Progress in the studies on tryptanthrin, an alkaloid of history
暂无分享,去创建一个
[1] Youngjoo Kwon,et al. Synthesis of benzo-annulated tryptanthrins and their biological properties. , 2012, Bioorganic & medicinal chemistry.
[2] P. Grundt,et al. The Chemistry of Tryptanthrin and Its Derivatives , 2012 .
[3] A. I. Kalinovskii,et al. Synthesis of tryptanthrin (couroupitine) derivatives by reaction of substituted isatins with phosphoryl chloride , 2012, Russian Journal of Organic Chemistry.
[4] Atul Kumar,et al. β-Cyclodextrin Catalyzed Synthesis of Tryptanthrin in Water. , 2011 .
[5] Seung Ho Lee,et al. Synthesis and biological properties of benzo-annulated rutaecarpines. , 2010, Biological & pharmaceutical bulletin.
[6] R. Sinden,et al. Antimicrobial activity of tryptanthrins in Escherichia coli. , 2010, Journal of medicinal chemistry.
[7] R. King. Biotransformations in Drug Metabolism , 2010 .
[8] J. Bergman,et al. A New Approach to Methoxyisatins Leading to the Total Synthesis of Ophiuroidine and Other Hydroxytryptanthrins. , 2010 .
[9] J. Chern,et al. Cytotoxicity and reversal of multidrug resistance by tryptanthrin-derived indoloquinazolines , 2010, Acta Pharmacologica Sinica.
[10] N. Mak,et al. Modulatory Effects and Action Mechanisms of Tryptanthrin on Murine Myeloid Leukemia Cells , 2009, Cellular and Molecular Immunology.
[11] J. Chern,et al. Downregulation of GSTπ expression by tryptanthrin contributing to sensitization of doxorubicin-resistant MCF-7 cells through c-jun NH2-terminal kinase-mediated apoptosis , 2009, Anti-cancer drugs.
[12] A. de Meijere,et al. ortho-Lithiophenyl isocyanide: a versatile precursor for 3H-quinazolin-4-ones and 3H-quinazolin-4-thiones. , 2009, Organic letters.
[13] T. M. Potewar,et al. Synthesis of tryptanthrin and deoxyvasicinone by a regioselective lithiation-intramolecular electrophilic reaction approach , 2008 .
[14] M. Novak,et al. Scanning Tunneling Microscopy of 8-Fluoroindolo[2,1-b]quinazolin-6,12-dione (8-Fluorotryptanthrin) at the Graphite-Solution Interface : Fully Resolved Molecular Orbitals , 2008 .
[15] Chen-Wei Jao,et al. Isolation, structure elucidation, and synthesis of cytotoxic tryptanthrin analogues from Phaius mishmensis. , 2008, Journal of natural products.
[16] Seung Ho Lee,et al. One-pot synthesis of simple alkaloids: 2,3-polymethylene-4(3H)-quinazolinones, luotonin A, tryptanthrin, and rutaecarpine. , 2008, Chemical & pharmaceutical bulletin.
[17] J. Niedziela,et al. Scanning Tunneling Microscopy , 2008 .
[18] Yen-Hui Chen,et al. Tryptanthrin inhibits MDR1 and reverses doxorubicin resistance in breast cancer cells. , 2007, Biochemical and biophysical research communications.
[19] V. Denisenko,et al. Ophiuroidine, the first indolo[2,1-b]quinazoline alkaloid from the Caribbean brittle star Ophiocoma riisei , 2007 .
[20] B. Batanero,et al. Electrosynthesis of Tryptanthrin. , 2007 .
[21] M. Elsegood,et al. Radical reactions with 3H-quinazolin-4-ones: synthesis of deoxyvasicinone, mackinazolinone, luotonin A, rutaecarpine and tryptanthrin. , 2007, Organic & biomolecular chemistry.
[22] M. Hamburger,et al. HPLC based activity profiling for 5-lipoxygenase inhibitory activity in Isatis tinctoria leaf extracts. , 2005, Fitoterapia.
[23] A. Tai,et al. Inhibition of hepatocyte growth factor induction in human dermal fibroblasts by tryptanthrin. , 2005, Biological & pharmaceutical bulletin.
[24] R. Crabtree. Metal–Ligand Multiple Bonds , 2005 .
[25] W. Keller-Schierlein,et al. The structure of tryptanthrin , 2005, Experientia.
[26] D. Sullivan,et al. Evaluation of 4-Azaindolo(2,1-b)quinazoline-6,12-diones' Interaction with Hemin and Hemozoin: A Spectroscopic, X- ray Crystallographic and Molecular Modeling Study # , 2005 .
[27] M. Hamburger. Isatis tinctoria – From the rediscovery of an ancient medicinal plant towards a novel anti-inflammatory phytopharmaceutical , 2002, Phytochemistry Reviews.
[28] Terry D. Lee,et al. Female-to-male sex pheromones of low volatility in the Asian elephant,Elephas maximus , 1993, Journal of Chemical Ecology.
