Design, synthesis, and biological evaluation of C1-phosphonamidate analogues of 2-deoxy-d-ribose-1-phosphate

[1]  J. Balzarini,et al.  Synthesis and biological evaluation of prodrugs of 2-fluoro-2-deoxyribose-1-phosphate and 2,2-difluoro-2-deoxyribose-1-phosphate , 2013, Bioorganic & Medicinal Chemistry Letters.

[2]  J. Balzarini,et al.  Inhibition of pyrimidine and purine nucleoside phosphorylases by a 3,5-dichlorobenzoyl-substituted 2-deoxy-D-ribose-1-phosphate derivative. , 2012, Biochemical pharmacology.

[3]  Mauro F. A. Adamo,et al.  Studies on the generation of unnatural C-nucleosides with 1-alkynyl-2-deoxy-D-riboses. , 2007, Organic letters.

[4]  F. Nicotra.  Synthesis of Glycosyl Phosphate Mimics , 2005 .

[5]  E. Clercq,et al.  Discovery and development of BVDU (brivudin) as a therapeutic for the treatment of herpes zoster. , 2004 .

[6]  R. B. Nazarski,et al.  [(Diphenoxyphosphinyl)methylidene]triphenylphosphorane—the double P+-stabilised carbanion: a crystallographic, computational and solution NMR comparative study on the ylidic bonding , 2003 .

[7]  Michael Bosco,et al.  Synthesis of sugar-derived phostones by activation of γ-hydroxyphosphonic acids , 2003 .

[8]  T. Lowary,et al.  Synthesis and antituberculosis activity of C-phosphonate analogues of decaprenolphosphoarabinose, a key intermediate in the biosynthesis of mycobacterial arabinogalactan and lipoarabinomannan. , 2002, The Journal of organic chemistry.

[9]  D. Stepinski,et al.  Facile High-Yielding Synthesis of Symmetric Esters of Methylenebisphosphonic Acid. , 2001 .

[10]  E. De Clercq,et al.  Synthesis and evaluation of novel amidate prodrugs of PMEA and PMPA. , 2001, Bioorganic & medicinal chemistry letters.

[11]  J. Balzarini,et al.  Syntheses of 4-[1-(2-deoxy-β-D-ribofuranosyl)]-derivatives of 2-substituted-5-fluoroaniline: "cytosine replacement" analogs of deoxycytidine for evaluation as anticancer and antihuman immunodeficiency virus (anti-HIV) agents , 2000 .

[12]  J. Balzarini,et al.  Synthesis and NMR conformational studies of stable analogues of 2-deoxy-α-D-ribose-1-phosphate , 1998 .

[13]  I. Stratford,et al.  Platelet-derived endothelial cell growth factor thymidine phosphorylase in tumour growth and response to therapy. , 1997, British Journal of Cancer.

[14]  P. Herdewijn,et al.  Synthesis of homo-N-nucleosides, a series of C1' branched-chain nucleosides , 1996 .

[15]  J. Witte,et al.  C-Glycosylphosphonyl Analogs of 5-Phosphorylribose 1-α-Diphosphate: II. The “2-Deoxy” Analog , 1996 .

[16]  R. Southgate,et al.  Synthesis of derivatives of muramic acid and C-1 homologated α-D-glucose as potential inhibitors of bacterial transglycosylase , 1995 .

[17]  J. Vederas,et al.  Synthesis of a C-phosphonate disaccharide as a potential inhibitor of peptidoglycan polymerization by transglycosylase , 1993 .

[18]  D. Liotta,et al.  Synthesis of C-arabinofuranosyl compounds. Phosphonate and carboxylate isosteres of d-arabinose 1,5-bisphosphate , 1987 .

[19]  R. McClard.  A facile route to methylenephosphonate sugars substituted at the anomeric carbon , 1983 .

[20]  J. G. Moffatt,et al.  A new stable Wittig reagent suitable for the synthesis of α,β-unsaturated phosphonates , 1968 .