied radiation and isotopes : including data, instrumentation and methods for use in agriculture, industry and medicine.
[33] J. Málly,et al. Potential role of adenosine antagonist therapy in pathological tremor disorders. , 1996, Pharmacology & therapeutics.
[34] B B Fredholm,et al. Distribution of adenosine receptors in the postmortem human brain: An extended autoradiographic study , 1997, Synapse.
[35] B. Fredholm,et al. Autoradiographic evidence for G-protein coupled A2-receptors in rat neostriatum using [3H]-CGS 21680 as a ligand , 1990, Naunyn-Schmiedeberg's Archives of Pharmacology.
[36] T. Yamashita,et al. A high resolution PET for animal studies , 1991, Conference Record of the 1991 IEEE Nuclear Science Symposium and Medical Imaging Conference.
[37] C. Gerfen,et al. D1 and D2 dopamine receptor-regulated gene expression of striatonigral and striatopallidal neurons. , 1990, Science.
[38] Stoessl Aj,et al. NEURORECEPTOR IMAGING : NEW DEVELOPMENTS IN PET AND SPECT IMAGING OF NEURORECEPTOR BINDING (INCLUDING DOPAMINE TRANSPORTERS, VESICLE TRANSPORTERS AND POST SYNAPTIC RECEPTOR SITES) , 1998 .
[40] K. Kubo,et al. Adenosine A1 antagonists. 2. Structure-activity relationships on diuretic activities and protective effects against acute renal failure. , 1992, Journal of medicinal chemistry.
[41] K. Kubo,et al. 8-(Dicyclopropylmethyl)-1,3-dipropylxanthine: a potent and selective adenosine A1 antagonist with renal protective and diuretic activities. , 1991, Journal of medicinal chemistry.
[42] Tadashi Nariai,et al. Mapping adenosine A1 receptors in the cat brain by positron emission tomography with [11C]MPDX , 2002 .
[43] M. Kiyosawa,et al. Carbon-11-labeled KF15372: a potential central nervous system adenosine A1 receptor ligand. , 1996, Journal of nuclear medicine : official publication, Society of Nuclear Medicine.
[44] H. Watabe,et al. Absorbed dose estimates in positron emission tomography studies based on the administration of 18F-labeled radiopharmaceuticals. , 1991, Journal of radiation research.
[45] M. Senda,et al. Further characterization of a CNS adenosine A2a receptor ligand [11C]KF18446 within vitro autoradiography andin vivo tissue uptake , 2000, Annals of nuclear medicine.
[46] Evaluation of iodinated and brominated [11C]styrylxanthine derivatives asin vivo radioligands mapping adenosine A2A receptor in the central nervous system , 2000, Annals of nuclear medicine.
[47] H. Kase. New Aspects of Physiological and Pathophysiological Functions of Adenosine A2A Receptor in Basal Ganglia , 2001, Bioscience, biotechnology, and biochemistry.
[48] S. Augood,et al. Adenosine A2a receptor mRNA is expressed by enkephalin cells but not by somatostatin cells in rat striatum: a co-expression study. , 1994, Brain research. Molecular brain research.
[49] K. Ishii,et al. Assessment of adenosine A2A receptors with PET as a new diagnostic tool for neurological disorders , 2002 .
[50] M. Kiyosawa,et al. Neuroreceptor bindings and synaptic activity in visual system of monocularly enucleated rat. , 2001, Japanese journal of ophthalmology.
[51] S. File,et al. Depletion in amygdaloid 5-hydroxytryptamine concentration and changes in social and aggressive behaviour , 2005, Journal of Neural Transmission.