Synthesis of functionalized 3-, 5-, 6- and 8-aminoquinolines via intermediate (3-pyrrolin-1-yl)- and (2-oxopyrrolidin-1-yl)quinolines and evaluation of their antiplasmodial and antifungal activity.
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Philip Smith | K. Chibale | C. de Kock | T. Desmet | Stéphanie Vandekerckhove | M. D’hooghe | B. Danneels | J. Willems | Sofie Van Herreweghe