[29] W. Milhous,et al. Structure-activity relationship study of antimalarial indolo [2,1-b]quinazoline-6,12-diones (tryptanthrins). Three dimensional pharmacophore modeling and identification of new antimalarial candidates. , 2004, European journal of medicinal chemistry.
[30] K. Nishimura,et al. Isolation of a new potent cytotoxic pigment along with indigotin from the pathogenic basidiomycetous fungus Schizophyllum commune , 2004, Mycopathologia.
[31] J. Bergman,et al. Recent Developments in the Field of Quinazoline Chemistry , 2003 .
[32] Y. Jahng,et al. A facile synthesis of simple alkaloids—synthesis of 2,3-polymethylene-4(3H)-quinazolinones and related alkaloids , 2003 .
[33] Y. Jahng,et al. A SIMPLE SYNTHESIS OF TRYPTANTHRIN , 2003 .
[34] H. Simon,et al. Inhibitory activity of tryptanthrin on prostaglandin and leukotriene synthesis. , 2002, Planta medica.
[35] A. Venkateswarlu,et al. Novel indolo[2,1-b]quinazoline analogues as cytostatic agents: synthesis, biological evaluation and structure-activity relationship. , 2002, Bioorganic & medicinal chemistry letters.
[36] M. Hamburger,et al. Synthesis of d-tryptanthrin. , 2002, Die Pharmazie.
[37] D. Skanchy,et al. Analysis of stereoelectronic properties, mechanism of action and pharmacophore of synthetic indolo[2,1-b]quinazoline-6,12-dione derivatives in relation to antileishmanial activity using quantum chemical, cyclic voltammetry and 3-D-QSAR CATALYST procedures. , 2002, Bioorganic & medicinal chemistry.
[38] T. Shapiro,et al. Antitrypanosomal Activities of Tryptanthrins , 2002, Antimicrobial Agents and Chemotherapy.
[39] M. Hamburger,et al. Quantitative determination of the dual COX-2/5-LOX inhibitor tryptanthrin in Isatis tinctoria by ESI-LC-MS. , 2002, Planta medica.
[40] M. Micallef,et al. Prevention of azoxymethane-induced intestinal tumors by a crude ethyl acetate-extract and tryptanthrin extracted from Polygonum tinctorium Lour. , 2001, Anticancer research.
[41] H. Matsuda,et al. Chemical Constituents of Two Oriental Orchids,Calanthe discolor and C.Liukiuensis: Precursor Indole Glycoside of Tryptanthrin and Indirubin , 2001 .
[42] M. Ikeda,et al. Antibacterial action of tryptanthrin and kaempferol, isolated from the indigo plant (Polygonum tinctorium Lour.), against Helicobacter pylori-infected Mongolian gerbils , 2001, Journal of Gastroenterology.
[43] K. Kohno,et al. Tryptanthrin inhibits nitric oxide and prostaglandin E(2) synthesis by murine macrophages. , 2000, European journal of pharmacology.
[44] P. Renard,et al. Synthesis and cytotoxic and antitumor activity of benzo[b]pyrano[3, 2-h]acridin-7-one analogues of acronycine. , 2000, Journal of medicinal chemistry.
[45] S. Bhattacharya,et al. Indole and flavanoid constituents of Wrightia tinctoria, W. tomentosa and W. coccinea , 2000 .
[46] M. Kurimoto,et al. Isolation and Identification of Anti-Helicobacter pylori Compounds from Polygonum tinctorium Lour. , 1999 .
[47] L. Mitscher,et al. Tuberculosis: A search for novel therapy starting with natural products , 1998, Medicinal research reviews.
[48] H. Matsuda,et al. Novel indole S,O-bisdesmoside, calanthoside, the precursor glycoside of tryptanthrin, indirubin, and isatin, with increasing skin blood flow promoting effects, from two Calanthe species (Orchidaceae). , 1998, Chemical & pharmaceutical bulletin.
[49] H. Matile,et al. A comparison and analysis of several ways to promote haematin (haem) polymerisation and an assessment of its initiation in vitro. , 1998, Biochemical pharmacology.
[50] L. Mitscher,et al. A search for novel chemotherapy against tuberculosis amongst natural products , 1998 .
[51] V. Ambrogi,et al. Synthesis and antimicrobial activity of some new derivatives of 6,12-dihydroindolo[2,1-b]quinazolin-6,12-dione. , 1997, Farmaco.
[52] D. Schrenk,et al. Tryptanthrins: a novel class of agonists of the aryl hydrocarbon receptor. , 1997, Biochemical pharmacology.
[53] P. Hitchcock,et al. Isatin Chloride: A Phantom. Reactions of 2‐(2,2‐Dichloro‐2,3‐dihydro‐3‐ oxoindol‐1‐yl)‐3H‐indol‐3‐one. , 1997 .
[54] X. Wu,et al. Chemical constituents of Isatis indigotica. , 1997, Planta medica.
[55] T. Moskovkina. New Synthesis of 6,12-Dihydro-6,12-dioxoindolo[2,1-b]quinazoline (Tryptanthrine, Couropitine A) , 1997 .
[56] P. Pushpangadan,et al. Tryptanthrin from Wrightia tinctoria , 1996 .
[57] K. Seifert,et al. Insecticidal and Fungicidal Compounds from Isatis tinctoria , 1994, Zeitschrift fur Naturforschung. C, Journal of biosciences.
[58] T. Kondo,et al. Transition-Metal Complex-Catalyzed Reductive N-Heterocyclization: Synthesis of 4(3H)-Quinazolinone Derivatives from N-(2-Nitrobenzoyl) amides. , 1993 .
[59] V. Ambrogi,et al. Synthesis and antimicrobial activity of some new indolo[2,1-b]quinazolin-6(12H)ones. , 1993, Farmaco.
[60] S. Eguchi,et al. Short-step synthesis of rutecarpine and tryptanthrin via intramolecular aza-Wittig reaction , 1992 .
[61] A. Katritzky,et al. 2‐Chloro‐3H‐indol‐3‐one and its reactions with nucleophiles , 1989 .
[62] Li Qing-hua. The Chemical Constituents of Qing Dai , 1987 .
[63] H. Laatsch,et al. Isolierung des indigoiden Pigmentes Candidin aus Urin und Hämofiltrat von Urämikern , 1986 .
[64] J. Zou,et al. [Minor constituents of qing dai, a traditional Chinese medicine. I. Isolation, structural determination and synthesis of tryptanthrin and qingdainone]. , 1985, Yao xue xue bao = Acta pharmaceutica Sinica.
[65] V. Thaller,et al. 300 MHZ PROTON NMR SPECTRA OF INDOLO(2,1-B)QUINAZOLINE-6,12-DIONE, TRYPTANTHRINE, AND ITS 2- AND 8-CHLORO DERIVATIVES , 1980 .
[66] G. Honda,et al. Isolation of an antidermatophytic, tryptanthrin, from indigo plants, Polygonum tinctorium and Isatis tinctoria. , 1980, Planta medica.
[67] G. Honda,et al. Isolation of antifungal principle tryptanthrin, from Strobilanthes cusia O. Kuntze. , 1979, Planta medica.
[68] H. Junek,et al. Thermolyse von isatin mittels eines CO2,-lasers , 1978 .
[69] M. Ihara,et al. IMINOKETENE CYCLOADDITION. 2. TOTAL SYNTHESES OF ARBORINE, GLYCOSMININE, AND RUTECARPINE BY CONDENSATION OF IMINOKETENE WITH AMIDES , 1977 .
[70] P. G. Gassman,et al. A general method for the synthesis of isatins , 1977 .
[71] J. Bergman,et al. The structure of some indolic constituents in Couroupita Guaianensis Aubl. , 1977 .
[72] J. Grimshaw,et al. Condensation between 2-chloro-3H-indol-3-one and phenols , 1975 .
[73] W. Fedeli,et al. Crystal structure of tryptanthrin (indolo[2,1-b]quinazoline-6,12-dione) , 1974 .
[74] C. Duke,et al. Reactions of α-chloroisatin (2-Chloroindoleninone) with methanethiol and 1,2-ethanedithiol. , 1972 .
[75] M. Hooper,et al. Isatogens. Part VI. Synthesis of isatogens via tolan (diphenylacetylene) intermediates , 1969 .
[76] H. Redkey,et al. A new approach. , 1967, Rehabilitation record.
[77] R. Kikumoto,et al. The reactions of oxindoles and isatin with nitrobenzyl chlorides , 1966 .
[78] C. W. Bird. The structure of methylisatoid , 1963 .
[79] E. G. Sherry,et al. STRUCTURE DETERMINATION I , 1960 .
[80] A. Wagstaff,et al. The Structure of Isatin. I , 1936 .
[81] G. Heller. Zur Kenntnis des Indigos; cis‐Indigo , 1936 .
[82] H. Machemer. Die Autoxydation der Metallkomplexe des Indigos , 1930 .
[83] H. Henze,et al. CONDENSATION REACTIONS OF CYCLIC KETONES. I. THE ACTION OF ISATIN AND ISATIN ALPHA CHLORIDE UPON CERTAIN HYDANTOINS1 , 1924 .
[84] A. Hantzsch. Über die wirklichen und angeblichen Isomerien in der Isatin‐Reihe , 1921 .
[85] G. Heller. Über die Farbenerscheinung der alkalischen Isatinlösung , 1907 .
[86] W. Bloxam. CIII.—Our present knowledge of the chemistry of indigo , 1905 .
[87] A. Baeyer. Ueber die Einwirkung des Fünffachchlorphosphors auf Isatin und auf verwandte Substanzen , 1879 .